Zobrazeno 1 - 4
of 4
pro vyhledávání: '"Hollis C. Tomaselli"'
Autor:
Nicholas Marcopulos, Gary M. Coppola, Beatriz Dardik, Paivi J. Kukkola, Jenny Tan, Hua Wang, Ricardo E. Chatelain, James L. Stanton, Alan D. Neubert, Natalie A. Bilci, Thomas D. Aicher, Arco Y. Jeng, Hollis C. Tomaselli, Douglas C. Knorr
Publikováno v:
Journal of Medicinal Chemistry. 48:6696-6712
High-throughput screening identified 5 as a weak inhibitor of 11beta-HSD1. Optimization of the structure led to a series of perhydroquinolylbenzamides, some with low nanomolar inhibitory potency. A tertiary benzamide is required for biological activi
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5abb3ffe30f7a8d7d4ca7e3980f503c2
https://doi.org/10.1021/jm058228q
https://doi.org/10.1021/jm058228q
Autor:
Zouhair F. Stephan, Ronald Dotson, Steele Ronald Edward, Jong M. Wasvary, Edna Cahill, Hollis C. Tomaselli, James L. Stanton, Jenny Tan
Publikováno v:
ChemInform. 31
The synthesis of substituted phenoxyphenyl oxamic acid derivatives related to l -thyronine ( l -T3) is described. The in vitro and in vivo cholesterol lowering and cardiovascular effects of these compounds are presented and discussed.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::d67d8c6525e856bccd91d9461c1f9784
https://doi.org/10.1002/chin.200044207
https://doi.org/10.1002/chin.200044207
Autor:
Jong M. Wasvary, Zouhair F. Stephan, James L. Stanton, Steele Ronald Edward, Ronald Dotson, Edna Cahill, Jenny Tan, Hollis C. Tomaselli
Publikováno v:
Bioorganicmedicinal chemistry letters. 10(15)
The synthesis of substituted phenoxyphenyl oxamic acid derivatives related to l -thyronine ( l -T3) is described. The in vitro and in vivo cholesterol lowering and cardiovascular effects of these compounds are presented and discussed.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::66a6d8b6d0814cda91a5737acef3fa73
https://pubmed.ncbi.nlm.nih.gov/10937719
https://pubmed.ncbi.nlm.nih.gov/10937719
Autor:
Mahesh Desai, Watthey Jeffrey W H, Barbara M. Finn, Joseph E. Babiarz, James L. Stanton, Hollis C. Tomaselli
Publikováno v:
Chemischer Informationsdienst. 17
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::73ce9fbbcec748c3d802c942e04805eb
https://doi.org/10.1002/chin.198609194
https://doi.org/10.1002/chin.198609194