Zobrazeno 1 - 7
of 7
pro vyhledávání: '"James Densmore Copp"'
Publikováno v:
The Journal of Organic Chemistry. 63:5050-5058
A general regio- and stereoselective synthesis of 3,3-diarylacrylamides is reported. Palladium-catalyzed coupling reactions of propiolamides with aryl halides provide arylpropiolamides. A subsequent hydroarylation reaction of these arylpropiolamides
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::da0b91b7430110fc8fc297f274ebe764
https://doi.org/10.1021/jo980235h
https://doi.org/10.1021/jo980235h
Publikováno v:
Synthetic Communications. 26:3491-3494
A robust process for the preparation of multikilogram quantities of 2-chloro-4,6-dimethoxy-1,3,5-triazine (1) is described.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::bb1cf67cf845612154711a04ab62c26b
https://doi.org/10.1080/00397919608003754
https://doi.org/10.1080/00397919608003754
Publikováno v:
ChemInform. 27
A robust process for the preparation of multikilogram quantities of 2-chloro-4,6-dimethoxy-1,3,5-triazine (1) is described.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::23e499ca2c48a8afec76c558e7a20149
https://doi.org/10.1002/chin.199650178
https://doi.org/10.1002/chin.199650178
Publikováno v:
ChemInform. 29
A general regio- and stereoselective synthesis of 3,3-diarylacrylamides is reported. Palladium-catalyzed coupling reactions of propiolamides with aryl halides provide arylpropiolamides. A subsequent hydroarylation reaction of these arylpropiolamides
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::b57848727023b606443a7fd5594e7281
https://doi.org/10.1002/chin.199850111
https://doi.org/10.1002/chin.199850111
Autor:
James Densmore Copp, Douglas Patton Kjell, Stephen C. Stirm, Francis Orerenyo Ginah, and Marvin M. Hansen, Slattery Brian James
Publikováno v:
Organic Process Research & Development. 4:295-297
The development of a manufacturable synthesis of LY213829 (4-thiazolidinone-5-[3,5-bis(1,1-dimethylethyl)-4-hydroxyphenyl] methyl) is described. Rather than reduction to eliminate the thiocarbonyl from the rhodanine moiety, the new route utilizes a n
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::d52ecc9bd957281a712c540eb094a520
https://doi.org/10.1021/op990197j
https://doi.org/10.1021/op990197j
Autor:
Hsiu-Chiung Yang, Patrick C. May, Guo Deqi, Jingdan Hu, David E. Timm, James Densmore Copp, Mccarthy James R, Shu-Hui Chen, Bruce D. Gitter, James McGee, Jason Eric Lamar, Ana B. Bueno
Publikováno v:
Bioorganicmedicinal chemistry letters. 14(1)
We describe herein the syntheses and evaluation of a series of C-termini pyridyl containing Phe*-Ala-based BACE inhibitors (5-19). In conjunction with four fixed residues at the P1 (Phe), P1 0 (Ala), P2 0 (Val), and P2 0 cap (Pyr.), rather detailed S
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e1ce111d1f972553e3d7ef26c8a3af7f
https://pubmed.ncbi.nlm.nih.gov/14684335
https://pubmed.ncbi.nlm.nih.gov/14684335
Autor:
Marvin M. Hansen, James Densmore Copp, Slattery Brian James, Douglas Patton Kjell, Francis Orerenyo Ginah
Publikováno v:
HETEROCYCLES. 48:1307
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::4fe57f3f68c6b520b3545696155c0352
https://doi.org/10.3987/com-98-8138
https://doi.org/10.3987/com-98-8138