Zobrazeno 1 - 10 of 63 pro vyhledávání: '"J. L. Mokrosz"'
1
Structure-Activity Relationship Studies of CNS Agents, Part 23[1]):N-(3-Phenylpropyl)- andN-[3(E)-Cinnamyl]-1,2,3,4-tetrahydroisoquinoline Mimic 1-Phenylpiperazine at 5-HT1A Receptors
Autor: J. L. Mokrosz, Maria H. Paluchowska, Andrzej J. Bojarski, Sijka Charakchieva-Minol, Maria J. Mokrosz, Beata Duszyńska
Publikováno v: Archiv der Pharmazie. 328:604-608
The 5-HT 1A receptor affinities and ionization constants of a set of 1-arylpiperazine (4) 1,2,3,4-tetrahydroisoquinoline (6), and -quinoline (7) containing N-(ω-arylalkyl) or N-(E)-cinnamyl substituents as well as two morpholine derivatives (8a, 8b)
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::9fdd2ab466e488d516d5f7c55289e7e7
https://doi.org/10.1002/ardp.19953280707
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2
Structure-Activity Relationship Studies of CNS Agents, Part 26 4-[2-(Cycloalkanecarboxamido)ethyl]-1-(2-methoxyphenyl)-piperazines: High-Affinity 5-HT1A Agonists
Autor: J. L. Mokrosz, Sijka Charakchieva-Minol, Maria H. Paluchowska, Aleksandra Kłodzińska, Ewa Chojnacka-Wójcik
Publikováno v: Archiv der Pharmazie. 328:770-774
Cycloalkanecarboxamido)ethyl]-1-(2-methoxyphenyl)piperazin es 8a-c, 8e, and 8h were obtained by acylation of 4-(2-aminoethyl)-1-(2-methoxyphenul)piperazine, and their 5-HT 1A , 5-HT 2A and α 1 receptor affinities were determined. It was found that t
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::fd76f3c0171e67e4dad1f02b4efa246f
https://doi.org/10.1002/ardp.19953281108
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3
ChemInform Abstract: Synthesis and Quantitative Structure-Activity Relationship Analysis of 2-(Aryl or Heteroaryl)quinolin-4-amines, a New Class of Anti-HIV-1 Agents
Autor: Lucjan Strekowski, Steven E. Patterson, Agnieszka Czarny, Marek T. Cegla, Roman L. Wydra, Raymond F. Schinazi, J. L. Mokrosz, Vidya A. Honkan
Publikováno v: ChemInform. 22
Thirty-eight 2-(aryl or heteroaryl)quinolin-4-amines, N,N-disubstituted, N-monosubstituted, and without a substituent at the amino group have been synthesized with use of novel chemistries developed by us recently. Some of these derivatives show anti
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::d51502755dcfc19dfdd419b7fb14c5ec
https://doi.org/10.1002/chin.199145180
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4
ChemInform Abstract: Structure and Spectral Properties of β-Carbolines. Part 4. Synthesis of the New Ring System: 9,10,15,15b-Tetrahydroindolo(1′,2′:4, 3)pyrazino(2,1-a)carbolin-7(6H)-one
Autor: Zofia Bielecka, J. L. Mokrosz, S. Misztal
Publikováno v: ChemInform. 22
1-Indol-2-yl-1,2,3,4-tetrahydro-β-carboline and its 5-methoxy derivative were synthesized by the Pictet-Spengler reaction between tryptamine or 5-methoxytryptamine and indole-2-carbaldehyde, with a high yield. A step-by-step oxidation of the indolyl
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::553d5d8e6a35833fc876f04dca4c4902
https://doi.org/10.1002/chin.199146296
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