Zobrazeno 1 - 10
of 100
pro vyhledávání: '"Jean-François Willart"'
Publikováno v:
Pharmaceutics, Vol 15, Iss 5, p 1505 (2023)
This paper is dealing with the dissolution mechanism of crystalline sulindac into amorphous Polyvinylpyrrolidone (PVP) upon heating and annealing at high temperatures. Special attention is paid on the diffusion mechanism of drug molecules in the poly
Externí odkaz:
https://doaj.org/article/97174b16e8cf48658457b49c879a7ff7
Autor:
Anna Krupa, Florence Danède, Dorota Majda, Agnieszka Węgrzyn, Dominik Strojewski, Ita Kondera, Jean-François Willart
Publikováno v:
European Journal of Pharmaceutics and Biopharmaceutics. 188:137-146
Autor:
J. Verin, Pierre-Emmanuel Lemesre, G. Tourrel, Christophe Vincent, Florence Siepmann, Jean-François willart, V. Solarczyk, Juergen Siepmann, Florence Danede, P. Stahl, Adam Qnouch
Publikováno v:
International Journal of Pharmaceutics: X, Vol 3, Iss, Pp 100088-(2021)
International Journal of Pharmaceutics: X
International Journal of Pharmaceutics: X, 2021, 3, pp.100088. ⟨10.1016/j.ijpx.2021.100088⟩
International Journal of Pharmaceutics: X, Elsevier, 2021, 3, pp.100088. ⟨10.1016/j.ijpx.2021.100088⟩
International Journal of Pharmaceutics: X
International Journal of Pharmaceutics: X, 2021, 3, pp.100088. ⟨10.1016/j.ijpx.2021.100088⟩
International Journal of Pharmaceutics: X, Elsevier, 2021, 3, pp.100088. ⟨10.1016/j.ijpx.2021.100088⟩
Cochlear implants containing iridium platinum electrodes are used to transmit electrical signals into the inner ear of patients suffering from severe or profound deafness without valuable benefit from conventional hearing aids. However, their placeme
Autor:
Catherine Dejoie, Juergen Siepman, Charline Henaff, Florence Siepman, Mathieu Guerain, Frédéric Affouard, Jean-François willart, Florence Danede
Publikováno v:
Acta Crystallographica Section C Structural Chemistry
Acta Crystallographica Section C Structural Chemistry, International Union of Crystallography, 2021, Acta Crystallographica Section C Structural Chemistry, 77 (12), pp.800-806. ⟨10.1107/s2053229621012171⟩
Acta Crystallographica Section C : Structural Chemistry [2014-...]
Acta Crystallographica Section C : Structural Chemistry [2014-..], 2021, 77 (12), pp.800-806. ⟨10.1107/s2053229621012171⟩
Acta Crystallographica Section C Structural Chemistry, International Union of Crystallography, 2021, Acta Crystallographica Section C Structural Chemistry, 77 (12), pp.800-806. ⟨10.1107/s2053229621012171⟩
Acta Crystallographica Section C : Structural Chemistry [2014-...]
Acta Crystallographica Section C : Structural Chemistry [2014-..], 2021, 77 (12), pp.800-806. ⟨10.1107/s2053229621012171⟩
The crystal structure of the stable form of vitamin B2 or riboflavin (C17H20N4O6) was solved using high-resolution powder X-ray diffraction (PXRD). The high-resolution PXRD pattern of riboflavin was recorded at room temperature at the European Synchr
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::392acc834b5070095e733f5d35d77181
https://hal.univ-lille.fr/hal-03469379
https://hal.univ-lille.fr/hal-03469379
Publikováno v:
Journal of Pharmaceutical Sciences
Journal of Pharmaceutical Sciences, Wiley, 2019, 108 (8), pp.2635-2642. ⟨10.1016/j.xphs.2019.03.017⟩
Journal of Pharmaceutical Sciences, 2019, 108 (8), pp.2635-2642. ⟨10.1016/j.xphs.2019.03.017⟩
Journal of Pharmaceutical Sciences, Wiley, 2019, 108 (8), pp.2635-2642. ⟨10.1016/j.xphs.2019.03.017⟩
Journal of Pharmaceutical Sciences, 2019, 108 (8), pp.2635-2642. ⟨10.1016/j.xphs.2019.03.017⟩
International audience; This paper shows how milling can be used to explore the phase diagram of pharmaceuticals. This process has been applied to sulindac. A short milling has been found to trigger a polymorphic transformation between form II and fo
Publikováno v:
International Journal of Pharmaceutics
International Journal of Pharmaceutics, 2022, 622, pp.121846. ⟨10.1016/j.ijpharm.2022.121846⟩
International Journal of Pharmaceutics, 2022, 622, pp.121846. ⟨10.1016/j.ijpharm.2022.121846⟩
International audience; New clinical indications for an orphan drug bosentan are prompting the improvement of the drug formulation. Since bosentan is available as monohydrate, the information on its anhydrous form together with the assessment of its
Autor:
Juergen Siepmann, Youcef Benzine, Florence Danede, Jean-François willart, Florence Siepmann, Youness Karrout, Christel Neut
Publikováno v:
European Journal of Pharmaceutics and Biopharmaceutics
European Journal of Pharmaceutics and Biopharmaceutics, 2021, 168, pp.1-14. ⟨10.1016/j.ejpb.2021.08.007⟩
European Journal of Pharmaceutics and Biopharmaceutics, 2021, 168, pp.1-14. ⟨10.1016/j.ejpb.2021.08.007⟩
International audience; A variety of polymer:polymer blends was used to prepare hot melt extrudates and empty capsules (bodies and caps) by injection-molding using a benchtop extruder (Babyplast). Kollidon SR:inulin and Carbothane:inulin blends were
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::35790275f577d870817b79c4f2ff34d3
https://hal.univ-lille.fr/hal-03814465
https://hal.univ-lille.fr/hal-03814465
Autor:
Jean-François willart, Oriane Cantin, Florence Danede, Youness Karrout, Florence Siepmann, Juergen Siepmann
Publikováno v:
Journal of Drug Delivery Science and Technology
Journal of Drug Delivery Science and Technology, Elsevier, 2021, 61, pp.102238. ⟨10.1016/j.jddst.2020.102238⟩
Journal of Drug Delivery Science and Technology, 2021, 61, pp.102238. ⟨10.1016/j.jddst.2020.102238⟩
Journal of Drug Delivery Science and Technology, Elsevier, 2021, 61, pp.102238. ⟨10.1016/j.jddst.2020.102238⟩
Journal of Drug Delivery Science and Technology, 2021, 61, pp.102238. ⟨10.1016/j.jddst.2020.102238⟩
International audience; A variety of poly(ethylene oxide) (PEO)-based matrix tablets loaded with theophylline, ibuprofen or metoprolol tartrate was prepared via hot melt extrusion. The initial drug loading was varied from 10 to 60 %, the PEO polymer
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d3c1952a89720026d5d6fe29fcd3f4e4
https://hal.univ-lille.fr/hal-03023791/document
https://hal.univ-lille.fr/hal-03023791/document
Autor:
Laurent Paccou, Anthony Dupont, Alain Hédoux, Florence Danede, Yannick Guinet, Mathieu Guerain, Jean-François willart
Publikováno v:
International Journal of Pharmaceutics
International Journal of Pharmaceutics, 2020, International Journal of Pharmaceutics, 590, pp.119902. ⟨10.1016/j.ijpharm.2020.119902⟩
International Journal of Pharmaceutics, Elsevier, 2020, International Journal of Pharmaceutics, 590, pp.119902. ⟨10.1016/j.ijpharm.2020.119902⟩
International Journal of Pharmaceutics, 2020, International Journal of Pharmaceutics, 590, pp.119902. ⟨10.1016/j.ijpharm.2020.119902⟩
International Journal of Pharmaceutics, Elsevier, 2020, International Journal of Pharmaceutics, 590, pp.119902. ⟨10.1016/j.ijpharm.2020.119902⟩
International audience; In this paper, we present a kinetic investigation of the polymorphic transformation γ → α of sorbitol under milling in the objective to identify the microscopic mechanisms that govern this type of solid-state transformatio
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5020660c7c94d292afb18dbbffb5bb96
https://hal.univ-lille.fr/hal-02965510
https://hal.univ-lille.fr/hal-02965510