Zobrazeno 1 - 7
of 7
pro vyhledávání: '"Jamal A. Jilani"'
Publikováno v:
Pharmaceuticals, Vol 7, Iss 4, Pp 453-463 (2014)
The N-ethoxycarbonylmorpholine moiety was evaluated as a novel prodrug moiety for carboxylic acid containing drugs represented by diclofenac (1). Compound 2, the N-ethoxycarbonylmorpholine ester of diclofenac was synthesized and evaluated as a potent
Externí odkaz:
https://doaj.org/article/03c3d07b6d7b460ab3d5958958842383
Publikováno v:
Biomedical Chromatography. 30:1416-1422
In the current work, the investigation and development of a chemo-enzymatic approach for the synthesis of neo-glycoproteins have been studied. This strategy is based on the regioselective enzymatic hydrolysis of peracetylated monosaccharide, function
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::76f6fc6d5f8bca8cd5678915d822747e
https://doi.org/10.1002/bmc.3699
https://doi.org/10.1002/bmc.3699
Publikováno v:
Biomedical chromatography : BMC. 30(9)
In the current work, the investigation and development of a chemo-enzymatic approach for the synthesis of neo-glycoproteins have been studied. This strategy is based on the regioselective enzymatic hydrolysis of peracetylated monosaccharide, function
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::2181ec102b1b892c32d670765db18b12
https://pubmed.ncbi.nlm.nih.gov/26864255
https://pubmed.ncbi.nlm.nih.gov/26864255
Publikováno v:
American Journal of Pharmacological Sciences. 2:100-102
Aim of the study is to establish physiologically-based in vitro in vivo correlation (IVIVC) of azithromycin, a biopharmaceutics classification system (BCS) class II drug (high permeability/ low solubility). In vitro dissolution was done using USP app
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::5927d48e83d9c818481e0048b5e3a578
https://doi.org/10.12691/ajps-2-6-1
https://doi.org/10.12691/ajps-2-6-1
Publikováno v:
Pharmaceuticals
Volume 7
Issue 4
Pages 453-463
Pharmaceuticals, Vol 7, Iss 4, Pp 453-463 (2014)
Volume 7
Issue 4
Pages 453-463
Pharmaceuticals, Vol 7, Iss 4, Pp 453-463 (2014)
The N-ethoxycarbonylmorpholine moiety was evaluated as a novel prodrug moiety for carboxylic acid containing drugs represented by diclofenac (1). Compound 2, the N-ethoxycarbonylmorpholine ester of diclofenac was synthesized and evaluated as a potent
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ebf43524278b405b66bf9d55b453ea75
Publikováno v:
Drug Development and Industrial Pharmacy. 23:319-323
Hydroxyethyl esters of diclofenac and mefenamic acid were prepared with the aim of obtaining enzymatically labile prodrugs, and their stability was evaluated in aqueous buffer solutions of pH 7.4, 1 N HCl, and also in human plasma. The hydrolytic deg
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::bd010982c5740d27b23223cb7521b1a0
https://doi.org/10.3109/03639049709149810
https://doi.org/10.3109/03639049709149810
Publikováno v:
Drug Design, Development and Therapy
Jamal A Jilani,1 Maha Shomaf,2 Karem H Alzoubi3 1Department of Medicinal Chemistry and Pharmacognosy, Jordan University of Science and Technology, Irbid, Jordan; 2Department of Pathology, Jordan University, Amman, Jordan; 3Department of Clinical Phar
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8935a5889d13362c97060c1d870e4833
https://www.dovepress.com/synthesis-and-evaluation-of-mutual-azo-prodrug-of-5-aminosalicylic-aci-peer-reviewed-article-DDDT
https://www.dovepress.com/synthesis-and-evaluation-of-mutual-azo-prodrug-of-5-aminosalicylic-aci-peer-reviewed-article-DDDT