Zobrazeno 1 - 10
of 14
pro vyhledávání: '"Jonathan G. Pabalan"'
Autor:
Brent A. Rupnow, Tai W. Wong, R. Michael Lawrence, Malavi T. Madireddi, Jun Zhu, Wen-Pin Yang, Benjamin J. Henley, Joseph Fargnoli, Rolf-Peter Ryseck, Xinyu Wang, Jonathan G. Pabalan, Urvashi V. Roongta
PDF file - 70K
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3a5f19996f7b7be9db5b7fb7f371b35a
https://doi.org/10.1158/1541-7786.22518582
https://doi.org/10.1158/1541-7786.22518582
Autor:
Brent A. Rupnow, Tai W. Wong, R. Michael Lawrence, Malavi T. Madireddi, Jun Zhu, Wen-Pin Yang, Benjamin J. Henley, Joseph Fargnoli, Rolf-Peter Ryseck, Xinyu Wang, Jonathan G. Pabalan, Urvashi V. Roongta
PDF file - 71K
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::26056af1bb8f6abaaf3538a0f9578a1c
https://doi.org/10.1158/1541-7786.22518573
https://doi.org/10.1158/1541-7786.22518573
Autor:
Brent A. Rupnow, Tai W. Wong, R. Michael Lawrence, Malavi T. Madireddi, Jun Zhu, Wen-Pin Yang, Benjamin J. Henley, Joseph Fargnoli, Rolf-Peter Ryseck, Xinyu Wang, Jonathan G. Pabalan, Urvashi V. Roongta
PDF file - 70K
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9ec24b96c95c22de17c639d58869cf8e
https://doi.org/10.1158/1541-7786.22518576.v1
https://doi.org/10.1158/1541-7786.22518576.v1
Autor:
Brent A. Rupnow, Tai W. Wong, R. Michael Lawrence, Malavi T. Madireddi, Jun Zhu, Wen-Pin Yang, Benjamin J. Henley, Joseph Fargnoli, Rolf-Peter Ryseck, Xinyu Wang, Jonathan G. Pabalan, Urvashi V. Roongta
Emerging literature suggests that metabolic pathways play an important role in the maintenance and progression of human cancers. In particular, recent studies have implicated lipid biosynthesis and desaturation as a requirement for tumor cell surviva
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1744961da814489eb070a9b55c9e7207
https://doi.org/10.1158/1541-7786.c.6542004
https://doi.org/10.1158/1541-7786.c.6542004
Autor:
Brent A. Rupnow, Tai W. Wong, R. Michael Lawrence, Malavi T. Madireddi, Jun Zhu, Wen-Pin Yang, Benjamin J. Henley, Joseph Fargnoli, Rolf-Peter Ryseck, Xinyu Wang, Jonathan G. Pabalan, Urvashi V. Roongta
PDF file - 39K
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8112b61c9fece78abeaaa07d5a8f9ff9
https://doi.org/10.1158/1541-7786.22518579.v1
https://doi.org/10.1158/1541-7786.22518579.v1
Autor:
Emily Luk, Karen E. Parrish, Yue-Zhong Shu, Anwar Murtaza, Yongnian Sun, Jinwen Huang, Robert M. Borzilleri, Paul Stetsko, Mary Ellen Cvijic, Jonathan G. Pabalan, Lihong Cheng, Zheng Yang, Jesse Swanson, James R. Burke, Tatyana Zvyaga, James Smalley, Karen A. Augustine
Publikováno v:
Biopharmaceutics & Drug Disposition. 42:137-149
Transforming growth factor beta (TGF-β) is a pleiotropic cytokine that has a wide array of biological effects. For decades, tumor biology implicated TGF-β as an attractive therapeutic target due to its immunosuppressive effects. Toward this end, mu
Autor:
Steven P. Seitz, John T. Hunt, Kelly L. Covello, Lisa Elkin, Gregory D. Vite, Yuval Blat, Jay A. Markwalder, Jonathan G. Pabalan, Maria Jure-Kunkel
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 27:582-585
The discovery of a series of structurally-novel biaryl urea IDO inhibitors is described. Optimization of a micromolar hit through iterative cycles of synthesis and screening in an assay measuring IDO-mediated intracellular conversion of tryptophan to
Autor:
Saini Jasmine, Steven G. Nadler, Ashok Dongre, Aiqing He, Dmitry V. Ostanin, Clarence K. Zhang, Vishal Patel, Manling Ma-Edmonds, Jonathan G. Pabalan, Laurence Menard, Sherif Daouti, Sunil Kuppasani, Julie Carman, Li Fan, Omar Jabado, Matthew Loya, John R. Thompson, Ji Gao, Amy Truong, Urvashi V. Roongta
Publikováno v:
Gastroenterology. 156:S-873
Autor:
R. Michael Lawrence, Brent A. Rupnow, Malavi Madireddi, Xinyu Wang, Jonathan G. Pabalan, Tai W. Wong, Wen-Pin Yang, Benjamin J. Henley, Rolf-Peter Ryseck, Urvashi V. Roongta, Joseph Fargnoli, Jun Zhu
Publikováno v:
Molecular Cancer Research. 9:1551-1561
Emerging literature suggests that metabolic pathways play an important role in the maintenance and progression of human cancers. In particular, recent studies have implicated lipid biosynthesis and desaturation as a requirement for tumor cell surviva
Autor:
Joseph Fargnoli, Jonathan Lippy, Ashok V. Purandare, John T. Hunt, Libing Chen, Brian E. Fink, John S. Tokarski, Andrew Nation, Soong-Hoon Kim, Yufen Zhao, William R. Foster, Ashvinikumar V. Gavai, Tai W. Wong, Gregory D. Vite, Urvashi V. Roongta, Aberra Fura, Brent A. Rupnow, Jonathan G. Pabalan, Benjamin J. Henley, Christine M. Tarby, Mary T. Obermeier, Chiang Yu, Liqi He, Paul A. Elzinga
Publikováno v:
Cancer Research. 75:5417-5417
CK2 is a highly conserved, and constitutively active family of serine/threonine kinases abnormally elevated in a wide variety of cancers and linked to poor prognosis and disease progression. The enzymes form as hetero-tetrameric complexes comprised o