Zobrazeno 1 - 10
of 15
pro vyhledávání: '"IMAN A. AL-MASOUDI"'
Publikováno v:
Phosphorus, Sulfur, and Silicon and the Related Elements. 183:1571-1583
A series of new 5-nitro- and 5-amino-6-arylsulfanyl-1-propyl-1H-pyrimidin-2,4-diones (4–9) were synthesized with the aim to develop new non-nucleoside reverse transcriptase inhibitors (NNRTIs). Similarly, 6-arylsulfanyl-1,3-dimethyl-5-nitro-1H-pyri
Publikováno v:
Nucleosides, Nucleotides and Nucleic Acids. 27:146-156
A series of acyclonucleosides substituted 1-(4,5-dihydroxypentyl) (13-8) and 2-(4,5-dihydroxypentyloxy)quinoxalines (19-24) were synthesized by the sharpless asymmetric dihydroxylation of the derivatives 1-6 and 7-12, respectively. Treatment of the q
Publikováno v:
Chemistry of Heterocyclic Compounds. 43:1052-1059
A series of acyclonucleosides 6,7-disubstituted 1-(pent-4-enyl)quinoxalin-2-one derivatives and the O-analogs were synthesized by a one-step condensation of the corresponding quinoxaline bases with 5-bromo-1-pentene.The acyclonucleosides prepared wer
Publikováno v:
Chemistry of Heterocyclic Compounds. 42:1377-1403
The synthetic routes of 1,2,4-triazole compounds as well as their pharmacological properties have been described. The review focuses intensively on two methods: cycloaddition reaction in the syntheses of various 1,5-dialky-1H-1,2,4-triazole derivativ
Publikováno v:
Chemistry of Heterocyclic Compounds. 42:583-590
A variety of 7-[(1,5-dialkyl-1H-1,2,4-triazolyl)methoxy(and methyl)]coumarins were synthesized from cycloaddition of 2-(2H-benzopyran-7-yloxy)acetonitrile and 2-(5-methoxy-4-methyl-2H-benzopyran-7-yloxy)acetonitrile, respectively, with various reacti
Publikováno v:
Heteroatom Chemistry. 16:576-586
A series of peptide derivatives conjugated naphthalene residue 11–25, the glycoside 27 as well as the 7-glycoside 30, and the 2-(2-hydroxy-3-(N-benzyl-N-isopropylamino)propoxy)naphthalene bearing methionine 31 were synthesized. The new compounds we
Autor:
Iman A. Al-Masoudi
Publikováno v:
Phosphorus, Sulfur, and Silicon and the Related Elements. 178:2393-2402
Reaction of the 6-chloro-7-fluoroquinoline 7 with methyl 2-mercaptoacetate, methyl 3-mercaptopropionate, or sodium thiophenolate furnished the quinolone derivatives of 3-carbonylsulfanyl-acetic acid methyl ester 8, the propionoate analogue 10, and 3-
Autor:
Najim A. Al-Masoudi, Luma Sabri, Nahed H. Al-Haidery, Iman A. Al-Masoudi, Nawar S. Hamad, Mey Sabri
Publikováno v:
Archiv der Pharmazie. 343(7)
A new series of 2-(naphthalen-2-yloxy)-N-[(aryl-5-thioxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl] acetamides 5a-f was synthesized from naphthalene-derived glycine derivative 2 via the hydrazinoacetamide analogs 4a-f. Alternatively, treatment of 4a w
Publikováno v:
ChemInform. 39
A series of acyclonucleosides substituted 1-(4,5-dihydroxypentyl) (13-8) and 2-(4,5-dihydroxypentyloxy)quinoxalines (19-24) were synthesized by the sharpless asymmetric dihydroxylation of the derivatives 1-6 and 7-12, respectively. Treatment of the q
Publikováno v:
ChemInform. 39
A series of acyclonucleosides 6,7-disubstituted 1-(pent-4-enyl)quinoxalin-2-one derivatives and the O-analogs were synthesized by a one-step condensation of the corresponding quinoxaline bases with 5-bromo-1-pentene.The acyclonucleosides prepared wer