Zobrazeno 1 - 10
of 10
pro vyhledávání: '"Joan Basset"'
Publikováno v:
Tetrahedron. 68:6269-6275
We report a direct iodination of indole and derivative compounds with iodine monochloride (ICl) in the presence of Celite ® . This procedure has now been extended to the iodination of substituted indoles, azaindoles and pyrroles. The scope of this p
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::33bdef109005794e00ca631b63bf3bb5
https://doi.org/10.1016/j.tet.2012.05.053
https://doi.org/10.1016/j.tet.2012.05.053
Publikováno v:
Tetrahedron. 68:356-362
Efficient synthesis of furo[3,4-b]indoles starting from the corresponding indole is reported. The first route involves derivatization, protection, and deprotection steps, which stretch the syntheses. The second method provides a shorter and more effi
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::ff1be03db0cb35a07c2634674bfac531
https://doi.org/10.1016/j.tet.2011.10.022
https://doi.org/10.1016/j.tet.2011.10.022
Autor:
Giovanni Casula, Salvatore Plescia, Ramon Pouplana, Joan Basset, Y. Harrak, Glòria Rosell, Maria Grazia Cusimano, Demetrio Raffa, Maria Dolors Pujol
Publikováno v:
Journal of Medicinal Chemistry. 53:6560-6571
Following our previous research on anti-inflammatory drugs (NSAIDs), we report on the design and synthesis of 4-(aryloyl)phenyl methyl sulfones. These substances were characterized for their capacity to inhibit cyclooxygenase (COX-1 and COX-2) isoenz
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::04705a2aa28acdddd9ac225539b232ed
https://doi.org/10.1021/jm100398z
https://doi.org/10.1021/jm100398z
Publikováno v:
Tetrahedron. 65:1951-1956
Aryl halides and triflates are coupled with primary amides to give the corresponding arylamines in the presence of a palladium catalyst, a suitable ligand, and a base. The catalyst system performs well for a large number of different substrates at 10
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::59d87642f682a9f0930d5b9d4274d6d5
https://doi.org/10.1016/j.tet.2009.01.033
https://doi.org/10.1016/j.tet.2009.01.033
Publikováno v:
ChemInform. 43
A mild, efficient, and safe method for the iodination of indoles and azaindoles is developed.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::f02d254850f102c761aace0bd080201b
https://doi.org/10.1002/chin.201250117
https://doi.org/10.1002/chin.201250117
Autor:
Charlotte Chaulet, Marie-Claude Viaud-Massuard, Cécile Croix, Joan Basset, Maria-Dolores Pujol
Publikováno v:
ChemInform. 41
The optimized conditions allow the deprotection of a broad spectrum of substrates without affecting the functional groups.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::ae69090f583bd1225f551bfac780a28d
https://doi.org/10.1002/chin.201043110
https://doi.org/10.1002/chin.201043110
Autor:
Charlotte Chaulet, Marie-Claude Viaud-Massuard, Joan Basset, Maria-Dolores Pujol, Cécile Croix
Publikováno v:
SYNLETT
SYNLETT, Georg Thieme Verlag, 2010, pp.1481-1484
SYNLETT, Georg Thieme Verlag, 2010, pp.1481-1484
International audience; A mild method for the desulfonylation of N-indoles and N-azaindoles is described. Deprotection is carried out under basic conditions, using sodium tert-butoxide in dioxane. Several functionalized indoles and 7-azaindoles were
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f54e23b714ae867c27faec6d84a9f2c4
https://hal.science/hal-00614869
https://hal.science/hal-00614869
Publikováno v:
ChemInform. 40
Aryl halides and triflates are coupled with primary amides to give the corresponding arylamines in the presence of a palladium catalyst, a suitable ligand, and a base. The catalyst system performs well for a large number of different substrates at 10
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::236dc10dfb63ed535d29866b16d18a13
https://doi.org/10.1002/chin.200927054
https://doi.org/10.1002/chin.200927054
Publikováno v:
ChemInform. 38
Aryl bromides are coupled with N -compounds to give the corresponding arylamines in the presence of a palladium catalyst, a suitable ligand, and a weak base. The catalysts perform well for a large number of different starting material combinations at
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d75daa8c61042767ba14c6dc1a3c9593
https://doi.org/10.1002/chin.200701156
https://doi.org/10.1002/chin.200701156
Autor:
Youssef Harrak, Giovanni Casula, Joan Basset, GloÌria Rosell, Salvatore Plescia, Demetrio Raffa, Maria Grazia Cusimano, Ramon Pouplana, Maria Dolors Pujol
Publikováno v:
Journal of Medicinal Chemistry; Sep2010, Vol. 53 Issue 18, p6560-6571, 12p