Zobrazeno 1 - 6
of 6
pro vyhledávání: '"Jiro Haga"'
Publikováno v:
The Journal of Organic Chemistry. 60:4363-4374
Publikováno v:
ChemInform. 26
Publikováno v:
Chemistry Letters. 20:2175-2178
Michael addition reactions of acyl oxazolidinones to ethyl 3-trifluoromethylacrylate were found to proceed smoothly with a high degree of diastereo- as well as diastereofacial selectivity at the new carbon–carbon bond.
Publikováno v:
Chemistry Letters. 20:2171-2174
Michael addition reactions of lithium enolates derived from ketones, esters, and amides to ethyl 3-trifluoromethylacrylate were found to proceed smoothly in moderate to excellent chemical yields as well as with a high degree of diastereoselectivity a
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 1:271-276
Both enantiomers of unnatural 4,4-difluorinated threonine were readily prepared via enzymatic optical resolution and only the corresponding (2 S , 3 S ) isomer was found to possess comparable or even stronger in vitro antitumor activity than the curr
Publikováno v:
Journal of Fluorine Chemistry. 54:293
The authors would like to report our recent result on highly diastereoselective Michael addition of enolates derived from ketones, esters, and amides towards ethyl 3-trifluoromethylacrylate ( E )-1 . Lithium enolates were found to react with this acc