Zobrazeno 1 - 10
of 12
pro vyhledávání: '"Jessica Lombino"'
Autor:
Jessica Lombino, Rosario Vallone, Maura Cimino, Maria Rita Gulotta, Giada De Simone, Maria Agnese Morando, Raffaele Sabbatella, Simona Di Martino, Mario Fogazza, Federica Sarno, Claudia Coronnello, Maria De Rosa, Chiara Cipollina, Lucia Altucci, Ugo Perricone, Caterina Alfano
Publikováno v:
Clinical Epigenetics, Vol 15, Iss 1, Pp 1-16 (2023)
Abstract Background Lysine demethylase enzymes (KDMs) are an emerging class of therapeutic targets, that catalyse the removal of methyl marks from histone lysine residues regulating chromatin structure and gene expression. KDM4A isoform plays an impo
Externí odkaz:
https://doaj.org/article/b96d859348f0461a9deca1a52950e217
A New Family of Jumonji C Domain-Containing KDM Inhibitors Inspired by Natural Product Purpurogallin
Autor:
José A. Souto, Federica Sarno, Angela Nebbioso, Chiara Papulino, Rosana Álvarez, Jessica Lombino, Ugo Perricone, Alessandro Padova, Lucia Altucci, Ángel R. de Lera
Publikováno v:
Frontiers in Chemistry, Vol 8 (2020)
Aberrant epigenetic modifications are involved in cancer development. Jumonji C domain-containing histone lysine demethylases (KDMs) are found mainly up-regulated in breast, prostate, and colon cancer. Currently, growing interest is focusing on the i
Externí odkaz:
https://doaj.org/article/71962f45271b4c1eaa2a7fa7aa8241a3
Autor:
Nedra Mekni, Maria De Rosa, Chiara Cipollina, Maria Rita Gulotta, Giada De Simone, Jessica Lombino, Alessandro Padova, Ugo Perricone
Publikováno v:
International Journal of Molecular Sciences, Vol 20, Iss 20, p 4974 (2019)
NLRP3 (NOD-like receptor family, pyrin domain-containing protein 3) activation has been linked to several chronic pathologies, including atherosclerosis, type-II diabetes, fibrosis, rheumatoid arthritis, and Alzheimer’s disease. Therefore, NLRP3 re
Externí odkaz:
https://doaj.org/article/e274187d1cce4e418a484f45b51c15f9
Autor:
Johannes Schimunek, Philipp Seidl, Katarina Elez, Tim Hempel, Tuan Le, Frank Noé, Simon Olsson, Lluís Raich, Robin Winter, Hatice Gokcan, Filipp Gusev, Evgeny M. Gutkin, Olexandr Isayev, Maria G. Kurnikova, Chamali H. Narangoda, Roman Zubatyuk, Ivan P. Bosko, Konstantin V. Furs, Anna D. Karpenko, Yury V. Kornoushenko, Mikita Shuldau, Artsemi Yushkevich, Mohammed B. Benabderrahmane, Patrick Bousquet-Melou, Ronan Bureau, Beatrice Charton, Bertrand C. Cirou, Gérard Gil, William J. Allen, Suman Sirimulla, Stanley Watowich, Nick A. Antonopoulos, Nikolaos E. Epitropakis, Agamemnon K. Krasoulis, Vassilis P. Pitsikalis, Stavros T. Theodorakis, Igor Kozlovskii, Anton Maliutin, Alexander Medvedev, Petr Popov, Mark Zaretckii, Hamid Eghbal-zadeh, Christina Halmich, Sepp Hochreiter, Andreas Mayr, Peter Ruch, Michael Widrich, Francois Berenger, Ashutosh Kumar, Yoshihiro Yamanishi, Kam Y.J. Zhang, Emmanuel Bengio, Yoshua Bengio, Moksh J. Jain, Maksym Korablyov, Cheng-Hao Liu, Gilles Marcou, Enrico Glaab, Kelly Barnsley, Suhasini M. Iyengar, Mary Jo Ondrechen, V. Joachim Haupt, Florian Kaiser, Michael Schroeder, Luisa Pugliese, Simone Albani, Christina Athanasiou, Andrea Beccari, Paolo Carloni, Giulia D'Arrigo, Eleonora Gianquinto, Jonas Goßen, Anton Hanke, Benjamin P. Joseph, Daria B. Kokh, Sandra Kovachka, Candida Manelfi, Goutam Mukherjee, Abraham Muñiz-Chicharro, Francesco Musiani, Ariane Nunes-Alves, Giulia Paiardi, Giulia Rossetti, S. Kashif Sadiq, Francesca Spyrakis, Carmine Talarico, Alexandros Tsengenes, Rebecca C. Wade, Conner Copeland, Jeremiah Gaiser, Daniel R. Olson, Amitava Roy, Vishwesh Venkatraman, Travis J. Wheeler, Haribabu Arthanari, Klara Blaschitz, Marco Cespugli, Vedat Durmaz, Konstantin Fackeldey, Patrick D. Fischer, Christoph Gorgulla, Christian Gruber, Karl Gruber, Michael Hetmann, Jamie E. Kinney, Krishna M. Padmanabha Das, Shreya Pandita, Amit Singh, Georg Steinkellner, Guilhem Tesseyre, Gerhard Wagner, Zi-Fu Wang, Ryan J. Yust, Dmitry S. Druzhilovskiy, Dmitry A. Filimonov, Pavel V. Pogodin, Vladimir Poroikov, Anastassia V. Rudik, Leonid A. Stolbov, Alexander V. Veselovsky, Maria De Rosa, Giada De Simone, Maria R. Gulotta, Jessica Lombino, Nedra Mekni, Ugo Perricone, Arturo Casini, Amanda Embree, D. Benjamin Gordon, David Lei, Katelin Pratt, Christopher A. Voigt, Kuang-Yu Chen, Yves Jacob, Tim Krischuns, Pierre Lafaye, Agnès Zettor, M. Luis Rodríguez, Kris M. White, Daren Fearon, Frank Von Delft, Martin A. Walsh, Dragos Horvath, Charles L. Brooks III, Babak Falsafi, Bryan Ford, Adolfo García-Sastre, Sang Yup Lee, Nadia Naffakh, Alexandre Varnek, Günter Klambauer, Thomas M. Hermans
The COVID-19 pandemic continues to pose a substantial threat to human lives and is likely to do so for years to come. Despite the availability of vaccines, searching for efficient small-molecule drugs that are widely available, including in low- and
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::28010b1a0350f378ef0dcc633e87f6e1
https://doi.org/10.26434/chemrxiv-2023-1d5w8
https://doi.org/10.26434/chemrxiv-2023-1d5w8
Autor:
Nada Elkholy, Ahmad Abdelwaly, Karim Mohamed, Emanuele Amata, Jessica Lombino, Giuseppe Cosentino, Sebastiano Intagliata, Mohamed A. Helal
Publikováno v:
Chemical Biology & Drug Design. 100:25-40
Sigma receptor is a transmembrane non-GPCR protein expressed mainly in the endoplasmic reticulum membrane associated with mitochondria. It is classified into two types: Sigma-1 (S1R) and Sigma-2 (S2R) based on their biological functions. S1R has been
Autor:
Giuliana Costanzo, Vincenzo Patamia, Rita Turnaturi, Carmela Parenti, Chiara Zagni, Jessica Lombino, Emanuele Amata, Agostino Marrazzo, Lorella Pasquinucci, Antonio Rescifina
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f7342e45f8868a48599166380250c844
https://hdl.handle.net/20.500.11769/551232
https://hdl.handle.net/20.500.11769/551232
Autor:
Saad Touqeer, Laura Ielo, Cristina Prandi, Wolfgang Holzer, Alexander Roller, Laura Castoldi, Jessica Lombino, Vittorio Pace
Publikováno v:
Angewandte Chemie International Edition. 59:20852-20857
The selective formal insertion (homologation) of a carbon unit bridging the two trifluoroacetamidoyl chlorides (TFAICs) units is reported. The tactic is levered on a highly chemoselective homologation-metalation-acyl nucleophilic substitution sequenc
Autor:
Laura Ielo, Laura Castoldi, Saad Touqeer, Jessica Lombino, Alexander Roller, Cristina Prandi, Wolfgang Holzer, Vittorio Pace
Publikováno v:
Angewandte Chemie. 132:21038-21043
A new family of Jumonji C domain-containing KDM inhibitors inspired by natural product Purpurogallin
Autor:
Ugo Perricone, Chiara Papulino, Lucia Altucci, Jessica Lombino, Federica Sarno, José A. Souto, Rosana Alvarez, Angela Nebbioso, Alessandro Padova, Angel R. de Lera
Publikováno v:
Investigo. Repositorio Institucional de la Universidade de Vigo
Universidade de Vigo (UVigo)
Frontiers in Chemistry, Vol 8 (2020)
Frontiers in Chemistry
Universidade de Vigo (UVigo)
Frontiers in Chemistry, Vol 8 (2020)
Frontiers in Chemistry
Aberrant epigenetic modifications are involved in cancer development. Jumonji C domain-containing histone lysine demethylases (KDMs) are found mainly up-regulated in breast, prostate, and colon cancer. Currently, growing interest is focusing on the i
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8dce7c939771f243318972c10026548f
http://hdl.handle.net/11093/2344
http://hdl.handle.net/11093/2344
Autor:
Patrizia Diana, Ugo Perricone, Stella Cascioferro, Alessandro Padova, Barbara Parrino, Girolamo Cirrincione, Jessica Lombino, Maria Rita Gulotta
Molecular dynamics (MD) has become increasingly popular due to the development of hardware and software solutions and the improvement in algorithms, which allowed researchers to scale up calculations in order to speed them up. MD simulations are usua
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d6cc6c8ea9ef64b053b9fa3abeb3eaf6
http://hdl.handle.net/10447/291780
http://hdl.handle.net/10447/291780