Zobrazeno 1 - 10
of 85
pro vyhledávání: '"Jerzy Kossakowski"'
Autor:
Jarosław Walory, Lidia Mielczarek, Małgorzata Jarończyk, Mirosława Koronkiewicz, Jerzy Kossakowski, Ryszard Bugno, Andrzej J. Bojarski, Zdzisław Chilmonczyk
Publikováno v:
International Journal of Molecular Sciences, Vol 19, Iss 10, p 3260 (2018)
The cytotoxic activity of several serotonin transporter (SERT) inhibitors and subtype of serotonin receptor 1A (5-HT1A receptor) ligands have been examined in androgen-insensitive human PC-3 prostate and neuroblastoma SH-SY5Y cancer cells. Almost all
Externí odkaz:
https://doaj.org/article/263959c90c5944e18b4fa8a54defd5a2
Publikováno v:
Molecules, Vol 15, Iss 7, Pp 4737-4749 (2010)
Halogen derivatives of selected 3-benzofurancarboxylic acids were prepared using 6-acetyl-5-hydroxy-2-methyl-3-benzofuranocarboxylic acid as starting material. 1H-NMR spectra were obtained for all of the synthesized structures, and for compound VI, a
Externí odkaz:
https://doaj.org/article/544bef1776044487a233d22a820bbee3
Autor:
David Collu, Roberta Loddo, Cristina Ibba, Laura Ester Marongiu, Paolo La Colla, Izabela Dybala, Anna E. Koziol, Marta Struga, Jerzy Kossakowski, Magdalena Pakosinska-Parys
Publikováno v:
Molecules, Vol 14, Iss 12, Pp 5189-5202 (2009)
A series of twenty arylpiperazine derivatives of 1,7,8,9-tetrachloro-10,10-dimethoxy-4-azatricyclo[5.2.1.02,6]dec-8-ene-3,5-dione have been prepared. These derivatives were tested in vitro with the aim of identifying novel lead compounds active again
Externí odkaz:
https://doaj.org/article/09ccea67bbe9474cbc64bd51680a7cb9
Autor:
Marta Struga, Izabela Dybała, Anna E. Kozioł, Barbara Mirosław, Anna Bielenica, Jerzy Kossakowski
Publikováno v:
Molecules, Vol 13, Iss 8, Pp 1570-1583 (2008)
A series of twenty six arylpiperazine and aminoalkanol derivatives of 4-azatricyclo[ 5.2.2.02,6]undecane-3,5,8-trione have been prepared. The synthesized compounds were evaluated for their cytotoxicity and anti-HIV-1 activity in MT-4 cells.
Externí odkaz:
https://doaj.org/article/ea9e75eae0a84f0d93e3422b9e46d0c6
Publikováno v:
Molecules, Vol 11, Iss 8, Pp 615-626 (2006)
The preparation of a number of cyclic imide 5-HT1A receptor ligandderivatives has been described. Their structures were conformationally constrained byintroducing rigid linkers containing unsaturated bonds or aromatic benzene rings. Thesecompounds ar
Externí odkaz:
https://doaj.org/article/fe7ef9e231b240718f8a02126bccfa95
Publikováno v:
Molbank, Vol 2010, Iss 3, p M697 (2010)
The title compound was synthesized by condensation of an oxiran imide derivative with an appropriate amine and its IR, 1H NMR, 13C NMR and mass spectroscopic data are reported. The synthesized compound was evaluated for its cytotoxicity and anti-HIV-
Externí odkaz:
https://doaj.org/article/7f43fb5c31824d41a6fc0f14cff28e48
Autor:
Anna Bielenica, Jerzy Kossakowski
Publikováno v:
Molbank, Vol 2010, Iss 2, p M685 (2010)
9-Methyl-3,5-dioxo-4-azatricyclo[5.2.2.02,6]undec-8-ene-1,8-diyl diacetatewas synthesized from 2-methylcyclohexane-1,3-dione and 1H-pyrrole-2,5-dione. The title compound was characterized by 1H NMR, 13C NMR, elemental analysis and MS.
Externí odkaz:
https://doaj.org/article/57529c5eb76d44889ae5a7eb194d4c07
Autor:
Jerzy Kossakowski, Marta Struga
Publikováno v:
Molbank, Vol 2007, Iss 2, p M534 (2007)
n/a
Externí odkaz:
https://doaj.org/article/e17921fad2684a058270691a355c2176
Autor:
Mariola Napiórkowska, Karolina Królewska, Bożena Kuran, Jerzy Kossakowski, Barbara Nawrot, Marcin Cieślak, Julia Kaźmierczak-Barańska
Publikováno v:
Anti-Cancer Agents in Medicinal Chemistry. 16:852-864
A large group of aminoalkyl and aminoalkanol derivatives of selected dicarboximides were synthesized and characterized by 1HNMR, 13CNMR and ESI MS spectra analysis. The thirty nine new compounds were tested for their cytotoxic properties in human chr
Autor:
Jerzy Kossakowski, Andrzej J. Bojarski, Ryszard Bugno, Małgorzata Jarończyk, Zdzisław Chilmonczyk, Mirosława Koronkiewicz, Lidia Mielczarek, Jarosław Walory
Publikováno v:
International Journal of Molecular Sciences
Volume 19
Issue 10
International Journal of Molecular Sciences, Vol 19, Iss 10, p 3260 (2018)
Volume 19
Issue 10
International Journal of Molecular Sciences, Vol 19, Iss 10, p 3260 (2018)
The cytotoxic activity of several serotonin transporter (SERT) inhibitors and subtype of serotonin receptor 1A (5-HT1A receptor) ligands have been examined in androgen-insensitive human PC-3 prostate and neuroblastoma SH-SY5Y cancer cells. Almost all