Zobrazeno 1 - 10
of 18
pro vyhledávání: '"J S, Bontekoe"'
Autor:
H. C. Beyerman, J. S. Bontekoe
Publikováno v:
Recueil des Travaux Chimiques des Pays-Bas. 72:262-268
The high anti-tuberculosis activity of pyridine-4-carboxylic acid hydrazide (isonicotinic acid hydrazide, INH), together with the chemical similarity of pyridine and thiazole, has induced us to synthesize the thiazole carboxylic acid hydrazides and t
Publikováno v:
Recueil des Travaux Chimiques des Pays-Bas. 78:935-946
The synthesis is described of the “protected” linear nonapeptide: N-benzyloxycarbonyl-S-benzyl-L-cysteinyl-L-tyrosyl-L-isoleucyl-L-glutaminyl-L-asparaginyl-S-benzyl-L-cysteinyl-L-prolyl-L-leucylglycine amide (XI). In the new reaction steps N,N′
Publikováno v:
Recueil des Travaux Chimiques des Pays-Bas. 73:109-117
The synthesis is described of a number of 1- and 4-substituted derivatives of pyridine related to isonicotinic acid hydrazide (INH) and of isonicotinoyl hydrazones of some aldehydes. These compounds were prepared in order to test them for possible gr
Publikováno v:
Recueil des Travaux Chimiques des Pays-Bas. 73:325-332
Two syntheses of the hitherto unknown 5-bromothiazole are described. 2-Bromothiazole and 5-bromothiazole could be converted via the corresponding thiazolyllithium compounds into thiazole-2- and thiazole-5-carboxylic acid respectively. This constitute
Autor:
H. C. Beyerman, J. S. Bontekoe
Publikováno v:
Recueil des Travaux Chimiques des Pays-Bas. 79:1165-1173
A synthesis is described of the protected linear decapeptide: N-benzyloxycarbonyl-S-benzyl-L-cysteinyl-L-tyrosyl-L-tyrosyl-L-tyrosyl-L-glutaminyl-L-asparaginyl-S-benzyl-L-cysteinyl-L-prolyl-Ne-p-toluene-sulphonyl-L-lysylglycineamide (VI) in analytica
Publikováno v:
Recueil des Travaux Chimiques des Pays-Bas. 98:78-81
The retro configuration (9β,10α) was introduced into pregnane derivatives containing substituents at C(16) and/or C(17) by irradiation of a suitable 5,7-diene. In this way the title compounds became much more accessible than by the introduction of
Autor:
J. S. Bontekoe, H. C. Beyerman
Publikováno v:
Recueil des Travaux Chimiques des Pays-Bas. 83:255-275
A synthesis is described of the N-terminal octapeptide sequence derived from the pancreatic hormone glucagon (glucagon 1–8).
Autor:
H. C. Beyerman, J. S. Bontekoe
Publikováno v:
Recueil des Travaux Chimiques des Pays-Bas. 72:643-652
The syntheses of 4-guanidino-salicylic acid, 4-(N′-cyanoguanidino)- salicylic acid, and some related compounds are described. Intermolecular coupling of the diazonium salt of ρ-amino-salicylic acid and of its methyl ester yielded products which ar
Autor:
J. S. Bontekoe, H. C. Beyerman
Publikováno v:
Recueil des Travaux Chimiques des Pays-Bas. 81:699-709
A synthesis is described of the partially protected carboxyl-terminal tetrapeptide sequence, L-leucyl-L-methionyl-L-asparaginyl-O-t-butyl-L-threonine t-butyl ester, which is derived from the pancreatic hormone glucagon. In this synthesis we used succ
Autor:
H. C. Beyerman, P. J. Oud, V. Gerris, J. S. Bontekoe, W. L. C. Veer, J. E. Ribbers, P. J. van Ree
Publikováno v:
Recueil des Travaux Chimiques des Pays-Bas. 76:839-840