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pro vyhledávání: '"Hiromi Kaku"'
Autor:
Shoki Okuda, Minoru Ikoma, Masashi Takahashi, Shizuo Kasai, Yasutaka Nagisa, Hiromi Kaku, Syunsuke Yamamoto, Tsuyoshi Maekawa, Toshihiro Noguchi, Asato Kina, Keiko Kakegawa, Natsu Hotta, Yayoi Kawata, Hideyuki Igawa, Jumpei Aida, Masaharu Nakayama
Publikováno v:
Bioorganic & Medicinal Chemistry. 24:2504-2518
To develop non-basic melanin-concentrating hormone receptor 1 (MCHR1) antagonists with a high probability of target selectivity and therapeutic window, we explored neutral bicyclic motifs that could replace the previously reported imidazo[1,2-a]pyrid