Zobrazeno 1 - 10
of 20
pro vyhledávání: '"Hongmok Kwon"'
Autor:
Seulgi Lee, Bernie Byeonghoon Park, Hongmok Kwon, Vitchan Kim, Jang Su Jeon, Rowoon Lee, Milan Subedi, Taehyeong Lim, Hyunsoo Ha, Dongju An, Jaehoon Kim, Donghak Kim, Sang Kyum Kim, Seyun Kim, Youngjoo Byun
Publikováno v:
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 37, Iss 1, Pp 269-279 (2022)
Inositol hexakisphosphate kinase (IP6K) is an important mammalian enzyme involved in various biological processes such as insulin signalling and blood clotting. Recent analyses on drug metabolism and pharmacokinetic properties on TNP (N2-(m-trifluoro
Externí odkaz:
https://doaj.org/article/b92d8702f213451b962add5ca26a8351
Publikováno v:
Expert Opinion on Therapeutic Patents. 31:525-547
Prostate-specific membrane antigen (PSMA), also known as glutamate carboxypeptidase II, is a potential target protein for imaging and treatment of patients with prostate cancer because of its overexpression during metastasis. Various PSMA-targeted im
Autor:
Hongmok Kwon, Youngjoo Byun, Han Shin Kim, Sang Hyun Son, Suhyun Moon, Taehyeong Lim, So Young Ham, Jeong Hoon Lee, Hee Deung Park, Sang Jin Nam
Publikováno v:
Journal of Medicinal Chemistry. 63:8388-8407
Pseudomonas aeruginosa (P. aeruginosa) is an opportunistic human pathogen that forms biofilms and produces virulence factors via quorum sensing (QS). Blocking the QS system in P. aeruginosa is an e...
Autor:
Xing Yang, Xiaojiang Duan, Futao Liu, Youngjoo Byun, Hongmok Kwon, Jingming Zhang, Martin G. Pomper, Xi Zhen, Il Minn, Xuekang Cai, Yang Zhi
Publikováno v:
Journal of Medicinal Chemistry. 63:3563-3576
In an effort to seek novel agents targeting prostate-specific membrane antigen (PSMA), 16 ligands (L1-L16) with structural modifications in S1' binding pocket were synthesized and evaluated for PSMA inhibition. (S)-3-(Carboxyformamido)-2-(3-(carboxym
Autor:
Seulgi Lee, Bernie Byeonghoon Park, Hongmok Kwon, Vitchan Kim, Jang Su Jeon, Rowoon Lee, Milan Subedi, Taehyeong Lim, Hyunsoo Ha, Dongju An, Jaehoon Kim, Donghak Kim, Sang Kyum Kim, Seyun Kim, Youngjoo Byun
Publikováno v:
Journal of Enzyme Inhibition and Medicinal Chemistry
article-version (VoR) Version of Record
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 37, Iss 1, Pp 269-279 (2022)
article-version (VoR) Version of Record
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 37, Iss 1, Pp 269-279 (2022)
Inositol hexakisphosphate kinase (IP6K) is an important mammalian enzyme involved in various biological processes such as insulin signalling and blood clotting. Recent analyses on drug metabolism and pharmacokinetic properties on TNP (N2-(m-trifluoro
Publikováno v:
Asian Journal of Organic Chemistry. 8:1588-1600
Autor:
Jaebong Jang, Song-Kyu Park, Youngjoo Byun, Hongmok Kwon, Sang-Hyun Son, Hyunsoo Ha, Kiho Lee, Hayoung Jeon
Publikováno v:
Bioorganic chemistry. 107
Hepsin is a type II transmembrane serine protease (TTSP) associated with cell proliferation and overexpressed in several types of cancer including prostate cancer (PCa). Because of its significant role in cancer progression and metastasis, hepsin is
Autor:
SangJin, Nam, So-Young, Ham, Hongmok, Kwon, Han-Shin, Kim, Suhyun, Moon, Jeong-Hoon, Lee, Taehyeong, Lim, Sang-Hyun, Son, Hee-Deung, Park, Youngjoo, Byun
Publikováno v:
Journal of medicinal chemistry. 63(15)
Autor:
Youngjoo Byun, Hwanhee Nam, Hyunwoong Lim, Sang Hyun Son, Hongmok Kwon, Hyunsoo Ha, Doyoung Choi, Il Minn
Publikováno v:
Bioorganic chemistry. 104
Prostate-specific membrane antigen (PSMA), a type II membrane glycoprotein, is considered an excellent target for the diagnosis or treatment of prostate cancer. We previously investigated the effect of β- and γ-amino acids with (S)- or (R)-configur
Autor:
Jeong Hoon Park, Youngjoo Byun, Hee Deung Park, So Young Ham, Sang Jin Nam, Han Shin Kim, Eunji Cha, Hongmok Kwon
Publikováno v:
Biotechnology and bioengineeringREFERENCES. 118(1)
Bacterial biofilm formation causes serious problems in various fields of medical, clinical, and industrial settings. Antibiotics and biocide treatments are typical methods used to remove bacterial biofilms, but biofilms are difficult to remove effect