Tyrosinase Inhibition and Antimelanogenic Effects of Resorcinol-Containing Compounds.

Autor: Beaumet M; Univ. Grenoble Alpes, CNRS, DPM, 38000, Grenoble, France., Lazinski LM; Univ. Grenoble Alpes, CNRS, DPM, 38000, Grenoble, France.; Univ. Grenoble Alpes, CNRS, DCM, 38000, Grenoble, France., Maresca M; Aix Marseille Univ., CNRS, Centrale Marseille, iSm2, 13013, Marseille, France., Haudecoeur R; Univ. Grenoble Alpes, CNRS, DPM, 38000, Grenoble, France.

Publikováno v: ChemMedChem [ChemMedChem] 2024 Dec 02; Vol. 19 (23), pp. e202400314. Date of Electronic Publication: 2024 Sep 30.

Design and Synthesis of Novel Amino and Acetamidoaurones with Antimicrobial Activities.

Autor: Di Maio A; Aix Marseille University, University Avignon, CNRS, IRD, IMBE, 13013 Marseille, France., Olleik H; Aix Marseille University, CNRS, Centrale Marseille, iSm2, 13013 Marseille, France., Courvoisier-Dezord E; Aix Marseille University, CNRS, Centrale Marseille, iSm2, 13013 Marseille, France., Guillier S; Aix Marseille University, INSERM, SSA, MCT, 13385 Marseille, France., Neulat-Ripoll F; Aix Marseille University, INSERM, SSA, MCT, 13385 Marseille, France., Haudecoeur R; University Grenoble Alpes, CNRS, DPM, 38000 Grenoble, France., Bolla JM; Aix Marseille University, INSERM, SSA, MCT, 13385 Marseille, France., Casanova M; Aix-Marseille University, CNRS, LISM UMR7255, IMM FR3479, 13009 Marseille, France., Cavalier JF; Aix-Marseille University, CNRS, LISM UMR7255, IMM FR3479, 13009 Marseille, France., Canaan S; Aix-Marseille University, CNRS, LISM UMR7255, IMM FR3479, 13009 Marseille, France., Pique V; Aix Marseille University, University Avignon, CNRS, IRD, IMBE, 13013 Marseille, France., Charmasson Y; Aix Marseille University, CNRS, Centrale Marseille, iSm2, 13013 Marseille, France., Baydoun E; Department of Biology, American University of Beirut, Beirut 1107, Lebanon., Hijazi A; Plateforme de Recherche et D'analyse en Sciences de L'environnement (EDST-PRASE), Beirut 1107, Lebanon., Perrier J; Aix Marseille University, CNRS, Centrale Marseille, iSm2, 13013 Marseille, France., Maresca M; Aix Marseille University, CNRS, Centrale Marseille, iSm2, 13013 Marseille, France., Robin M; Aix Marseille University, University Avignon, CNRS, IRD, IMBE, 13013 Marseille, France.

Publikováno v: Antibiotics (Basel, Switzerland) [Antibiotics (Basel)] 2024 Mar 26; Vol. 13 (4). Date of Electronic Publication: 2024 Mar 26.

Aurones and derivatives as promising New Delhi metallo-β-lactamase (NDM-1) inhibitors.

Autor: Caburet J; Univ. Grenoble Alpes, CNRS, DPM, 38000 Grenoble, France., Verdirosa F; Dipartimento di Biotecnologie Mediche, Università degli Studi di Siena, 53100 Siena, Italy., Moretti M; Univ. Grenoble Alpes, CNRS, DPM, 38000 Grenoble, France., Roulier B; Univ. Grenoble Alpes, CNRS, DPM, 38000 Grenoble, France., Simoncelli G; Dipartimento di Biotecnologie Mediche, Università degli Studi di Siena, 53100 Siena, Italy., Haudecoeur R; Univ. Grenoble Alpes, CNRS, DPM, 38000 Grenoble, France., Ghazi S; Univ. Grenoble Alpes, CNRS, DPM, 38000 Grenoble, France., Jamet H; Univ. Grenoble Alpes, CNRS, DCM, 38000 Grenoble, France., Docquier JD; Dipartimento di Biotecnologie Mediche, Università degli Studi di Siena, 53100 Siena, Italy; Laboratoire de Bactériologie Moléculaire, UR-InBioS, Université de Liège, 4000 Liège, Belgium., Boucherle B; Univ. Grenoble Alpes, CNRS, DPM, 38000 Grenoble, France., Peuchmaur M; Univ. Grenoble Alpes, CNRS, DPM, 38000 Grenoble, France. Electronic address: marine.peuchmaur@univ-grenoble-alpes.fr.

Publikováno v: Bioorganic & medicinal chemistry [Bioorg Med Chem] 2024 Jan 01; Vol. 97, pp. 117559. Date of Electronic Publication: 2023 Dec 12.

Resorcinol-based hemiindigoid derivatives as human tyrosinase inhibitors and melanogenesis suppressors in human melanoma cells.

Autor: Roulier B; Univ. Grenoble Alpes, CNRS 5063, DPM, 38000, Grenoble, France., Rush I; Department of Biotechnology and Food Engineering, Technion - Israel Institute of Technology, Haifa, 3200003, Israel., Lazinski LM; Univ. Grenoble Alpes, CNRS 5063, DPM, 38000, Grenoble, France; Univ. Grenoble Alpes, CNRS 5250, DCM, 38000, Grenoble, France., Pérès B; Univ. Grenoble Alpes, CNRS 5063, DPM, 38000, Grenoble, France., Olleik H; Aix Marseille Univ., CNRS, Centrale Marseille, iSm2, 13397, Marseille, France., Royal G; Univ. Grenoble Alpes, CNRS 5250, DCM, 38000, Grenoble, France., Fishman A; Department of Biotechnology and Food Engineering, Technion - Israel Institute of Technology, Haifa, 3200003, Israel., Maresca M; Aix Marseille Univ., CNRS, Centrale Marseille, iSm2, 13397, Marseille, France., Haudecoeur R; Univ. Grenoble Alpes, CNRS 5063, DPM, 38000, Grenoble, France. Electronic address: Romain.Haudecoeur@univ-grenoble-alpes.fr.

Publikováno v: European journal of medicinal chemistry [Eur J Med Chem] 2023 Jan 15; Vol. 246, pp. 114972. Date of Electronic Publication: 2022 Nov 28.

Design, Synthesis, Structural Insights, Tyrosinase Inhibition, and Sun Protection Factor of New Thiosemicarbazone Derivatives.

Autor: Masuri, Sebastiano¹ (AUTHOR) sebastiano.masuri@unica.it, Era, Benedetta² (AUTHOR) era@unica.it, Pintus, Francesca² (AUTHOR) fpintus@unica.it, Floris, Sonia² (AUTHOR) s.floris@unica.it, Meloni, Francesca¹ (AUTHOR) francesca.meloni96t@unica.it, Pettinau, Francesca¹ (AUTHOR) francesca.pettinau@unica.it, Podda, Enrico³ (AUTHOR) enrico.podda@unica.it, Cabiddu, Maria Grazia¹ (AUTHOR) mgcabidd@unica.it, Fais, Antonella² (AUTHOR) fais@unica.it, Pivetta, Tiziana¹ (AUTHOR) fais@unica.it

Publikováno v: Molecules. Dec2024, Vol. 29 Issue 23, p5629. 19p.