Zobrazeno 1 - 10
of 58
pro vyhledávání: '"Jarmila Kaustová"'
Autor:
Jarmila Vinsova, Ales Imramovsky, Vladimir Buchta, Martina Ceckova, Martin Dolezal, Frantisek Staud, Josef Jampilek, Jarmila Kaustova
Publikováno v:
Molecules, Vol 12, Iss 1, Pp 1-12 (2008)
A new series of salicylanilide acetates was synthesized and evaluated for their in vitro antifungal and antituberculotic activity. Some of the evaluated compounds possessed comparable or better antifungal activity than a fluconazole standard. All the
Externí odkaz:
https://doaj.org/article/ed46a365389149c8b7df0d87852a27ef
Publikováno v:
Molecules, Vol 10, Iss 7, Pp 783-793 (2005)
A series of lipophilic 2-substituted 5,7-di-tert-butylbenzoxazoles was prepared in average yields by the reaction of 3,5-di-tert-butyl-1,2-benzoquinone with amino acids and dipeptides bearing N-terminal glycine. Dipeptides having other N-terminal ami
Externí odkaz:
https://doaj.org/article/ff712574b97e4f7db63936f66976c71f
Autor:
Jarmila Kaustová, MiloÅ¡ MacháÄÂek, Pia Vuorela, Luděk Jahodář, Jitka VytlaÄÂilová, VladimÃÂr Chobot, KatarÃÂna Kráľová, Martin Ã…Â ustr, Lenka Kubicová
Publikováno v:
Molecules, Vol 8, Iss 11, Pp 756-769 (2003)
Several 2,2-dimethyl-3-phenyl-1,2-dihydroquinazoline-4(3H)-thiones and 2-methyl-3-phenylquinazoline-4(3H)-thiones were synthesized and tested for their antimycobacterial, photosynthesis-inhibiting, and antialgal activity. Antimycobacterially active c
Externí odkaz:
https://doaj.org/article/a1ca30281a404bce8d77427591625b70
Autor:
Ute Möllmann, Hans-Martin Dahse, Karel Palát, Věra Klimešová, Eva Petrlikova, Jiří Kuneš, Jarmila Kaustová, Milan Peřina, Karel Waisser
Publikováno v:
European Journal of Medicinal Chemistry. 45:2719-2725
New 3-benzyl-4-thioxo-2H-1,3-benzoxazine-2(3H)-ones and 3-benzyl-2H-1,3-benzoxazine-2,4(3H)-dithiones were synthesized. The compounds were tested for in vitro antimycobacterial activity against Mycobacterium tuberculosis, Mycobacterium kansasii and M
Publikováno v:
European Journal of Medicinal Chemistry. 44:2286-2293
A set of 2-benzylsulfanyl derivatives of benzoxazole was synthesized and evaluated for their in vitro antimycobacterial activity against Mycobacterium tuberculosis, non-tuberculous mycobacteria and multidrug-resistant M. tuberculosis. The activities
Publikováno v:
Archiv der Pharmazie. 341:800-803
A series of 6-chloro-3-(4-alkylphenyl)-4-thioxo-2H-1,3-benzoxazine-2(3H)-ones, 7-chloro-3-(4-alkylphenyl)-4-thioxo-2H-1,3-benzoxazine-2(3H)-ones, 6-bromo-3-(4-alkylphenyl)-4-thioxo-2H-1,3-benzoxazine-2(3H)-ones, 6,8-dibromo-3-(4-alkylphenyl)-4-thioxo
Autor:
Josef Matyk, Jarmila Kaustová, Petra Husáková, Hana Divišová, Karel Waisser, Jiri Kunes, Vera Klimesova, Karel Palát
Publikováno v:
Archiv der Pharmazie. 340:264-267
Based on our previous studies, 21 new halogenated 3-(4-alkylphenyl)-1,3-benzoxazine-2,4-(3H)-diones were synthesized by the reaction of salicylanilides and methyl-chloroformate. All compounds were screened in vitro against three different strains of
Autor:
Bohumila Kozáková, Jarmila Kaustová, Lev Mezenský, Carolin Lechleitner, Maria Müllerová, Wolfgang M. Prodinger, Vladimír Polanecký, Milan Kubín
Publikováno v:
Central European Journal of Public Health. 14:168-174
SummaRy Objectives: To compare M. tuberculosis complex genotypes from representative regions of the Czech Republic in order to estimate changes in strain prevalence and in the extent of imported drug-resistant tuberculosis. Methods: Primary M. tuberc
Publikováno v:
Il Farmaco. 59:615-625
The series of derivatives of substituted N-pyridinylsalicylamides were synthesized. The compounds were evaluated for in vitro antimycobacterial activity against Mycobacterium avium and two strains of Mycobacterium kansasii. In the quantitative struct
Autor:
Jisi Kunes, Milan Pour, Petra Kubanová, Milan Pesina, Karel Waisser, Jarmila Kaustová, Vladimír Buchta, Bures O, Vsra Klimesova, Pavel Holy
Publikováno v:
Scopus-Elsevier
A set of 40 derivatives of 3-hydroxypicolinic acid and 2-sulfanylbenzoic acid, isosteric to salicylanilides was synthesized. The compounds were evaluated for in vitro activity against Mycobacterium tuberculosis, Mycobacterium kansasii and Mycobacteri