Zobrazeno 1 - 8
of 8
pro vyhledávání: '"K. D. Lovasz"'
Autor:
Chong Kt, J. C. Lynn, Paul K. Tomich, Karen Rene Romines, M.‐M. Horng, Lester A. Dolak, Howe Wj, Joel Morris, K. D. Lovasz, R. R. Hinshaw, K. D. Watenpaugh, M.N. Janakiraman
Publikováno v:
ChemInform. 27
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::a997a9a8ef0f2ff95323244b37781367
https://doi.org/10.1002/chin.199610192
https://doi.org/10.1002/chin.199610192
Autor:
K. D. Lovasz, Karen Rene Romines, Lester A. Dolak, J. M. Tustin, Gillian Phillips, Thomas M. Judge, R. A. Chrusciel, Strohbach Joseph Walter, Joel Morris, S. L. Vander Velde, G. P. Luke, Steve A. Mizsak, Ronald B. Gammill, John Tulinsky, W. Watt
Publikováno v:
ChemInform. 28
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::1622c65c8295675a1e8e15a38ee2e982
https://doi.org/10.1002/chin.199732114
https://doi.org/10.1002/chin.199732114
Autor:
K. D. Lovasz, Stephen A. Mizsak, Thomas M. Judge, Karen Rene Romines, Eric P. Seest, John Tulinsky, Jeanette Kay Morris, Ronald B. Gammill, Fusen Han
Publikováno v:
ChemInform. 30
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::5cf51a6f2356f55b6db8b7d9697d0ac1
https://doi.org/10.1002/chin.199930106
https://doi.org/10.1002/chin.199930106
Autor:
K. D. Lovasz, D. M. Gleave, Gary E. Zurenko, D. C. Rohrer, Manninen Peter Rudolph, John A. Tucker, D. A. Allwine, Steven J. Brickner, Ford Charles W
Publikováno v:
Bioorganicmedicinal chemistry letters. 8(10)
A series of conformationally restricted, [6,5,5] and [6,6,5] tricyclic fused oxazolidinones were synthesized and tested for antibacterial activity. Several compounds in the trans-[6,5,5] series demonstrated potent in vitro and in vivo activity. This
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a63cd76ca19684f30132594755dd09b2
https://pubmed.ncbi.nlm.nih.gov/9871741
https://pubmed.ncbi.nlm.nih.gov/9871741
Autor:
G.L Zipp, Lester A. Dolak, K. D. Watenpaugh, W.-Z Zhong, R. R. Hinshaw, C.W Johnson, David J. Anderson, L. S. Banitt, Johnson Paul D, Paul A. Aristoff, G.M Howard, M.N. Janakiraman, R J Reischer, Howe Wj, Harvey Irving Skulnick, Theresa M. Schwartz, L. N. Toth, K.R Wilkinson, Bob D. Rush, Karen Rene Romines, J. C. Lynn, Serena L. Cole, M. G. Williams, Eric P. Seest, Renee M. Zaya, Joel Morris, Chong Kt, Thomas J. Kakuk, R.J Dalga, K D Lovasz, Tomich Pk, M.‐M. Horng, P.L Possert, F.J Schwende
Publikováno v:
Journal of medicinal chemistry. 40(7)
Recently, cyclooctylpyranone derivatives with m-carboxamide substituents (e.g. 2c) were identified as potent, nonpeptidic HIV protease inhibitors, but these compounds lacked significant antiviral activity in cell culture. Substitution of a sulfonamid
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::edc7a130b4b392170feddcbcdbfa6abe
https://pubmed.ncbi.nlm.nih.gov/9089336
https://pubmed.ncbi.nlm.nih.gov/9089336
Autor:
Tomich Pk, Howe Wj, K D Lovasz, M.‐M. Horng, K. D. Watenpaugh, J. C. Lynn, Jeanette Kay Morris, Karen Rene Romines, Chong Kt, M.N. Janakiraman
Publikováno v:
Journal of medicinal chemistry. 38(22)
Recently, the novel cyclooctylpyranone HIV protease inhibitor 1 was identified in our labs, and an X-ray structure of this inhibitor complexed with HIV-2 protease was obtained. This crystal structure was used to develop two strategies for creating de
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8a7edbf2fae1fd29b53c403e81525e8a
https://pubmed.ncbi.nlm.nih.gov/7473573
https://pubmed.ncbi.nlm.nih.gov/7473573
Autor:
J. C. Lynn, Karen Rene Romines, K.D. Watenpaugh, Tomich Pk, M.‐M. Horng, A.M. Mulichak, K D Lovasz, J K Morris, Howe Wj, Barry C. Finzel
Publikováno v:
Journal of medicinal chemistry. 38(11)
A unique strategy for the enhancement of secondary binding of an inhibitor to an enzyme has been demonstrated in the design of new human immunodeficiency virus (HIV) protease inhibitors. When the planar benzene ring of a 4-hydroxycoumarin lead compou
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8aeb107b768f5904c01a75e29ec78769
https://pubmed.ncbi.nlm.nih.gov/7783120
https://pubmed.ncbi.nlm.nih.gov/7783120
Autor:
Ronald B. Gammill, and J. W. Strohbach, Thomas M. Judge, Lester A. Dolak, Gillian Phillips, Steve A. Mizsak, R. A. Chrusciel, J. M. Tustin, Joel Morris, S. L. Vander Velde, John Tulinsky, W. Watt, G. P. Luke, K. D. Lovasz, Karen Rene Romines
Publikováno v:
Journal of the American Chemical Society. 119:3627-3628
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::ce96eea487180a376ab991b30e8fa4c1
https://doi.org/10.1021/ja963434w
https://doi.org/10.1021/ja963434w