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pro vyhledávání: '"K. Cosmopolous"'
Autor:
K. Cosmopolous, J. Garnsey, Allison Berger, J. Donelan, Pete Smith, Mark Manfredi, T. Traore, M. Mihollen
Publikováno v:
Journal of Clinical Oncology. 29:8594-8594
8594 Background: MLN4924 is a novel, small molecule inhibitor of Nedd8-activating enzyme (NAE) currently in Phase I clinical trials. Conjugation of NEDD8 to cullin scaffold proteins is required for...