Zobrazeno 1 - 4
of 4
pro vyhledávání: '"Jacob W. Herman"'
Autor:
Feyisola P. Olatunji, Michael Pun, Jacob W. Herman, Oscar Romero, Mitchell Maniatopoulos, Joseph D. Latoche, Robert A. Parise, Jianxia Guo, Jan H. Beumer, Carolyn J. Anderson, Clifford E. Berkman
Publikováno v:
Mol Cancer Ther
New targeted chemotherapeutics are urgently needed to minimize off-target toxicity and reduce the high-mortality rate associated with metastatic prostate cancer. Herein, we report on the modular synthesis, pharmacokinetics, and efficacy of two small-
Autor:
Clifford E. Berkman, Carolyn J. Anderson, Jan H. Beumer, Jianxia Guo, Robert A. Parise, Joseph D. Latoche, Mitchell Maniatopoulos, Oscar Romero, Jacob W. Herman, Michael Pun, Feyisola P. Olatunji
Supplementary Data from Modular Smart Molecules for PSMA-Targeted Chemotherapy
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3b2208a0a3a162c0934bede2fe5cdfa0
https://doi.org/10.1158/1535-7163.22523347
https://doi.org/10.1158/1535-7163.22523347
Autor:
Feyisola P. Olatunji, Jacob W. Herman, Brittany N. Kesic, Damilola Olabode, Clifford E. Berkman
Publikováno v:
Tetrahedron Letters. 71:152955
Autor:
Clifford E. Berkman, Damilola Olabode, Feyisola P. Olatunji, Jacob W. Herman, Brittany N. Kesic
Publikováno v:
Tetrahedron Lett
In this work, we developed a novel “click”-ready pH-cleavable phosphoramidate linker for controlled-release of monomethyl auristantin E (MMAE) in antibody- and small molecule-drug conjugates application. This water-soluble linker was found to hav