Zobrazeno 1 - 10 of 21 pro vyhledávání: '"Javad Ameri Rad"'
1
Akademický článek
Crystal structure of 2-[(3S,4S)-4-(anthracen-9-yl)-1-(4-methoxyphenyl)-2-oxoazetidin-3-yl]-2-aza-2H-phenalene-1,3-dione unknown solvate
Autor: Ísmail Çelik, Mehmet Akkurt, Aliasghar Jarrahpour, Javad Ameri Rad, Ömer Çelik
Publikováno v: Acta Crystallographica Section E: Crystallographic Communications, Vol 71, Iss 3, Pp o184-o185 (2015)
The central β-lactam ring of the title compound, C36H24N2O4, is almost planar (r.m.s. deviation = 0.003 Å) and makes dihedral angles of 17.17 (19), 89.76 (17) and 78.44 (17)° with the benzene ring, the anthracene ring (r.m.s. deviation = 0.003 Å)
Externí odkaz: https://doaj.org/article/652987b89c1f4f53810bc9e1133e1993
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2
Akademický článek
Crystal structure of 2-[4-(4-chlorophenyl)-1-(4-methoxyphenyl)-2-oxoazetidin-3-yl]benzo[de]isoquinoline-1,3-dione dimethyl sulfoxide monosolvate
Autor: Ísmail Çelik, Mehmet Akkurt, Aliasghar Jarrahpour, Javad Ameri Rad, Ömer Çelik
Publikováno v: Acta Crystallographica Section E: Crystallographic Communications, Vol 71, Iss 2, Pp o129-o130 (2015)
In the title solvated compound, C28H19N2O4·C2H6OS, the central β-lactam ring is almost planar (r.m.s. deviation = 0.002 Å). It makes dihedral angles of 1.92 (11), 83.23 (12) and 74.90 (10)° with the methoxy- and chlorophenyl rings and the ring pl
Externí odkaz: https://doaj.org/article/ad2ff21636cd4077807d1dec463df341
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3
Synthesis, in-vitro biological evaluation, and molecular docking study of novel spiro-β-lactam-isatin hybrids
Autor: Aliasghar Jarrahpour, Zahra Jowkar, Zahra Haghighijoo, Roghayeh Heiran, Javad Ameri Rad, Véronique Sinou, Florent Rouvier, Christine Latour, Jean Michel Brunel, Namık Özdemir
Publikováno v: Medicinal Chemistry Research
Medicinal Chemistry Research, Springer Verlag, 2022, 31 (6), pp.1026-1034. ⟨10.1007/s00044-022-02898-8⟩
Medicinal Chemistry Research, 2022, 31 (6), pp.1026-1034. ⟨10.1007/s00044-022-02898-8⟩
International audience; In our ongoing search for bioactive compounds, a class of novel spiro-β-lactam isatin hybrids has been synthesized through a [2 + 2] cycloaddition reaction from 1-allyl-3-(arylimino)indolin-2-one, ketenes and various aryloxy
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::86d00b5489b702855fa94302ad8a14c2
https://doi.org/10.1007/s00044-022-02898-8
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5
Cytotoxicity, anticancer, and antioxidant properties of mono and bis-naphthalimido β-lactam conjugates
Autor: Javad Ameri Rad, Mohammad Ghanbari, Edward Turos, Aida Iraji, Sedigheh Kianpour, S. Masoud Nabavizadeh, Nassim Borazjani, Aliasghar Jarrahpour, Maryam Behzadi, Gyula Batta, Marzieh Dadkhah Aseman
Publikováno v: Medicinal Chemistry Research. 29:1355-1375
This article reports the diastereoselective synthesis of some novel naphthalimido and bis-naphthalimido β-lactam derivatives and a preliminary evaluation of their anticancer properties. The reactions were completely diastereoselective, leading exclu
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::7b55eadac7b714d2cb2a31f8cad8690e
https://doi.org/10.1007/s00044-020-02552-1
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7
Synthesis and antimicrobial/antimalarial activities of novel naphthalimido trans-β-lactam derivatives
Autor: Edward Turos, Véronique Sinou, Javad Ameri Rad, Christine Latour, Aliasghar Jarrahpour, Yahia N. Mabkhot, H. Zgou, Taibi Ben Hadda, Jean Michel Brunel
Publikováno v: Medicinal Chemistry Research. 26:2235-2242
This paper describes for the first time the synthesis and microbiological assessment of some new β-lactam derivatives containing a 1,8-naphthalimide functional group. These compounds were obtained through a [2 + 2] cyclocondensation (Staudinger reac
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::14873ac88ac763644df5098b7e3e0322
https://doi.org/10.1007/s00044-017-1920-z
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8
Design, synthesis and biological evaluation of some novel diastereoselective β-lactams bearing 2-mercaptobenzothiazole and benzoquinoline
Autor: Milad Mohkam, Javad Ameri Rad, Somayyeh Mirzaeinia, Gyula Batta, Hamid Reza Karbalaei-Heidari, Edward Turos, Younes Ghasemi, Nassim Borazjani, Mohammad Ghanbari, Aliasghar Jarrahpour, Maryam Behzadi
We report the synthesis of some novel β-lactam hybrids of 2-mercaptobenzothiazole and benzoquinoline. These compounds were synthesized by a [2 + 2]-cycloaddition reaction of imines 8a-d and ketenes derived from substituted acetic acids. The reaction
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bd1ef3ee2758c39adbe484aa49c7632d
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9
Three-Component Synthesis of Chromeno β-Lactam Hybrids for Inflammation and Cancer Screening
Autor: Jean Michel Brunel, Younes Ghasemi, Gyula Batta, Saghi Sepehri, Carole Digiorgio, Amin Reza Akbarizadeh, Maryam Sasanipour, Milad Mohkam, Nassim Borazjani, Mohammad Ghanbari, Edward Turos, Javad Ameri Rad, Aliasghar Jarrahpour, Maryam Behzadi
Publikováno v: European Journal of Medicinal Chemistry
European Journal of Medicinal Chemistry, 2019, 179, pp.389-403. ⟨10.1016/j.ejmech.2019.06.036⟩
European Journal of Medicinal Chemistry, Elsevier, 2019, 179, pp.389-403. ⟨10.1016/j.ejmech.2019.06.036⟩
International audience; Highly diastereoselective synthesis of chromeno β-lactam hybrids was achieved by an efficient one-pot three-component reaction. With this procedure, the desired β-lactam products were obtained in good yields and with exclusi
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::46cf316a902022198398112b0750dac0
https://hal-amu.archives-ouvertes.fr/hal-02392426/document
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10
Design, synthesis, activity evaluation and QSAR studies of novel antimalarial 1,2,3-triazolo-beta-lactam derivatives
Autor: Saeed Yousefinejad, Javad Ameri Rad, Jean Michel Brunel, Véronique Sinou, Malihe Aye, Christine Latour, Aliasghar Jarrahpour, Edward Turos
Publikováno v: Journal-Iranian Chemical Society
Journal-Iranian Chemical Society, Iranian Chemical Society, 2018, 15 (6), pp.1311-1326. ⟨10.1007/s13738-018-1330-2⟩
Journal of the Iranian Chemical Society
Journal of the Iranian Chemical Society, 2018, 15 (6), pp.1311-1326. ⟨10.1007/s13738-018-1330-2⟩
This paper describes the synthesis of some new beta-lactam derivatives containing the 1,2,3-triazole moiety. All the compounds were evaluated for their in vitro antimicrobial and antimalarial activities. Moderate to excellent antimalarial activities
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fa0c7da774e4a111b6bb654c390db36c
https://hal-amu.archives-ouvertes.fr/hal-02143574
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