Spiroindolines identify the vesicular acetylcholine transporter as a novel target for insecticide action.

Autor: Ann Sluder, Sheetal Shah, Jérôme Cassayre, Ralph Clover, Peter Maienfisch, Louis-Pierre Molleyres, Elizabeth A Hirst, Anthony J Flemming, Min Shi, Penny Cutler, Carole Stanger, Richard S Roberts, David J Hughes, Thomas Flury, Michael P Robinson, Elke Hillesheim, Thomas Pitterna, Fredrik Cederbaum, Paul A Worthington, Andrew J Crossthwaite, John D Windass, Richard A Currie, Fergus G P Earley

Publikováno v: PLoS ONE, Vol 7, Iss 5, p e34712 (2012)

The efficacy of all major insecticide classes continues to be eroded by the development of resistance mediated, in part, by selection of alleles encoding insecticide insensitive target proteins. The discovery of new insecticide classes acting at nove

Externí odkaz: https://doaj.org/article/01ae6528af6c47e98391b659caff9a2a

List of Contributors

Autor: Y. Abe, Douglas D. Anspaugh, Takao Aoki, Raphael Aponte, Sadayuki Arimori, Gregory Armel, Shinichi Banba, Fabien Barreteau, James Barry, Anika Bartholomaeus, Dave Bartlett, Guillaume Berthon, Pascal Bindschaedler, Judith Blythe, Mohamed Boussemghoune, Peter Bowerman, Karla Bravo-Altamirano, Twyla A. Briddell, Zachary Buchan, A. Buchholz, Ruth Campe, Xiaofeng Cao, Jérôme Cassayre, Fredrik Cederbaum, Kang Chang, Yaning Chang, Lai Chen, Xiulei Chen, Yuzhong Chen, Jiagao Cheng, Thomas S. Churcher, Daniel Cordova, Dongliang Cui, John F. Daeuble, Peter Dahmen, H. Daido, M. Daniels, Kyle DeKorver, Jonathan DeLorbe, Alain De Mesmaeker, Philippe Desbordes, Willem Desmedt, Joachim Dickhaut, Jingao Dong, Myriem El Qacemi, Bernd Essigmann, Zhijin Fan, Marcus Fehr, Michael Flaeschel, A.J. Flemming, Raymonde Fonné-Pfister, Kosuke Fukatsu, Y. Furukawa, Stephanie Gary, Birgit Gockel, C.R. Godfrey, E. Godineau, Edouard Godineau, Aiying Guan, Oliver Gutbrod, Hans Ulrich Haas, Takahiro Hamada, Taku Hamamoto, M. Hamer, Nick Hamon, Hiroto Harayama, Patrick L. Havens, Hong-Wu He, Ron Heemstra, Yewande T. Henry, Katrin Hermann, Rafael Herrera, Jessica Herrick, Kangetsu Hirase, Akihiro Hisamatsu, Patrik Hoegger, Caleb W. Holyoke, M. Hoppé, O. Hueter, Kenneth A. Hughes, James S. Hunter, Nikolas Huwyler, Takuya Inoue, Mai Ito, Fukumatsu Iwahashi, M. Iwasa, Atsushi Iwata, Haowu Jia, David Jones, Junji Kadotani, Ryota Kasahara, H. Katsuta, A. Kawahara, So Kiguchi, T. Kikuchi, Jochen Kleemann, D.P. Kloer, Y. Kobayashi, M. Komoda, Christopher Koradin, Toru Koyanagi, Tina Kyndt, Mathilde Lachia, George P. Lahm, Mukul Lal, Clemens Lamberth, Peter Lancashire, Laura A. Laughlin, Robert M. Leighty, BaoJu Li, Honglin Li, Pengfei Li, Wei Li, Yongqiang Li, Zhong Li, Hong-Yan Lin, Changling Liu, Brian A. Loy, Aidang Lu, Yu Lu, Torsten Luksch, Alexandre Lumbroso, Hongjuan Ma, Peter Maienfisch, Sven Mangelinckx, Pamela G. Marrone, Simonetta Masala, M. Matsumoto, Yuichi Matsuzaki, Michael Maue, Stephen F. McCann, Charles Meng, Giovanna Meregalli, Kevin G. Meyer, Anna Michrowska-Pianowska, Thomas Mietzner, T. Mita, S. Mitani, Andrea Molt, Mauricio Morell, Masayuki Morita, M. Muehlebach, Tetsuya Murata, Kenichi Nakamoto, Y. Nakamura, T. Nakao, Jia-Xu Nan, Trevor Newton, Yoshihiko Nokura, M. Nomura, R. Nourani, S. Oliver, Satoshi Ōmura, Kazuhiko Oyama, Thomas F. Pahutski, Sabitha Papineni, Rupesh Patre, Ralph Paulini, Hao Peng, F. Perruccio, Thomas Pitterna, Matthias Pohlman, C. Popp, Aimone Porri, C.S. Prasanna, Xuhong Qian, Ren-Yu Qu, Ramya Rajan, Nancy B. Rankl, Girish Rawal, Stefano Rendine, Peter Renold, Jared Rigoli, Johannes Röckl, Hiroshi Sakaguchi, Vincent L. Salgado, Eikoh Satoh, J. Schaetzer, Hartwig Schröder, Hans-Georg Schwarz, Claudio Screpanti, Thomas Seitz, R. Senn, Guomin Shan, Xusheng Shao, Hongfeng Shen, Ellie Sherrard-Smith, Qinjie Shi, Yanxia Shi, Yoshio Shigematsu, Mamiko Shino, Helge Sierotzki, Anja Simon, R. Slater, Tomas Smejkal, Helmars Smits, Sebastian Soergel, Hongjian Song, D. Stafford, Daniel Stierli, Daniel Strickman, Sarah Sulzer-Mosse, Akiyuki Suwa, Masaki Takahashi, Xiao-song Tan, Helen Tinwell, My-Hanh T. Tong, Masamitsu Tsukamoto, Yoshihisa Tsukamoto, S. Tsukuda, Bartel Vanholme, Russell Viner, F. Vock-Hatt, Juliane Vogt, T. Wakita, Harald Walter, Gaolei Wang, Nick X. Wang, Qingmin Wang, Tao Wang, Ziwen Wang, P. Wege, Monte R. Weimer, J. Wenger, L. Wildsmith, Derek W. Willis, Jeremy Wilmot, Christian Winter, Matthias Witschel, Qiao Wu, Youxin Xiao, Ming Xu, Xiaoyong Xu, Yufang Xu, Zheng Xu, Hiroji Yamada, Yao-Chao Yan, Guang-Fu Yang, Jichun Yang, Wen-Chao Yang, Chenglin Yao, T. Yoneda, Yuya Yoshimoto, David Young, Jun-Lin Yuan, W. Zambach, Jingjing Zhang, Jingwei Zhang, Ruifeng Zhang, Wenming Zhang, Bin Zhao, Zhenjiang Zhao, Cong Zhou, Yuan Zhou, Weiping Zhu

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::9c77cfbc3b2cba7962ef272ee1a88f31
https://doi.org/10.1016/b978-0-12-821035-2.00051-6

Nickel powder promoted 5-endo radical cyclisations. A concise approach to Erythrina alkaloids

Autor: Jérôme Cassayre, Béatrice Quiclet-Sire, Jean-Baptiste Saunier, Samir Z. Zard

Publikováno v: Tetrahedron Letters. 39:8995-8998

N-Alkenyl trichloroacetamides 3 undergo, upon refluxing with nickel powder and acetic acid in 2-propanol, exclusive 5-endo-trig cyclisation to afford functionalised lactams 4; these are attractive precursors of erythrina alkaloids, as demonstrated by

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::c41c410cc0985d668d3895c17d10343c
https://doi.org/10.1016/s0040-4039(98)02036-x

Amidyls in radical cascades. The total synthesis of (+/-)-aspidospermidine and (+/-)-13-deoxyserratine

Autor: Jérôme Cassayre, Anne-Claude Callier-Dublanchet, Samir Z. Zard, Béatrice Quiclet-Sire, Fabien Gagosz, Lisa A. Sharp

Publikováno v: Tetrahedron
Tetrahedron, Elsevier, 2008, 64 (21), pp.4803-4816. ⟨10.1016/j.tet.2008.02.107⟩

Concise routes to aspidospermidine and 13-deoxyserratine are described, hinging on a cascade starting from an amidyl radical and allowing the construction of the key indolizidine cores in one step.

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b961480cb32f48100401f39e9365e09b
https://hal.archives-ouvertes.fr/hal-00322556

Influence of copper(II) acetate on Ni/AcOH-promoted 5-endo and 5-exo radical cyclisations of trichloroacetamides

Autor: Samir Zard, Jérôme Cassayre, Delphine Dauge

Publikováno v: SYNLETT
SYNLETT, Georg Thieme Verlag, 2000, pp.471-474. ⟨10.1055/s-2000-6556⟩

International audience; Incorporation of Cu(OAc)2 as oxidant in Ni/AcOH-promoted 5-endo radical cyclisations of N-alkenyl-trichloroacetamides allows an interesting control of the oxidation level of the products, as illustrated by the conversion of 3

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e35fba64c0705ca6f624e161678fa6ae
https://hal-polytechnique.archives-ouvertes.fr/hal-00954902