Imidazoquinoline Derivatives as Potential Inhibitors of InhA Enzyme and Mycobacterium tuberculosis

Autor: Pascal Hoffmann, Joëlle Azéma-Despeyroux, Fernanda Goncalves, Alessandro Stamilla, Nathalie Saffon-Merceron, Frédéric Rodriguez, Giulia Degiacomi, Maria Rosalia Pasca, Christian Lherbet

Publikováno v: Molecules, Vol 29, Iss 13, p 3076 (2024)

Tuberculosis is a serious public health problem worldwide. The search for new antibiotics has become a priority, especially with the emergence of resistant strains. A new family of imidazoquinoline derivatives, structurally analogous to triazolophtha

Externí odkaz: https://doaj.org/article/2c1ad0e2eed648a4ab889c946f63fcb2

Quantum chemistry-based interpretations on the lowest triplet state of luminescent lanthanides complexes. Part 2. Influence of the electrostatic interactions on the triplet state energy of terbium complexes

Autor: Laurent Maron, Romuald Poteau, Claude Picard, Joëlle Azéma, Christine Tedeschi, Fabien Gutierrez, Jean-Pierre Daudey, Pierre Tisnès

Publikováno v: Journal of Molecular Structure: THEOCHEM. 756:151-162

In part I of this series, we have focused our attention on a theoretical interpretation of the luminescent properties of some recently synthetized lanthanide–hydroxamate complexes (LnL 3 stoichiometry, with L − =[CO–N(R)O] − ). Following the

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::ab8da3004d01fad51fc045c9ccbb15d3
https://doi.org/10.1016/j.theochem.2005.09.004

A solid-state study of eight-coordinate lanthanide(iii) complexes (Ln = Eu, Gd, Tb, Dy) with 1-hydroxy-2-pyridinone

Autor: Christine Tedeschi, Pierre Tisnès, Heinz Gornitzka, Joëlle Azéma, Claude Picard

Publikováno v: Dalton Transactions. :1738-1745

Four lanthanide complexes of 1-hydroxy-2-pyridinone (HOPO) have been synthesised from aqueous solution at pH ≈ 7 and their structures and luminescent properties have been established. This ligand coordinates to lanthanide(III) ions as an anionic bi

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::0f1b5b3e7455ad1fb60880b908fc1252
https://doi.org/10.1039/b300159h

Antimalarial Bicyclic Peroxides Belonging to the G-Factor Family: Mechanistic Aspects of their Formation and Iron (II) Induced Reduction

Autor: Henri Vial, Corinne Payrastre, Jérémy Ruiz, Joëlle Azéma, Michel Baltas, Béatrice Tuccio, Christiane André-Barrès

Publikováno v: Current Topics in Medicinal Chemistry
Current Topics in Medicinal Chemistry, 2014, 14 (14), pp.1668--1683. ⟨10.2174/1568026614666140808154326⟩
Current Topics in Medicinal Chemistry, 2014, 14 (14), pp.1668-1683. ⟨10.2174/1568026614666140808154326⟩
Current Topics in Medicinal Chemistry, Bentham Science Publishers, 2014, 14 (14), pp.1668-1683. ⟨10.2174/1568026614666140808154326⟩

International audience; Artemisinin and its derivatives are peroxide-containing compounds targeting P. falciparum. We review here structural analogues of bicyclic peroxides belonging to the G factors family presenting antimalarial properties. They we

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::79d5a7e5d22b4b69652e8891847b005f
https://hal.archives-ouvertes.fr/hal-01460534

New Macrobicycles Containing a Tetralactam Moiety: Template Synthesis and Study of their Binding with Lanthanides

Autor: Juan Carlos Rodríguez-Ubis, Claude Picard, Pierre Tisnès, Ernesto Brunet, Joëlle Azéma, Patricia Ramos, Chantal Galaup, Olga Juanes

Publikováno v: Tetrahedron. 56:2673-2681

The synthesis of macrobicyclic cryptands 1 , 2 from an 18-membered diazatetralactam and 6,6′-bis(bromomethyl)-2,2′-bipyridine or 2,6-bis(3-bromomethyl-1-pyrazolyl)pyridine has been investigated using various metal carbonates. The analysis of the

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::84a5bd52d68f6a9ff76b36badf19cf48
https://doi.org/10.1016/s0040-4020(00)00164-2