Zobrazeno 1 - 4
of 4
pro vyhledávání: '"Isabelle Daffix"'
Autor:
Jean Martinez, Jean-Michel Luccarini, Pierre Dodey, Isabelle Daffix, Jean-Luc Paquet, Muriel Amblard, Philippe Bedos, Didier Pruneau, Christophe Olivier
Publikováno v:
Journal of Medicinal Chemistry. 43:2382-2386
We recently described a potent bradykinin B(2) receptor agonist (JMV1116) obtained by replacing the D-Tic-Oic dipeptide moiety of HOE140 by a (3S)-amino-5-(carbonylmethyl)-2,3-dihydro-1, 5-benzothiazepin-4(5H)-one (D-BT) moiety. This compound inhibit
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4f48b33620d57e24ae2cbfaa18af8f2d
https://doi.org/10.1021/jm990961s
https://doi.org/10.1021/jm990961s
Autor:
Jean Martinez, Monique Calmes, Didier Pruneau, Isabelle Daffix, Muriel Amblard, Pierre Bélichard, Pierre Dodey, Jean-Luc Paquet, Gilbert Bergé, Jean-Michel Luccarini
Publikováno v:
Journal of Medicinal Chemistry. 42:4193-4201
We have previously shown that substitution of the D-Tic-Oic dipeptide by a (3S)-[amino]-5-(carbonylmethyl)-2,3-dihydro-1, 5-benzothiazepin-4(5H)-one (D-BT) moiety in the bradykinin B(2) receptor antagonist HOE 140 resulted in a full potent and select
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3fdb681fd38cee46725c5e66488a959e
https://doi.org/10.1021/jm9901531
https://doi.org/10.1021/jm9901531
Autor:
Jean Martinez, Pierre Bélichard, Jean-Luc Paquet, Pierre Dodey, Didier Pruneau, Gilbert Bergé, Isabelle Daffix, Philippe Bedos, Muriel Amblard, Jean-Michel Luccarini
Publikováno v:
Journal of Medicinal Chemistry. 42:4185-4192
A bradykinin analogue (H-Arg-Pro-Pro-Gly-Phe-Ser-D-BT-Arg-OH, 3) in which the Pro-Phe dipeptide was replaced by the (3S)[amino]-5-(carbonylmethyl)-2,3-dihydro-1, 5-benzothiazepin-4(5H)-one (D-BT) moiety has been synthesized. The same modification was
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fe1c133b8ba3c3e1b1343a027cbfa637
https://doi.org/10.1021/jm9901529
https://doi.org/10.1021/jm9901529
Autor:
Isabelle Daffix, Muriel Amblard, Jean-Michel Luccarini, Pierre Dodey, Pierre Bélichard, Didier Pruneau, Jean-Luc Paquet, Gilbert Bergé, Jean Martinez
Publikováno v:
Peptides Frontiers of Peptide Science ISBN: 9780792351603
Muriel Amblard, Isabelle Daffix, Gilbert Berge, Pierre Dodey, Didier Pruneau, Jean-Luc Paquet, Pierre Belichard, Jean-Michel Luccarini and Jean Martineza Laboratoire des Aminoacides Peptides et Proteines (LAPP), ESA CNRS 5075, Universites de Montpell
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::e3a699b32bf92a65051dc94ee49d6ab3
https://doi.org/10.1007/0-306-46862-x_34
https://doi.org/10.1007/0-306-46862-x_34
