Zobrazeno 1 - 10
of 110
pro vyhledávání: '"Joji Yui"'
Autor:
Tomoteru Yamasaki, Masayuki Fujinaga, Joji Yui, Hidekatsu Wakizaka, Tomoyuki Ohya, Nobuki Nengaki, Masanao Ogawa, Yoko Ikoma, Akiko Hatori, Lin Xie, Kazunori Kawamura, Ming-Rong Zhang
Publikováno v:
PLoS ONE, Vol 10, Iss 6, p e0130006 (2015)
Metabotropic glutamate receptor subtype 1 (mGluR1) is a crucial target in the development of new medications to treat central nervous system (CNS) disorders. Recently, we developed N-[4-[6-(isopropylamino)pyrimidin-4-yl]-1,3-thiazol-2-yl]-4-[11C]meth
Externí odkaz:
https://doaj.org/article/f3cefafae69444f3913d026fcb7a7b84
Autor:
Akiko Hatori, Joji Yui, Lin Xie, Tomoteru Yamasaki, Katsushi Kumata, Masayuki Fujinaga, Hidekatsu Wakizaka, Masanao Ogawa, Nobuki Nengaki, Kazunori Kawamura, Ming-Rong Zhang
Publikováno v:
PLoS ONE, Vol 9, Iss 1, p e86625 (2014)
Liver damage induced by drug toxicity is an important concern for both medical doctors and patients. The aim of this study was to noninvasively visualize acute liver damage using positron emission tomography (PET) with N-benzyl-N-methyl-2-[7,8-dihydr
Externí odkaz:
https://doaj.org/article/36f3c0d3f0cd49eca570c947608ab53f
Autor:
Akiko Hatori, Joji Yui, Tomoteru Yamasaki, Lin Xie, Katsushi Kumata, Masayuki Fujinaga, Yuichiro Yoshida, Masanao Ogawa, Nobuki Nengaki, Kazunori Kawamura, Toshimitsu Fukumura, Ming-Rong Zhang
Publikováno v:
PLoS ONE, Vol 7, Iss 9, p e45065 (2012)
PURPOSE: The translocator protein (18 kDa) (TSPO) is highly expressed on the bronchial and bronchiole epithelium, submucosal glands in intrapulmonary bronchi, pneumocytes and alveolar macrophages in human lung. This study aimed to perform positron em
Externí odkaz:
https://doaj.org/article/e52b38ac317940859f49cb580984f3f7
Autor:
Hideki, Ishii, Tomoteru, Yamasaki, Joji, Yui, Yiding, Zhang, Masayuki, Hanyu, Masanao, Ogawa, Nobuki, Nengaki, Atsushi B, Tsuji, Yuya, Terashima, Kouji, Matsushima, Ming-Rong, Zhang
Publikováno v:
Bioorganicmedicinal chemistry letters. 30(6)
[Thiocarbonyl
Autor:
Masayuki Fujinaga, Wakana Mori, Katsushi Kumata, Joji Yui, Yiding Zhang, Masanao Ogawa, Yusuke Kurihara, Ming-Rong Zhang
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 27:4521-4524
The purpose of this study was to synthesize a new positron emission tomography radiotracer, N-(4-tertiarybutylphenyl)-4-(3-chloropyridin-2-yl)tetrahydropyrazine-1(2H)-[11C]carboxamide ([11C]BCTC, [11C]1), and assess its in vivo binding to the transie
Autor:
Akiko Hatori, Masayuki Fujinaga, Yufei Ma, Tomoteru Yamasaki, Lin Xie, Yiding Zhang, Katsushi Kumata, Nobuki Nengaki, Joji Yui, Ming-Rong Zhang, Hui Wang
Publikováno v:
Bioorganic & Medicinal Chemistry. 25:1014-1021
Brain metabotropic glutamate receptor 2 (mGluR2) has been proposed as a therapeutic target for the treatment of schizophrenia-like symptoms arising from increased glutamate transmission in the forebrain. However, there does not exist a reliable tool
Autor:
Kazunori Kawamura, Nobuki Nengaki, Yusuke Kurihara, Tomoteru Yamasaki, Katsushi Kumata, Masayuki Fujinaga, Yoko Shimoda, Ming-Rong Zhang, Akiko Hatori, Lin Xie, Masanao Ogawa, Joji Yui, Yiding Zhang, Hidekatsu Wakizaka
Publikováno v:
Nuclear Medicine and Biology. 45:1-7
Introduction A positron emission tomography (PET) probe with ultra-high specific radioactivity (SA) enables measuring high receptor specific binding in brain regions by avoiding mass effect of the PET probe itself. It has been reported that PET probe
Autor:
Lu Wang, Yiding Zhang, Benjamin H. Rotstein, Akiko Hatori, Steven H. Liang, Yuji Nagai, Masayuki Fujinaga, Wakana Mori, Yoko Shimoda, Lin Xie, Makoto Higuchi, Joji Yui, Takafumi Minamimoto, Ming-Rong Zhang, Longle Ma, Ran Cheng, Tomoteru Yamasaki, Neil Vasdev
Publikováno v:
Theranostics
Monoacylglycerol lipase (MAGL) is a 33 kDa member of the serine hydrolase superfamily that preferentially degrades 2-arachidonoylglycerol (2-AG) to arachidonic acid in the endocannabinoid system. Inhibition of MAGL is not only of interest for probing
Autor:
Yiding Zhang, Hideki Ishii, Lin Xie, Ming-Rong Zhang, Akiko Hatori, Nobuki Nengaki, Yusuke Kurihara, Katsushi Kumata, Masayuki Fujinaga, Yoko Shimoda, Joji Yui, Tomoteru Yamasaki
Publikováno v:
Bioorganic & medicinal chemistry. 24(4):627-634
To visualize fatty acid amide hydrolase (FAAH) in brain in vivo, we developed a novel positron emission tomography (PET) ligand N-(3,4-dimethylisoxazol-5-yl)piperazine-4-[4-(2-fluoro-4-[(11)C]methylphenyl)thiazol-2-yl]-1-carboxamide ([(11)C]DFMC, [(1
Autor:
Tomoteru Yamasaki, Lin Xie, Masayuki Fujinaga, Kazunori Kawamura, Ming-Rong Zhang, Yoko Shimoda, Kenji Furutsuka, Akiko Hatori, Hiroki Hashimoto, Nobuki Nengaki, Makoto Takei, Hidekatsu Wakizaka, Katsushi Kumata, Satoshi Shiomi, Joji Yui
Publikováno v:
The Journal of neuroscience : the official journal of the Society for Neuroscience. 36(2):375-384
Parkinson's disease (PD) is a prevalent degenerative disorder affecting the CNS that is primarily characterized by resting tremor and movement deficits. Group I metabotropic glutamate receptor subtypes 1 and 5 (mGluR1 and mGluR5, respectively) are im