Versatile Synthetic Approach for Selective Diversification of Bicyclic Aza-Diketopiperazines

Autor: Florent Péron, Stéphanie Riché, Brigitte Lesur, Marcel Hibert, Philippe Breton, Jean-Marie Fourquez, Nicolas Girard, Dominique Bonnet

Publikováno v: ACS Omega, Vol 3, Iss 11, Pp 15182-15192 (2018)

Externí odkaz: https://doaj.org/article/c4d6b21dab3c4184bf1a90c890f0c662

Chemoselective borylation of bromoiodoarene in continuous flow: synthesis of bromoarylboronic acids

Autor: Guillaume Reynard, Eric Wimmer, Jérémi Richelet, Jean-Marie Fourquez, Hélène Lebel

Publikováno v: Journal of Flow Chemistry. 13:21-29

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::0e8e5cfcff431916d2a7a91dc4e0df12
https://doi.org/10.1007/s41981-022-00246-w

Productive Syntheses of Privileged Scaffolds Inspired by the Recognition of a Diels–Alder Pattern Common to Three Classes of Natural Products

Autor: Philippe Breton, Léon Ghosez, Solo Goldstein, Brigitte Lesur, Eduard Badarau, Jean Michel Henlin, K. Harsha Vardhan Reddy, Aurore Loudet, Etienne Pair, Jean Marie Fourquez, Stijn Claerhout, Stéphane Massip, Laurent Trembleau, Charles Simon

Publikováno v: Chemistry – A European Journal. 26:15477-15481

Identification of a common Diels-Alder pattern in three classes of bioactive natural products led us to study the synthesis and cycloaddition of a new class of cyclic dienes readily available from β,γ-unsaturated lactams. A practical and readily sc

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b7208784b43ad0034592963c96644e70
https://doi.org/10.1002/chem.202002372

Versatile Synthetic Approach for Selective Diversification of Bicyclic Aza-Diketopiperazines

Autor: Jean-Marie Fourquez, Brigitte Lesur, Nicolas Girard, Stéphanie Riché, Florent Péron, Marcel Hibert, Dominique Bonnet, Philippe Breton

Publikováno v: ACS Omega
ACS Omega, ACS Publications, 2018, 3 (11), pp.15182-15192. ⟨10.1021/acsomega.8b01752⟩
ACS Omega, 2018, 3 (11), pp.15182-15192. ⟨10.1021/acsomega.8b01752⟩
ACS Omega, Vol 3, Iss 11, Pp 15182-15192 (2018)

Herein, we report a convenient synthesis of unprecedented aza-diketopiperazines (aza-DKPs). The strategy is based on selective diversification of bicyclic aza-DKP scaffolds by click reaction, N-acylation, and/or N-alkylation. These scaffolds containi

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::96110c3ba5615a13a4b696fc9fa9d7d8
https://doi.org/10.1021/acsomega.8b01752

Indium-Catalyzed Cycloisomerization of 1,6-Cyclohexenylalkynes

Autor: Fabien Fontaine-Vive, Jean-Marie Fourquez, Véronique Michelet, Vincent Davenel, Christian Nisole, Chloé Puteaux

Publikováno v: Catalysts, Vol 11, Iss 546, p 546 (2021)

Efficient four- and five-step routes to access functionalized bicyclo[3.2.1]oct-2-ene and bicyclo[3.3.1]nonadiene via indium-mediated cycloisomerization of 1,6-enynes has been developed. This atom-economical catalytic process was optimized and relied

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b141d87e98b876bb181210b3ba59feea
https://doi.org/10.3390/catal11050546