Zobrazeno 1 - 10
of 15
pro vyhledávání: '"I A, Vosekalna"'
Publikováno v:
Tetrahedron. 49:4671-4676
Synthesis of optically active 3-amino-2H-azirines using the modified Neber reaction has been carried out for the first time. The structure and absolute configuration of diastereomeric derivatives of 3-amino-2H-azirines have been determined.
Publikováno v:
ChemInform. 24
Synthesis of optically active 3-amino-2H-azirines using the modified Neber reaction has been carried out for the first time. The structure and absolute configuration of diastereomeric derivatives of 3-amino-2H-azirines have been determined.
Publikováno v:
Doklady Akademii nauk. 364(6)
Publikováno v:
Bioorganicheskaia khimiia. 21(4)
A cyclic analog of enkephalin, cyclo(Lys-Tyr-DMet-Gly-Phe-Pro-) and two corresponding linear hexapeptides with lysine residue on the N- and C-termini of the pentapeptide sequence, Lys-Tyr-DMet-Gly-Phe-Pro and Tyr-DMet-Gly-Phe-Pro-Lys were synthesized
Publikováno v:
Bioorganicheskaia khimiia. 16(3)
Five angiotensin cycloanalogues have been synthesised by classical methods of peptide chemistry, cyclisation being carried out via pentafluorophenyl esters. Cycloanalogues (I-IV) with a fixed potential turn in the C-terminal part of the angiotensin m
Autor:
I. A. Vosekalna, F. D. Polyak, R. G. Kostyanovskii, Sh. S. Nasibov, I. I. Chervin, A. V. Eremeev
Publikováno v:
Chemistry of Heterocyclic Compounds. 20:1102-1107
Individual diastereomers of a number of anilides of N-substituted aziridine-2-carboxylic acids have been obtained. Conclusions regarding the spatial structure of the compounds indicated have been drawn on the basis of the 1H NMR, 15N NMR, and CD spec
Autor:
M. A. Shokhen, G. V. Shustov, R. G. Kostyanovskii, Anton V. Eremeev, F. D. Polyak, R. K. Alekperov, I. A. Vosekalna, G. K. Kadorkina
Publikováno v:
Chemistry of Heterocyclic Compounds. 25:32-39
The optically active 1-acyl-substituted (1R,2R)-2-methyl- and (1R,2S)-2-methoxycarbonylaziridines were synthesized. The nonplanarity of the amide chromophore in them and its high conformational mobility, which was caused by the rotation around the N-
Autor:
I. A. Vosekalna, F. D. Polyak, R. G. Kostyanovskii, É. É. Liepin'sh, A. V. Eremeev, I. V. Solodin, I. I. Chervin
Publikováno v:
Chemistry of Heterocyclic Compounds. 21:1110-1113
Individual diastereomers of aziridine-2-carboxylic acid esters that contain R- and S-valine and R- and S-hexafluorovaline fragments were isolated by high-performance liquid chromatogrpahy (HPLC). The absolute configurations of both asymmetric centers
Publikováno v:
Bioorganicheskaia khimiia. 11(11)
The spatial structure of an enkephaline cycloanalogue Lys-Tyr-Gly-Gly-Phe-Leu--has been investigated by means of energy calculations, fluorescence and CD-spectroscopy. Despite the high conformational mobility of the cycloanalogue, little resemblance
Publikováno v:
Bioorganicheskaia khimiia. 11(9)
Using solid-phase approach, new cyclic and linear analogues of C-terminal neurotensin (NT) fragments were synthesized and their vasodepressor and miotropic activities were assayed. The cyclic structures were fixed by a peptide bond linking the lysine