Zobrazeno 1 - 6
of 6
pro vyhledávání: '"Isabelle Forfar-Bares"'
Autor:
Christian Jarry, Jean Guillon, Jean-Michel Léger, Jean-Jacques Bosc, Ouro-Sama Adetchessi, Isabelle Forfar-Bares
Publikováno v:
Tetrahedron. 61:4453-4460
2-Substituted-4a-hydroxy-9H-cycloalkyl[1,2-e]oxazolo[3,2-a]pyrimidin-9-ones 2a–c were synthesized by an one-step cyclocondensation from the 5-substituted-2-amino-2-oxazolines 1a–c with ethyl 2-oxocyclohexanecarboxylate in ethanol at room temperat
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::29dfebf570eea297b196bdecfeeee875
https://doi.org/10.1016/j.tet.2005.02.079
https://doi.org/10.1016/j.tet.2005.02.079
Autor:
Daniel-Henri Caignard, Claudine Quentin, Stéphane Moreau, Corinne Arpin, Jean Guillon, Christian Jarry, Jean Grellet, Boubakar B. Ba, Isabelle Forfar-Bares, Céline Vidaillac
Publikováno v:
Antimicrobial agents and chemotherapy. 51(3)
A series of 11 pyrrolo[1,2- a ]quinoxaline derivatives, 1a to 1k, sharing structural analogies with omeprazole, a eukaryotic efflux pump inhibitor (EPI) used as an antiulcer agent, was synthesized. Their inhibitory effect was evaluated using Staphylo
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::66fff3d3def9758c782a47f7df6a2510
https://pubmed.ncbi.nlm.nih.gov/17101679
https://pubmed.ncbi.nlm.nih.gov/17101679
Autor:
Natascha Chavain, Christophe Biot, Cheikh M. N'Diaye, Patricia Melnyk, Jamal Khalife, Alain Pellet, Christian Jarry, Jacques Brocard, Lydie Pelinski, Isabelle Forfar-Bares, Daniel Dive, Wassim Daher, Bruno Pradines, Laurent Fraisse
Publikováno v:
Journal of Medicinal Chemistry
Journal of Medicinal Chemistry, American Chemical Society, 2006, 49, pp.4707-4714. ⟨10.1021/jm060259d⟩
Journal of Medicinal Chemistry, 2006, 49, pp.4707-4714. ⟨10.1021/jm060259d⟩
Journal of Medicinal Chemistry, American Chemical Society, 2006, 49, pp.4707-4714. ⟨10.1021/jm060259d⟩
Journal of Medicinal Chemistry, 2006, 49, pp.4707-4714. ⟨10.1021/jm060259d⟩
A new therapeutic approach to malaria led to the discovery of ferroquine (FQ, SR97276). To assess the importance of the linkage of the ferrocenyl group to a 4-aminoquinoline scaffold, two series of 4-aminoquinolines, structurally related to FQ, were
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d48cbd66cfa5d3e1dec078dd4c02cae9
https://hal.archives-ouvertes.fr/hal-00097346
https://hal.archives-ouvertes.fr/hal-00097346
Autor:
Nicoletta Basilico, Christophe Biot, Lucien A. Maciejewski, Guy Nowogrocki, Jacques Brocard, Timothy J. Egan, Piero Olliaro, Mlandzeni Boyce, Isabelle Forfar-Bares, Donatella Taramelli
Publikováno v:
Molecular Pharmaceutics
Molecular Pharmaceutics, American Chemical Society, 2005, 2, pp.185. ⟨10.1021/mp0500061⟩
Molecular Pharmaceutics, 2005, 2, pp.185. ⟨10.1021/mp0500061⟩
Molecular Pharmaceutics, American Chemical Society, 2005, 2, pp.185. ⟨10.1021/mp0500061⟩
Molecular Pharmaceutics, 2005, 2, pp.185. ⟨10.1021/mp0500061⟩
Ferroquine (FQ) is a 4-aminoquinoline antimalarial which contains a quinoline nucleus similar to chloroquine, but a novel ferrocenic group in its side chain. Previous work has demonstrated that this compound has excellent activity against malaria par
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b62ed59b66bae55e7295e1f40fc89ce2
https://hal.archives-ouvertes.fr/hal-00100334
https://hal.archives-ouvertes.fr/hal-00100334
Publikováno v:
Journal of pharmaceutical and biomedical analysis. 36(4)
A rapid and sensitive high-performance liquid chromatography method with UV detection was developed for the determination of clonazepam in human plasma using 3-methylclonazepam, as internal standard. A one-step extraction of both compounds was perfor
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ae3e2ed55c75aa983bbf3d4c0f78ffdb
https://pubmed.ncbi.nlm.nih.gov/15533681
https://pubmed.ncbi.nlm.nih.gov/15533681
Autor:
Stéphane Massip, Pascal Sonnet, Jean-Michel Léger, Jean Guillon, Stéphane Moreau, Philippe Grellier, Christian Jarry, Isabelle Forfar-Bares
Publikováno v:
Analytical Sciences: X-ray Structure Analysis
Analytical Sciences: X-ray Structure Analysis Online, 2005, 21, pp.x209-x210. ⟨10.2116/analscix.21.x209⟩
Analytical Sciences: X-ray Structure Analysis Online, 2005, 21, pp.x209-x210. ⟨10.2116/analscix.21.x209⟩
The X-ray crystal structure of the antimalarial bis{N-(pyrrolo[1,2-a]quinoxalin-4-yl)-3-aminopropyl}piperazine was established. It crystallizes in the monoclinic space group P21/c. Solid-state data could be used to enlighten the mechanism of action,
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0af05a2610b9b14e9bb0d4d877e4abb7
https://doi.org/10.2116/analscix.21.x209
https://doi.org/10.2116/analscix.21.x209