Zobrazeno 1 - 10
of 88
pro vyhledávání: '"Junya Shirai"'
Autor:
Shinsuke Suzuki, Teni Godai, Shin Kato, Atsushi Onodera, Kazuya Endo, Shizune Onuma, Yui Honjo, Junya Shirai, Masakatsu Numata, Yutaka Kumakiri, Shinichiro Suzuki, Yuji Yamamoto
Publikováno v:
Journal of the Anus, Rectum and Colon, Vol 6, Iss 1, Pp 72-76 (2022)
We describe our experience with robotic posterior rectopexy for a patient with full-thickness rectal prolapse. To our knowledge, this is the first report of such a case in the literature. A 94-year-old woman presented with a history of gradually wors
Externí odkaz:
https://doaj.org/article/0e91ea1e138641dea0c34e79431a4461
Autor:
Shinsuke Hatori, Tsutomu Sato, Munetaka Masuda, Shinnosuke Kawahara, Koji Numata, Yasushi Rino, Kazuyuki Tani, Norio Yukawa, Junya Shirai, Hiroshi Tamagawa
Publikováno v:
Nihon Gekakei Rengo Gakkaishi (Journal of Japanese College of Surgeons). 45:356-362
Autor:
Junya Shirai, Yoshiyuki Fukase, Keiko Koga, Ryoukichi Koyama, Hideyuki Nakagawa, Isaac Hoffman, Bi-Ching Sang, Mitsunori Kono, Toshitake Okui, Satoshi Yamamoto, Yasushi Fujitani, Masaharu Nakayama, Yoshihide Tomata, Robert J. Skene, Kazuko Yonemori, Atsuko Ochida, Masashi Yamasaki, Ayumu Sato
Publikováno v:
Bioorganic & Medicinal Chemistry. 26:721-736
Novel small molecules were synthesized and evaluated as retinoic acid receptor-related orphan receptor-gamma t (RORγt) inverse agonists for the treatment of inflammatory and autoimmune diseases. A hit compound, 1, was discovered by high-throughput s
Autor:
Junya Shirai, Yoshiyuki Fukase, Tetsuji Kawamoto, Mitsunori Kono, Tsuneo Oda, Mikio Shirasaki, Yasushi Fujitani, Hiroyuki Watanabe, Hideyuki Nakagawa, Keiko Uga, Michiko Tawada, Naohiro Taya, Akira Shibata, Takashi Imada, Yoshihide Tomata, Masashi Yamasaki, Tomoya Yukawa, Shoji Fukumoto, Hidekazu Tokuhara, Satoshi Yamamoto, Naoki Ishii, Atsuko Ochida, Yoshihiro Banno
Publikováno v:
Bioorganic & Medicinal Chemistry. 26:470-482
A series of tetrahydroisoquinoline derivatives were designed, synthesized, and evaluated for their potential as novel orally efficacious retinoic acid receptor-related orphan receptor-gamma t (RORγt) inverse agonists for the treatment of Th17-driven
Autor:
Junya Shirai, Masato Yoshida, Ayumu Sato, Nobuki Sakauchi, Haruhiko Kuno, Reiko Saikawa, Hideki Furukawa
Publikováno v:
European Journal of Medicinal Chemistry. 139:114-127
A series of phenoxyethylamine derivatives was designed and synthesized to discover potent and selective human α 1D adrenoceptor (α 1D adrenergic receptor; α 1D –AR) antagonists. Compound 7 was taken from our internal compound collection as an at
Autor:
Soji Ozawa, Akio Kasahara, Takanobu Yamada, Yuji Yamamoto, Itaru Endo, Munetaka Masuda, Katsuya Yoneyama, Masahiko Watanabe, Junya Shirai, Yasushi Rino
Publikováno v:
International Surgery. 101:570-576
Comprehensive surveys on perioperative care in Japan, including that in community or private hospitals, have not been reported, and current trends remain unclear. The present survey was designed to investigate current routines for perioperative care
Autor:
Masashi Yamasaki, Ayumu Sato, Tsuneo Oda, Gyorgy Snell, Junya Shirai, Yoshiyuki Fukase, Bi-Ching Sang, Keiko Uga, Atsuko Ochida, Yusuke Sasaki, Hideyuki Nakagawa, Akira Shibata, Satoshi Yamamoto, Naoki Ishii, Yoshihide Tomata, Shoji Fukumoto, Mikio Shirasaki, Isaac Hoffman, Mitsunori Kono, Robert J. Skene, Yumi N. Imai
Publikováno v:
ChemMedChem. 14(22)
Retinoic-acid-related orphan receptor γt (RORγt) inverse agonists could be used for the treatment of autoimmune diseases. Previously, we reported a novel quinazolinedione 1 a with a flexible linear linker as a novel RORγt inverse agonist. A U-shap
Autor:
Naohiro Taya, Chien-Hung Chen, Tsuneo Oda, Bi-Ching Sang, Tomoya Yukawa, Takayuki Sato, Yoshi Nara, Noriko Uchiyama, Zenyu Shiokawa, Terufumi Takagi, Satoshi Yamamoto, Ayumu Sato, Ryokichi Koyama, Nobuyuki Negoro, Gyorgy Snell, Junya Shirai, Ryosuke Katsuyama, Takashi Imada, Yoshihiro Banno, Isaac Hoffman, Tetsuji Kawamoto, Mitsunori Kono, Robert J. Skene
Publikováno v:
Journal of medicinal chemistry. 62(3)
Retinoic acid receptor-related orphan receptor γt (RORγt) agonists are expected to provide a novel class of immune-activating anticancer drugs via activation of Th17 cells and Tc17 cells. Herein, we describe a novel structure-based functionality sw
Autor:
Hironobu Maezaki, Maki Miyamoto, Miki Hara, Norio Tada, Hisashi Fujita, Junya Shirai, Katsuhiko Miwa, Nobuki Sakauchi, Haruhiko Kuno, Nagako Kameoka, Ayumu Sato, Hideki Furukawa
Publikováno v:
Tetrahedron. 72:6334-6339
5-Chloro-1-(5-chloro-2-(methylsulfonyl)benzyl)-2-imino-1,2-dihydropyridine-3-carboxamide hydrochloride (TAK-259) is a novel, selective, and orally active α1D adrenoceptor antagonist with anti-urinary frequency effect. A metabolite (2) of TAK-259 was
Autor:
Yoshihiro Suzuki, Shinsuke Hatori, Munetaka Masuda, Katsuya Yoneyama, Junya Shirai, Mariko Kamiya
Publikováno v:
Nihon Rinsho Geka Gakkai Zasshi (Journal of Japan Surgical Association). 77:1255-1260