Zobrazeno 1 - 10
of 104
pro vyhledávání: '"J.-J. Vanden Eynde"'
Autor:
Jean-Marie Colet, Raphael Conotte, Bertrand Blankert, Maxime Helvenstein, J.-J. Vanden Eynde, Zehra Cagla Kahvecioglu, L. Verdy, Stéphanie Hambye
Publikováno v:
Journal of Pharmaceutical and Biomedical Analysis. 95:54-60
Pentamidine isethionate (PTMD) is an antiprotozoal agent used in different parasitic diseases as Human African Trypanosomiasis or Pneumocystis pneumonia. Given its side effects, numerous analogs are still under development worldwide. PTMD has been re
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1395ffa06049e69391f2de8d1bc9378b
https://doi.org/10.1016/j.jpba.2014.02.002
https://doi.org/10.1016/j.jpba.2014.02.002
Autor:
Olivier Denis, Emmanuel Gosselin, J. Conti, A. Van Cauwenberge, J.-J. Vanden Eynde, Kris Huygen, J. De Coninck
Publikováno v:
Sensors and Actuators B: Chemical. :549-555
Verrucarin A2 (VerA) is a toxic trichothecene mycotoxin that can be produced indoors at very low level by moulds contaminating dwellings and may be associated with several human health problems. In this study we describe a spectroscopic label-free bi
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::c2bc8fcca1fba1df1e40de7653a7b64a
https://doi.org/10.1016/j.snb.2012.03.008
https://doi.org/10.1016/j.snb.2012.03.008
Autor:
Delphine Forge, Tien Huang, Dimitri Stanicki, J.-J. Vanden Eynde, Julien Laurent, Davie Cappoen, Annie Mayence, Luc Verschaeve, Kris Huygen
Publikováno v:
European Journal of Medicinal Chemistry. 49:95-101
Despite progress in modern chemotherapy to combat tuberculosis, the causative pathogen Mycobacterium tuberculosis (M.tb.) is far from eradicated. Bacillary resistance to anti-mycobacterial agents, bacillary persistence and human immunodeficiency viru
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::84331f671d04588a86aa04aa8f1bdb74
https://doi.org/10.1016/j.ejmech.2011.12.035
https://doi.org/10.1016/j.ejmech.2011.12.035
Novel 4,5-Dihydropyrazolo[3,4-d]Pyrimidin-4-Ones and 3,4-Dihydropyrazolo[3,4-d]-1,2,3-Triazin-4-Ones
Publikováno v:
Bulletin des Sociétés Chimiques Belges. 100:401-406
β-benzylidene 3− and 5-amino-1-methyl-1H-pyrazole-4-carboxhydrazides 3 and 4 readily react with orthoesters to yield the 4,5-dihydropyrazolo [3,4-d] pyrimidin-4-ones 5-8. Syntheses of 3,4-dihydropyrazolo [3,4-d]-1,2,3-triazin-4-ones 9, 10, 13 and
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::4e3c2dcf5396de372e5287834afac064
https://doi.org/10.1002/bscb.19911000507
https://doi.org/10.1002/bscb.19911000507
Publikováno v:
Bulletin des Sociétés Chimiques Belges. 101:509-512
The title compounds can be synthesized readily by reaction of primary aromatic amines with the azinium salt obtained from thionyl chloride, pyridine, and 1,2-benzenedicarboxaldehyde.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::7c17b179fd14057d30c4ad65f45e50ce
https://doi.org/10.1002/bscb.19921010611
https://doi.org/10.1002/bscb.19921010611
Publikováno v:
Bulletin des Sociétés Chimiques Belges. 92:451-458
1-phenyl-3-methylpyrazolin-5-one, 1,5-dimethylpyrazolin-3-one and 1-phenyl-pyrazolidin-3,5-dione react with ethyl acetoacetate to yield pyrano [2,3-c] pyrazole-6-ones. Starting from 1-phenyl-3-aminopyrazolin-5-one or from 1-methyl-5-aminopyrazolin-3-
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::315324a3613d00e3f2b391b0c9a314bf
https://doi.org/10.1002/bscb.19830920505
https://doi.org/10.1002/bscb.19830920505
Autor:
J.-J. Vanden Eynde, A. Maquestiau
Publikováno v:
Bulletin des Sociétés Chimiques Belges. 95:641-648
Reactions between five β-dicarbonyl compounds (1–5) or their enaminocarbonyl analogues (6–10) and three heterocyclic amines (12–14) are studied. The two types of carbonyl derivatives give rise to the formation of the same final products. Kinet
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::f1521582486faeb0a32efae893c90d63
https://doi.org/10.1002/bscb.19860950807
https://doi.org/10.1002/bscb.19860950807
Publikováno v:
Bulletin des Sociétés Chimiques Belges. 94:575-583
Reactions between 4-amino-3-penten-2-one, ethyl 3-amino-2-butenoate or 3-amino-2-butenanilide and phenyl isocyanate yield mixtures of N- and C-adducts. Quantitative data allow to check the influence of the electronwithdrawing groups in the enaminocar
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::c509d9da69a16ec66455d010293d7125
https://doi.org/10.1002/bscb.19850940805
https://doi.org/10.1002/bscb.19850940805
Publikováno v:
Bulletin des Sociétés Chimiques Belges. 98:523-528
A comparison is established for the reactivity of benzaldehyde, N-(1-chlorobenzyl)pyridinium chloride or N-(1-chlorobenzyl)pyrimidinium chloride with several poorly nucleophilic and/or poorly soluble primary amines under mild experimental conditions.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::7718f8dfe3309e4abfc68d790c8154b3
https://doi.org/10.1002/bscb.19890980803
https://doi.org/10.1002/bscb.19890980803
Publikováno v:
Bulletin des Sociétés Chimiques Belges. 93:1073-1081
Various 1,3-disubstituted pyrazolin-5-ones, 3-phenylisoxazolin-5-one and 2-phenyloxazolin-5-one react with ethyl 3-amino-2-butenoate to yield compounds resulting from the elimination of ammonia between the precursors; subsequent intramolecular cycliz
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::7b6ca95825da5e645258bd46030d630f
https://doi.org/10.1002/bscb.19840931207
https://doi.org/10.1002/bscb.19840931207