Zobrazeno 1 - 10
of 13
pro vyhledávání: '"Jessica Sallander"'
Autor:
Silvana Vasile, Anders Hallberg, Jessica Sallander, Mathias Hallberg, Johan Åqvist, Hugo Gutiérrez-de-Terán
Publikováno v:
Biomolecules, Vol 10, Iss 4, p 649 (2020)
Angiotensin II receptor type 1 and 2 (AT1R and AT2R) are two G-protein coupled receptors that mediate most biological functions of the octapeptide Angiotensin II (Ang II). AT2R is upregulated upon tissue damage and its activation by selective AT2R ag
Externí odkaz:
https://doaj.org/article/409d868369ea4f3fabdf7e0d5112eaf4
Autor:
Anders Hallberg, Mathias Hallberg, Johan Åqvist, Silvana Vasile, Jessica Sallander, Hugo Gutiérrez-de-Terán
Publikováno v:
Biomolecules
Volume 10
Issue 4
Biomolecules, Vol 10, Iss 649, p 649 (2020)
Volume 10
Issue 4
Biomolecules, Vol 10, Iss 649, p 649 (2020)
Angiotensin II receptor type 1 and 2 (AT1R and AT2R) are two G-protein coupled receptors that mediate most biological functions of the octapeptide Angiotensin II (Ang II). AT2R is upregulated upon tissue damage and its activation by selective AT2R ag
Autor:
Ismael Rodríguez-Espigares, Mariona Torrens-Fontanals, Johanna K.S. Tiemann, David Aranda-García, Juan Manuel Ramírez-Anguita, Tomasz Maciej Stepniewski, Nathalie Worp, Alejandro Varela-Rial, Adrián Morales-Pastor, Brian Medel Lacruz, Gáspár Pándy-Szekeres, Eduardo Mayol, Toni Giorgino, Jens Carlsson, Xavier Deupi, Slawomir Filipek, Marta Filizola, José Carlos Gómez-Tamayo, Angel Gonzalez, Hugo Gutierrez-de-Teran, Mireia Jimenez, Willem Jespers, Jon Kapla, George Khelashvili, Peter Kolb, Dorota Latek, Maria Marti-Solano, Pierre Matricon, Minos-Timotheos Matsoukas, Przemyslaw Miszta, Mireia Olivella, Laura Perez-Benito, Davide Provasi, Santiago Ríos, Iván Rodríguez-Torrecillas, Jessica Sallander, Agnieszka Sztyler, Nagarajan Vaidehi, Silvana Vasile, Harel Weinstein, Ulrich Zachariae, Peter W. Hildebrand, Gianni De Fabritiis, Ferran Sanz, David E. Gloriam, Arnau Cordomi, Ramon Guixà-González, Jana Selent
Publikováno v:
Nature Methods
bioRxiv
bioRxiv
G protein-coupled receptors (GPCRs) are involved in numerous physiological processes and are the most frequent targets of approved drugs. The explosion in the number of new 3D molecular structures of GPCRs (3D-GPCRome) during the last decade has grea
Autor:
Minos-Timotheos Matsoukas, David E. Gloriam, Ismael Rodríguez-Espigares, Agnieszka Sztyler, Davide Provasi, Arnau Cordomí, Peter Kolb, David Aranda-García, Toni Giorgino, Ferran Sanz, Mariona Torrens-Fontanals, Peter W. Hildebrand, Maria Marti-Solano, Mireia Olivella, Alejandro Varela-Rial, Gianni De Fabritiis, José Carlos Gómez-Tamayo, Laura Pérez-Benito, Tomasz Maciej Stepniewski, Eduardo Mayol, Silvana Vasile, Slawomir Filipek, Ulrich Zachariae, Jens Carlsson, Dorota Latek, Harel Weinstein, Gáspár Pándy-Szekeres, Przemyslaw Miszta, Willem Jespers, Nathalie Worp, Mireia Jiménez-Rosés, Juan Manuel Ramírez-Anguita, Marta Filizola, George Khelashvili, Angel Gonzalez, Brian Medel Lacruz, Pierre Matricon, Iván Rodríguez-Torrecillas, Xavier Deupi, Adrián Morales-Pastor, Jessica Sallander, Hugo Gutiérrez-de-Terán, Johanna K. S. Tiemann, Jana Selent, Jon Kapla, Ramon Guixà-González, Santiago Ríos
Publikováno v:
Nature Methods
Nature methods (Online) 17 (2020): 777–787. doi:10.1038/s41592-020-0884-y
info:cnr-pdr/source/autori:Rodríguez-Espigares, Ismael; Torrens-Fontanals, Mariona; Tiemann, Johanna K.S.; Aranda-García, David; Ramírez-Anguita, Juan Manuel; Stepniewski, Tomasz Maciej; Worp, Nathalie; Varela-Rial, Alejandro; Morales-Pastor, Adrián; Medel-Lacruz, Brian; Pándy-Szekeres, Gáspár; Mayol, Eduardo; Giorgino, Toni; Carlsson, Jens; Deupi, Xavier; Filipek, Slawomir; Filizola, Marta; Gómez-Tamayo, José Carlos; Gonzalez, Angel; Gutiérrez-de-Terán, Hugo; Jiménez-Rosés, Mireia; Jespers, Willem; Kapla, Jon; Khelashvili, George; Kolb, Peter; Latek, Dorota; Marti-Solano, Maria; Matricon, Pierre; Matsoukas, Minos Timotheos; Miszta, Przemyslaw; Olivella, Mireia; Perez-Benito, Laura; Provasi, Davide; Ríos, Santiago; R. Torrecillas, Iván; Sallander, Jessica; Sztyler, Agnieszka; Vasile, Silvana; Weinstein, Harel; Zachariae, Ulrich; Hildebrand, Peter W.; De Fabritiis, Gianni; Sanz, Ferran; Gloriam, David E.; Cordomi, Arnau; Guixà-González, Ramon; Selent, Jana/titolo:GPCRmd uncovers the dynamics of the 3D-GPCRome/doi:10.1038%2Fs41592-020-0884-y/rivista:Nature methods (Online)/anno:2020/pagina_da:777/pagina_a:787/intervallo_pagine:777–787/volume:17
Nature methods (Online) 17 (2020): 777–787. doi:10.1038/s41592-020-0884-y
info:cnr-pdr/source/autori:Rodríguez-Espigares, Ismael; Torrens-Fontanals, Mariona; Tiemann, Johanna K.S.; Aranda-García, David; Ramírez-Anguita, Juan Manuel; Stepniewski, Tomasz Maciej; Worp, Nathalie; Varela-Rial, Alejandro; Morales-Pastor, Adrián; Medel-Lacruz, Brian; Pándy-Szekeres, Gáspár; Mayol, Eduardo; Giorgino, Toni; Carlsson, Jens; Deupi, Xavier; Filipek, Slawomir; Filizola, Marta; Gómez-Tamayo, José Carlos; Gonzalez, Angel; Gutiérrez-de-Terán, Hugo; Jiménez-Rosés, Mireia; Jespers, Willem; Kapla, Jon; Khelashvili, George; Kolb, Peter; Latek, Dorota; Marti-Solano, Maria; Matricon, Pierre; Matsoukas, Minos Timotheos; Miszta, Przemyslaw; Olivella, Mireia; Perez-Benito, Laura; Provasi, Davide; Ríos, Santiago; R. Torrecillas, Iván; Sallander, Jessica; Sztyler, Agnieszka; Vasile, Silvana; Weinstein, Harel; Zachariae, Ulrich; Hildebrand, Peter W.; De Fabritiis, Gianni; Sanz, Ferran; Gloriam, David E.; Cordomi, Arnau; Guixà-González, Ramon; Selent, Jana/titolo:GPCRmd uncovers the dynamics of the 3D-GPCRome/doi:10.1038%2Fs41592-020-0884-y/rivista:Nature methods (Online)/anno:2020/pagina_da:777/pagina_a:787/intervallo_pagine:777–787/volume:17
G-protein-coupled receptors (GPCRs) are involved in numerous physiological processes and are the most frequent targets of approved drugs. The explosion in the number of new three-dimensional (3D) molecular structures of GPCRs (3D-GPCRome) over the la
Autor:
Johanna K. S. Tiemann, George Khelashvili, Brian Medel-Lacruz, Ramon Guixà-González, Alejandro Varela-Rial, José Carlos Gómez-Tamayo, Marta Filizola, Dorota Latek, Gianni De Fabritiis, David Aranda-García, Juan Manuel Ramírez-Anguita, Santiago Ríos, Davide Provasi, David E. Gloriam, Jana Selent, Minos-Timotheos Matsoukas, Toni Giorgino, Ferran Sanz, Jon Kapla, Silvana Vasile, Slawomir Filipek, Xavier Deupi, Adrián Morales-Pastor, Przemyslaw Miszta, Àngel Puyol González, Mireia Jiménez-Rosés, Harel Weinstein, Peter Kolb, Agnieszka Sztyler, Nathalie Worp, Maria Marti-Solano, Arnau Cordomí, Ulrich Zachariae, Ismael Rodríguez-Espigares, Pierre Matricon, Ivan R. Torrecillas, Tomasz Maciej Stepniewski, Eduardo Mayol, Gáspár Pándy-Szekeres, Peter W. Hildebrand, Mireia Olivella, Mariona Torrens-Fontanals, Hugo Gutiérrez-de-Terán, Laura Pérez-Benito, Jens Carlsson, Willem Jespers, Jessica Sallander
Publikováno v:
Nature Methods. 17:861-862
Publikováno v:
Current Topics in Medicinal Chemistry. 17:40-58
The family of adenosine receptors (ARs) is focus of several medicinal chemistry programs aimed to find new potent and selective drugs. Each receptor subtype has been proposed as a relevant drug target in the treatment of, e.g., cardiovascular or infl
Autor:
Johan Åqvist, Jessica Sallander, Charlotta Wallinder, Hugo Gutiérrez-de-Terán, Anders Hallberg
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 26:1355-1359
Agonists of the angiotensin II receptor type 2 (AT2), a G-protein coupled receptor, promote tissue protective effects in cardiovascular and renal diseases, while antagonists reduce neuropathic pain. We here report detailed molecular models that expla
Autor:
Silvana, Vasile, Mauricio, Esguerra, Willem, Jespers, Ana, Oliveira, Jessica, Sallander, Johan, Åqvist, Hugo, Gutiérrez-de-Terán
Publikováno v:
Methods in molecular biology (Clifton, N.J.). 1705
The recent increase in available G protein-coupled receptor structures now contributes decisively to the structure-based ligand design. In this context, computational approaches in combination with medicinal chemistry and pharmacology are extremely h
Autor:
Silvana Vasile, Ana Oliveira, Johan Åqvist, Willem Jespers, Mauricio Esguerra, Jessica Sallander, Hugo Gutiérrez-de-Terán
Publikováno v:
Methods in Molecular Biology ISBN: 9781493974641
The recent increase in available G protein-coupled receptor structures now contributes decisively to the structure-based ligand design. In this context, computational approaches in combination with medicinal chemistry and pharmacology are extremely h
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::386ef2e5797e19cacdc14a8931bb29f8
https://doi.org/10.1007/978-1-4939-7465-8_2
https://doi.org/10.1007/978-1-4939-7465-8_2
Autor:
Jessica Sallander, Alexey Siretskiy, Xabier Bello, Hugo Gutiérrez-de-Terán, Mauricio Esguerra
Publikováno v:
Nucleic Acids Research
GPCR-ModSim (http://open.gpcr-modsim.org) is a centralized and easy to use service dedicated to the structural modeling of G-protein Coupled Receptors (GPCRs). 3D molecular models can be generated from amino acid sequence by homology-modeling techniq
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::88d3d4ec48d5dc84070beaba8fa5d71e
http://urn.kb.se/resolve?urn=urn:nbn:se:uu:diva-301022
http://urn.kb.se/resolve?urn=urn:nbn:se:uu:diva-301022