Zobrazeno 1 - 10
of 23
pro vyhledávání: '"Jatinder P. Bassin"'
Synthesis and Antibacterial Activity of Benzo[4,5]isothiazolo[2,3-a]pyrazine-6,6-dioxide Derivatives
Publikováno v:
Molecules, Vol 22, Iss 11, p 1889 (2017)
Using a routine procedure, a number of derivatives of the benzo[4,5]isothiazolo[2,3-a]pyrazine-6,6-dioxide ring system have been synthesized from readily available starting materials. A series of chalcones were synthesized, which were subsequently re
Externí odkaz:
https://doaj.org/article/192d27fba6af49189e7ad8c2992197aa
Autor:
Jatinder P. Bassin, Bhavani Anagani, Christopher Benham, Madhu Goyal, Maryam Hashemian, Ute Gerhard
Publikováno v:
Molecules, Vol 21, Iss 8, p 967 (2016)
A simple synthetic route affording 27%–85% yields of benzo[6,7][1,5]diazocino[2,1-a]isoindol-12(14H)-one ring systems from readily available 3-(2-oxo-2-phenylethyl) isobenzofuran-1(3H)-ones and 2-(aminomethyl)aniline starting materials in toluene a
Externí odkaz:
https://doaj.org/article/8dd6fea0f427427e851703ed21f56527
Autor:
Chandani Patel, Jatinder P. Bassin, Mark Scott, Jenna Flye, Ann P. Hunter, Lee Martin, Madhu Goyal
Publikováno v:
Molecules, Vol 21, Iss 7, p 861 (2016)
A number of 1,2-benzothiazines have been synthesized in a three-step process. Nine chalcones 1–9 bearing methyl, fluoro, chloro and bromo substituents were chlorosulfonated with chlorosulfonic acid to generate the chalcone sulfonyl chlorides 10–1
Externí odkaz:
https://doaj.org/article/f3a91f411c2c4fb3b3a23cd04c5095a8
Publikováno v:
Acta Crystallographica Section E, Vol 67, Iss 1, Pp o12-o12 (2011)
The title compound, C11H12ClNO4S, adopts a Z configuration about the C=C double bond. The benzisothiazole system is essentially planar [maximum deviation of 0.235 (2) Å for the S atom]. In the crystal, the molecules stack parallel to each other in t
Externí odkaz:
https://doaj.org/article/dcf9729100d14b9fa40616bac1d7809c
Autor:
Madhu Goyal, Jonathan A. G. Cox, Gurdyal S. Besra, Bhavani Anagani, Christopher D. Benham, Jatinder P. Bassin, Jagbir Singh, Tummala Rama Krishna Reddy
Publikováno v:
The Cell Surface, Vol 6, Iss, Pp 100041-(2020)
The Cell Surface
The Cell Surface
Highlights • Chalcone 1a inhibits the growth of Mycobacterium bovis BCG (MIC 6.25 µg.ml−1). • Chalcone 1a directly targets InhA.
Objectives The search for new TB drugs has become one of the great challenges for modern medicinal chemistry.
Objectives The search for new TB drugs has become one of the great challenges for modern medicinal chemistry.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8bd151125dfaf5b433544d0825fffe78
http://www.sciencedirect.com/science/article/pii/S2468233020300086
http://www.sciencedirect.com/science/article/pii/S2468233020300086
Autor:
Madhu Goyal, Ute Gerhard, Maryam Hashemian, Bhavani Anagani, Christopher D. Benham, Jatinder P. Bassin
Publikováno v:
Molecules, Vol 21, Iss 8, p 967 (2016)
Molecules; Volume 21; Issue 8; Pages: 967
Molecules
Molecules; Volume 21; Issue 8; Pages: 967
Molecules
A simple synthetic route affording 27%-85% yields of benzo[6,7][1,5]diazocino[2,1-a]isoindol-12(14H)-one ring systems from readily available 3-(2-oxo-2-phenylethyl) isobenzofuran-1(3H)-ones and 2-(aminomethyl)aniline starting materials in toluene and
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6a4ca0b50252dace291ebefda0a93918
http://www.mdpi.com/1420-3049/21/8/967
http://www.mdpi.com/1420-3049/21/8/967
Publikováno v:
Synthetic Communications. 30:3693-3701
We report a novel synthesis of 4-chloro-2-cyclohexyl-6,7-dimethoxy-2H-1,2-benzothiazine-1,1-dioxide 6 from 3,4-dimethoxychalcone 1. Chlorosulfonation of 1 followed by amination, then epoxidation under basic conditions with immediate elimination of th
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::846da8162c032890fc6917c2c0fac5f1
https://doi.org/10.1080/00397910008086996
https://doi.org/10.1080/00397910008086996
Publikováno v:
Synthetic Communications. 30:2961-2965
A facile synthesis of benzo[d]benzo[2,3][1,4]diazepino[1,7-b] isothiazole, a new heterocyclic ring system is reported.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::d9d14296c993e4ae22797e77743acc48
https://doi.org/10.1080/00397910008087446
https://doi.org/10.1080/00397910008087446
Publikováno v:
Phosphorus, Sulfur, and Silicon and the Related Elements. 142:83-91
Styrylpyridine (1) reacted with chlorosulfonic acid (6 mole equivalents) and excess thionyl chloride to the give the corresponding para sulfonyl chloride, which was characterized as the N,N-dimethyl sulfonamide. The pyridine ring appeared to deactiva
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::f71b32b243d41adc81ee3ee9d4b225c7
https://doi.org/10.1080/10426509808029668
https://doi.org/10.1080/10426509808029668
Publikováno v:
Acta Crystallographica Section E, Vol 67, Iss 1, Pp o12-o12 (2011)
Acta Crystallographica Section E: Structure Reports
Acta Crystallographica Section E: Structure Reports
The title compound, C11H12ClNO4S, adopts a Z configuration about the C=C double bond. The benzisothiazole system is essentially planar [maximum deviation of 0.235 (2) Å for the S atom]. In the crystal, the molecules stack parallel to each other in t
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1b4dd469798093fb5b385873be2dbf6a
http://scripts.iucr.org/cgi-bin/paper?S1600536810049561
http://scripts.iucr.org/cgi-bin/paper?S1600536810049561