Zobrazeno 1 - 10
of 40
pro vyhledávání: '"Jukka Sallinen"'
Autor:
Mohammed Shahid, Juha O. Rinne, Mika Scheinin, Jere Virta, Päivi Marjamäki, Olof Solin, Eveliina Arponen, Jukka Sallinen, Katja Kuokkanen, Juha Rouru
Publikováno v:
EJNMMI Research, Vol 10, Iss 1, Pp 1-9 (2020)
Abstract Background Availability of the α2C-adrenoceptor (α2C-AR) positron emission tomography (PET) tracer, [11C]ORM-13070, and the α2C-AR antagonist ORM-12741 allows probing of the roles of this G-protein coupled receptor subtype in brain functi
Externí odkaz:
https://doaj.org/article/f2ab19aa502748819823cd5dec03a851
Autor:
Jere Virta, Juha O. Rinne, Jukka Sallinen, Olof Solin, Katja Kuokkanen, Juha Rouru, Päivi Marjamäki, Mika Scheinin, Eveliina Arponen, Mohammed Shahid
Publikováno v:
EJNMMI Research
EJNMMI Research, Vol 10, Iss 1, Pp 1-9 (2020)
EJNMMI Research, Vol 10, Iss 1, Pp 1-9 (2020)
Background Availability of the α2C-adrenoceptor (α2C-AR) positron emission tomography (PET) tracer, [11C]ORM-13070, and the α2C-AR antagonist ORM-12741 allows probing of the roles of this G-protein coupled receptor subtype in brain function, both
Autor:
Mohammed Shahid, Juha O. Rinne, Mika Scheinin, Jere Virta, Päivi Marjamäki, Olof Solin, Eveliina Arponen, Jukka Sallinen, Katja Kuokkanen, Juha Rouru
Background Availability of the α2C -adrenoceptor (α2C-AR) positron emission tomography (PET) tracer, 11C -ORM-13070, and the selective α2C-AR antagonist ORM-12741 allows probing of the roles of this G-protein coupled receptor subtype in brain func
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::a6ff85f0f659d131d0cf66fd4f68a17c
https://doi.org/10.21203/rs.3.rs-45308/v1
https://doi.org/10.21203/rs.3.rs-45308/v1
Autor:
Edilio Borroni, Christer Halldin, Mohammed Shahid, Jussi Lehto, Mika Scheinin, Lars Farde, Sarah Grimwood, Sjoerd J. Finnema, Jukka Sallinen, Benny Bang-Andersen, Erik H. F. Wong
Publikováno v:
Psychopharmacology
Rationale This review attempts to summarize the current status in relation to the use of positron emission tomography (PET) imaging in the assessment of synaptic concentrations of endogenous mediators in the living brain. Objectives Although PET radi
Autor:
Vesa Oikonen, Pauliina Luoto, Jussi Lehto, Mika Scheinin, Juha Rouru, Sjoerd J. Finnema, Juha O. Rinne, Christer Halldin, Jukka Sallinen, Tarja Naukkarinen, Eveliina Arponen, Harry Scheinin, Jarkko Johansson, M. Hirvonen, Jukka Kemppainen, Lauri Vuorilehto
Publikováno v:
Synapse. 69:172-181
This study explored the use of the α2C-adrenoceptor PET tracer [11C]ORM-13070 to monitor α2C-AR occupancy in the human brain. The subtype-nonselective α2-AR antagonist atipamezole was administered to eight healthy volunteer subjects to determine i
Autor:
Tarja Malm, Asla Pitkänen, Mikko Hiltunen, Teemu Natunen, Joana I. Soares, Xavier Ekolle Ndode-Ekane, Pedro Andrade, Jukka Sallinen, Jari Nissinen, Katja M. Kanninen, Olena Shatillo
Publikováno v:
Epilepsy research. 136
Treatment of TBI remains a major unmet medical need, with 2.5 million new cases of traumatic brain injury (TBI) each year in Europe and 1.5 million in the USA. This single-center proof-of-concept preclinical study tested the hypothesis that pharmacol
Autor:
Juha M. Peltonen, Anne Roivainen, Juha Rouru, Sami Suilamo, Jukka Herttuainen, Iina Volanen, Kirsi A. Virtanen, Juha O. Rinne, Marita Kailajärvi, Jukka Sallinen, Vesa Oikonen, Semi Helin, Johanna Hietamäki, Pauliina Luoto, Jere Virta, Aila Holopainen, Mika Scheinin, Eveliina Arponen
Publikováno v:
European Journal of Nuclear Medicine and Molecular Imaging. 41:1947-1956
Purpose 11C-labelled 1-[(S)-1-(2,3-dihydrobenzo[1,2]dioxin-2-yl)methyl]-4-(3-methoxy-methylpyridin-2-yl)-piperazine (11C-ORM-13070) is a novel PET tracer for imaging of α2C-adrenoceptors in the human brain. Brain α2C-adrenoceptors may be therapeuti
Autor:
Olof Solin, Merja Haaparanta-Solin, Kjell Någren, Eliisa Löyttyniemi, Tove J. Grönroos, Patrik Holm, Jukka Sallinen, Semi Helin, Päivi Marjamäki, Mika Scheinin, Eveliina Arponen
Publikováno v:
Journal of Nuclear Medicine. 55:1171-1177
We report the development of a PET tracer for α2C adrenoceptor imaging and its preliminary preclinical evaluation. α2C adrenoceptors in the human brain may be involved in various neuropsychiatric disorders, such as depression, schizophrenia, and ne
Autor:
Jelena Mijatovic, Petteri Piepponen, Katja Kuokkanen, Heikki Tanila, Johanna Holappa, Jukka Sallinen, Raimo Virtanen, Jouni Sirviö, Hugh Chapman, Antti Haapalinna, Ari Koivisto, Jyrki Lehtimäki
Publikováno v:
Basic & Clinical Pharmacology & Toxicology. 113:239-249
The α2-adrenoceptors (ARs) are important modulators of a wide array of physiological responses. As only a few selective compounds for the three α2-AR subtypes (α2A , α2B and α2C ) have been available, the pharmacological profile of a new α2C-se
Autor:
Olof Solin, Merja Haaparanta-Solin, Päivi Marjamäki, Tove J. Grönroos, Jukka Sallinen, Semi Helin, Eveliina Arponen, Kjell Någren, Kimmo Ingman
Publikováno v:
Molecular Imaging and Biology. 12:500-1636