Zobrazeno 1 - 10
of 50
pro vyhledávání: '"Imai, Minoru"'
Autor:
Mori, Masaaki, Yoshizaki, Kanako, Watabe, Shinichi, Ishige, Mika, Hinoki, Akinari, Kondo, Takuya, Taguchi, Tomoaki, Hasegawa, Hisaya, Hatata, Tomoko, Tanuma, Naoyuki, Kirino, Kosuke, Hirakawa, Akihiro, Naruto, Takuya, Imai, Minoru, Koike, Ryuji, Hosoi, Kenichiro, Kusuda, Satoshi
Publikováno v:
In The Lancet Regional Health - Western Pacific October 2023 39
Akademický článek
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Autor:
Yano Yoshiko, Toguchi Keisuke, Kino Shigeo, Hirabayashi Kuniaki, Imai Minoru, Yamaguchi Takuya, Toyama Kazutaka
Publikováno v:
Nihon Gekakei Rengo Gakkaishi (Journal of Japanese College of Surgeons). 45:37-45
Publikováno v:
Asian Journal of Endoscopic Surgery. May2017, Vol. 10 Issue 2, p219-222. 4p.
Akademický článek
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Publikováno v:
Asian Journal of Endoscopic Surgery; Jan2021, Vol. 14 Issue 1, p90-93, 4p
Publikováno v:
International Cancer Conference Journal; Jul2020, Vol. 9 Issue 3, p107-111, 5p
Autor:
Kenichiro Kataoka, Hiroaki Makino, Keiichiro Imaizumi, Brad Sherborne, Gen Unoki, Donald James Simpson, Naotaka Suzuki, C. John Harris, Richard K. Gordon, Tomomi Kosugi, Vicky Cunliffe, Heidi Kalloo-Hosein, Dale Robert Mitchell, Peter S Thomas, Kanji Komatsu, Midori Takimoto-Kamimura, Sugiura Satoshi, Mika Kambe, Yuri Sakai, Shinji Kobayashi, Aiko Fujino, Gita Patel, Yuko Yamakoshi, Julie A. Frearson, Oue Yasuhiro, Takenouchi Osami, Imai Minoru, Joelle Le, Yohei Matsueda
Publikováno v:
Journal of Medicinal Chemistry. 55:6700-6715
A novel class of mitogen-activated protein kinase-activated protein kinase 2 (MAPKAP-K2) inhibitors was discovered through screening a kinase-focused library. A homology model of MAPKAP-K2 was generated and used to guide the initial SAR studies and t
Autor:
Noriaki Endo, Wilna J. Moree, Yumiko Muroga, Christine M. Tarby, Dewey Fanning, Hada Takahiko, Imai Minoru, Kenichiro Kataoka, John Saunders, Yoshinori Kato, Peter Myers, Tatsuki Shiota, Masaki Sudo, Takaharu Tsutsumi, Michele M. Ramirez-Weinhouse
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 18:1869-1873
SAR studies were conducted around lead compound 1 using high-throughput parallel solution and solid phase synthesis. Our lead optimization efforts led to the identification of several CCR2b antagonists with potent activity in both binding and functio
Autor:
Imai Minoru, Peter Myers, Kenichiro Kataoka, Takaharu Tsutsumi, Michele M. Ramirez-Weinhouse, Noriaki Endo, Chung-Ming Sun, Masaki Sudo, Jonathan W. Greene, Wilna J. Moree, Doug Barnum, Tatsuki Shiota, Hada Takahiko, Hiroko Tanaka, Shinsuke Yamagami, Yoshinori Kato, Christine M. Tarby, John Saunders, Morita Takuya, Daniel D. Comer
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 14:5407-5411
N , N ′-Disubstituted homopiperazine derivatives have been discovered as CC-chemokine receptor 2b (CCR2b) inhibitors with submicromolar activity in the CCR2b binding assay. A 4-substituted benzyl group on one homopiperazine nitrogen was an importan