Zobrazeno 1 - 10
of 48
pro vyhledávání: '"John Sensintaffar"'
Autor:
James D Joseph, Beatrice Darimont, Wei Zhou, Alfonso Arrazate, Amy Young, Ellen Ingalla, Kimberly Walter, Robert A Blake, Jim Nonomiya, Zhengyu Guan, Lorna Kategaya, Steven P Govek, Andiliy G Lai, Mehmet Kahraman, Dan Brigham, John Sensintaffar, Nhin Lu, Gang Shao, Jing Qian, Kate Grillot, Michael Moon, Rene Prudente, Eric Bischoff, Kyoung-Jin Lee, Celine Bonnefous, Karensa L Douglas, Jackaline D Julien, Johnny Y Nagasawa, Anna Aparicio, Josh Kaufman, Benjamin Haley, Jennifer M Giltnane, Ingrid E Wertz, Mark R Lackner, Michelle A Nannini, Deepak Sampath, Luis Schwarz, Henry Charles Manning, Mohammed Noor Tantawy, Carlos L Arteaga, Richard A Heyman, Peter J Rix, Lori Friedman, Nicholas D Smith, Ciara Metcalfe, Jeffrey H Hager
Publikováno v:
eLife, Vol 8 (2019)
Externí odkaz:
https://doaj.org/article/d1935c5b03e6433ea06acf491e7dc6f2
Autor:
James D Joseph, Beatrice Darimont, Wei Zhou, Alfonso Arrazate, Amy Young, Ellen Ingalla, Kimberly Walter, Robert A Blake, Jim Nonomiya, Zhengyu Guan, Lorna Kategaya, Steven P Govek, Andiliy G Lai, Mehmet Kahraman, Dan Brigham, John Sensintaffar, Nhin Lu, Gang Shao, Jing Qian, Kate Grillot, Michael Moon, Rene Prudente, Eric Bischoff, Kyoung-Jin Lee, Celine Bonnefous, Karensa L Douglas, Jackaline D Julien, Johnny Y Nagasawa, Anna Aparicio, Josh Kaufman, Benjamin Haley, Jennifer M Giltnane, Ingrid E Wertz, Mark R Lackner, Michelle A Nannini, Deepak Sampath, Luis Schwarz, Henry Charles Manning, Mohammed Noor Tantawy, Carlos L Arteaga, Richard A Heyman, Peter J Rix, Lori Friedman, Nicholas D Smith, Ciara Metcalfe, Jeffrey H Hager
Publikováno v:
eLife, Vol 5 (2016)
ER-targeted therapeutics provide valuable treatment options for patients with ER+ breast cancer, however, current relapse and mortality rates emphasize the need for improved therapeutic strategies. The recent discovery of prevalent ESR1 mutations in
Externí odkaz:
https://doaj.org/article/e0d8a246d19143f9bd877f0b6caa0659
Autor:
Jeffrey H. Hager, Beatrice Darimont, Isan Chen, Edna Chow Maneval, Michael Moon, Dan Brigham, Gang Shao, John Sensintaffar, Jing Qian, Nhin Lu, James D. Joseph
PDF file - 183K, Supplementary Table S1. 1st and 2nd generation AR antagonist activity on F876L-AR. Supplementary Table S2. LNCaP/SRF876L Xenograft Pharmacokinetics Supplementary Table S3. AR nucleotide changes monitored by BEAMing assay Supplemen
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::60f2e79c45774b04e048841baece0c01
https://doi.org/10.1158/2159-8290.22530719
https://doi.org/10.1158/2159-8290.22530719
Autor:
Michael R. Savona, Stephen W. Fesik, Edward T. Olejniczak, Gregory D. Ayers, Leah J. Hogdal, John Sensintaffar, Stephen A. Strickland, Kelli L. Boyd, Londa Fuller, Maria Pia Arrate, Agnieszka E. Gorska, Taekyu Lee, Melissa A. Fischer, Haley E. Ramsey
Supplementary figures and table
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::75a65705db4645e57301fe7bf49f1478
https://doi.org/10.1158/2159-8290.22534147.v1
https://doi.org/10.1158/2159-8290.22534147.v1
Autor:
Jeffrey H. Hager, Beatrice Darimont, Isan Chen, Edna Chow Maneval, Michael Moon, Dan Brigham, Gang Shao, John Sensintaffar, Jing Qian, Nhin Lu, James D. Joseph
PDF file - 401K, Supplementary Figure S1. Parental and 2nd generation anti-androgen resistant cell line proliferation. Supplementary Figure S2. AR levels in parental and 2nd generation anti-androgen resistant cell lines. Supplementary Figure S3. AR l
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1ba5f8f0deb91bd874dc4fd74d291586
https://doi.org/10.1158/2159-8290.22530722.v1
https://doi.org/10.1158/2159-8290.22530722.v1
Autor:
Michael R. Savona, Stephen W. Fesik, Edward T. Olejniczak, Gregory D. Ayers, Leah J. Hogdal, John Sensintaffar, Stephen A. Strickland, Kelli L. Boyd, Londa Fuller, Maria Pia Arrate, Agnieszka E. Gorska, Taekyu Lee, Melissa A. Fischer, Haley E. Ramsey
Suppression of apoptosis by expression of antiapoptotic BCL2 family members is a hallmark of acute myeloblastic leukemia (AML). Induced myeloid leukemia cell differentiation protein (MCL1), an antiapoptotic BCL2 family member, is commonly upregulated
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7f6e8f2266d8ea8d3407f3dac4b6921b
https://doi.org/10.1158/2159-8290.c.6547384
https://doi.org/10.1158/2159-8290.c.6547384
Autor:
Jeffrey H. Hager, Charles L. Sawyers, Michael E. Jung, Richard A. Heyman, Peter J. Rix, Ouathek Ouerfelli, Nian Wu, Elisa De Stanchina, Nicholas D. Smith, Mark Klang, Peter Smith-Jones, Howard I. Scher, Beatrice Darimont, Celine Bonnefous, Mark R. Herbert, Teresa Wasielewska, John Sensintaffar, Chunyan Cao, Guangbin Yang, Hong Zhao, Jing Qian, Gang Shao, Vivek Arora, Steven Dorow, Anna Aparicio, Ling Cai, Eric D. Bischoff, Kate Grillot, Yu Chen, Anna Dilhas, Samedy Ouk, Chris Tran, James D. Joseph, John Wongvipat, Nicola J. Clegg
PDF file - 185K
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ad0f57c8b6ecb96bc53146deeb63d113
https://doi.org/10.1158/0008-5472.22393724.v1
https://doi.org/10.1158/0008-5472.22393724.v1
Autor:
Jeffrey H. Hager, Charles L. Sawyers, Michael E. Jung, Richard A. Heyman, Peter J. Rix, Ouathek Ouerfelli, Nian Wu, Elisa De Stanchina, Nicholas D. Smith, Mark Klang, Peter Smith-Jones, Howard I. Scher, Beatrice Darimont, Celine Bonnefous, Mark R. Herbert, Teresa Wasielewska, John Sensintaffar, Chunyan Cao, Guangbin Yang, Hong Zhao, Jing Qian, Gang Shao, Vivek Arora, Steven Dorow, Anna Aparicio, Ling Cai, Eric D. Bischoff, Kate Grillot, Yu Chen, Anna Dilhas, Samedy Ouk, Chris Tran, James D. Joseph, John Wongvipat, Nicola J. Clegg
PDF file - 181K
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2a9d43c3d094fe2a4e4d08a204389238
https://doi.org/10.1158/0008-5472.22393718
https://doi.org/10.1158/0008-5472.22393718
Autor:
Jeffrey H. Hager, Charles L. Sawyers, Michael E. Jung, Richard A. Heyman, Peter J. Rix, Ouathek Ouerfelli, Nian Wu, Elisa De Stanchina, Nicholas D. Smith, Mark Klang, Peter Smith-Jones, Howard I. Scher, Beatrice Darimont, Celine Bonnefous, Mark R. Herbert, Teresa Wasielewska, John Sensintaffar, Chunyan Cao, Guangbin Yang, Hong Zhao, Jing Qian, Gang Shao, Vivek Arora, Steven Dorow, Anna Aparicio, Ling Cai, Eric D. Bischoff, Kate Grillot, Yu Chen, Anna Dilhas, Samedy Ouk, Chris Tran, James D. Joseph, John Wongvipat, Nicola J. Clegg
PDF file - 241K
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b95de4c884e1f7ad8e36b2ca14c471b7
https://doi.org/10.1158/0008-5472.22393730.v1
https://doi.org/10.1158/0008-5472.22393730.v1
Autor:
Jeffrey H. Hager, Charles L. Sawyers, Michael E. Jung, Richard A. Heyman, Peter J. Rix, Ouathek Ouerfelli, Nian Wu, Elisa De Stanchina, Nicholas D. Smith, Mark Klang, Peter Smith-Jones, Howard I. Scher, Beatrice Darimont, Celine Bonnefous, Mark R. Herbert, Teresa Wasielewska, John Sensintaffar, Chunyan Cao, Guangbin Yang, Hong Zhao, Jing Qian, Gang Shao, Vivek Arora, Steven Dorow, Anna Aparicio, Ling Cai, Eric D. Bischoff, Kate Grillot, Yu Chen, Anna Dilhas, Samedy Ouk, Chris Tran, James D. Joseph, John Wongvipat, Nicola J. Clegg
PDF file - 312K
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::318f3ae7f053ae4cf142c57f94aff43b
https://doi.org/10.1158/0008-5472.22393733.v1
https://doi.org/10.1158/0008-5472.22393733.v1