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pro vyhledávání: '"Jeffery E Campbell"'
Autor:
Robert B McCall, Michael D. Ennis, Nabil B Ghazal, Deborah K Hyslop, Lawrence W Fitzgerald, Dac M. Dinh, Nanette F. Nichols, Michelle L Kagey, Christopher S Knauer, Robert L Hoffman, Chris L Chio, Rebecca M. Olson, Christopher L. Haber, Kjell A. Svensson, Jeffery E Campbell
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 13:2369-2372
The design and synthesis of the novel 2,3,4,5-tetrahydro-1H-[1,4]diazepino[1,7-a]indole 5 is described. This azepinoindole has excellent affinity for 5-HT(2C) (K(i) 4.8 nM) and modest selectivity over 5-HT(2A) ( approximately 4-fold). Several N- and
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d7e865895ecbc42acd8733dd4f39d674
https://doi.org/10.1016/s0960-894x(03)00403-7
https://doi.org/10.1016/s0960-894x(03)00403-7
