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ChemInform Abstract: Characterization of Potent and Selective Antagonists at Postsynaptic 5- HT1A Receptors in a Series of N4-Substituted Arylpiperazines

Autor: Valérie Audinot, Millan Mark, Alain Gobert, Mauricette Brocco, K Bervoets, S Le Marouille-Girardon, H Canton, Jean-Louis Peglion

Publikováno v: ChemInform. 27

Benzocycloalkyl and benzocycloalkenyl moities linked, directly or via an alkyl chain, to oxygen-bearing heteroarylpiperazines were synthesized, in an attempt to obtain potent and selective antagonists at postsynaptic 5-HT 1A receptors. From the numer

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::3e94cf15c7824413d41583c98b721f8d
https://doi.org/10.1002/chin.199604185

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Identification, molecular cloning, and distribution of a short variant of the 5-hydroxytryptamine2C receptor produced by alternative splicing

Autor: H, Canton, R B, Emeson, E L, Barker, J R, Backstrom, J T, Lu, M S, Chang, E, Sanders-Bush

Publikováno v: Molecular pharmacology. 50(4)

The actions of the neurotransmitter 5-hydroxytryptamine (5-HT) (serotonin) are mediated by multiple receptor subtypes. One of the prominent serotonin receptors in the brain is the 5-HT2C receptor (5-HT2C-R). We report the occurrence of a second 5-HT2

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::67e1d767492e54eb37fd74ec677792c2
https://pubmed.ncbi.nlm.nih.gov/8863824

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The Economics of Living with Citrus Viroids in Belize

Autor: C. N. Roistacher, P. S. Reddy, H. Canton

Publikováno v: Roistacher, C. N.; Canton, H.; & Reddy, P. S.(1996). The Economics of Living with Citrus Viroids in Belize. International Organization of Citrus Virologists Conference Proceedings (1957-2010), 13(13), 370-375. Retrieved from: http://www.escholarship.org/uc/item/67r551kp

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::219ae5b2c32a9af94774ae8add00cdf5
https://doi.org/10.5070/c567r551kp

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5-HT1A receptors and the tail-flick response. VI. Intrinsic alpha 1A-adrenoceptor antagonist properties can mask the actions of 5-HT1A receptor agonists in the spontaneous tail-flick paradigm

Autor: M J, Millan, J M, Rivet, A, Gobert, H, Canton, S, Veiga, K, Bervoets

Publikováno v: The Journal of pharmacology and experimental therapeutics. 269(1)

In view of the involvement of central alpha 1-adrenoceptors in the expression of 5-HT1A receptor-mediated spontaneous tail-flicks (STFs) in the rat, this study examined whether the putative alpha 1-adrenoceptor antagonist (alpha 1-antagonist) propert

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::84354f8bd17945a9b5efa5b49176f5bc
https://pubmed.ncbi.nlm.nih.gov/7909555

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Presentation of a general algorithm to include effect assessment on secondary poisoning in the derivation of environmental quality criteria. 2. Terrestrial food chains

Autor: C A, Romijn, R, Luttik, J H, Canton

Publikováno v: Ecotoxicology and environmental safety. 27(2)

In a previous study a simple algorithm was presented for effect assessment on secondary poisoning of birds and mammals. This algorithm (MPC = NOECfish-eater/BCFfish) was drawn up by analyzing a two-step aquatic food chain (water-fish-bird/mammal). Th

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::e6e1268a4170fac3ac0a7cdd33b784df
https://pubmed.ncbi.nlm.nih.gov/7516280

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Novel benzodioxopiperazines acting as antagonists at postsynaptic 5-HT1A receptors and as agonists at 5-HT1A autoreceptors: a comparative pharmacological characterization with proposed 5-HT1A antagonists

Autor: M J, Millan, H, Canton, A, Gobert, F, Lejeune, J M, Rivet, K, Bervoets, M, Brocco, P, Widdowson, T, Mennini, V, Audinot

Publikováno v: The Journal of pharmacology and experimental therapeutics. 268(1)

The novel benzodioxopiperazines [4-(benzodioxan-5-yl)1-[2- (benzocyclobutane-1-yl)ethyl]piperazine] (S 14489), [4-(benzodioxan-5-yl)1-(indan-2-yl)piperazine)] (S 15535) and [4-(benzodioxan-5-yl)1-[2(indan-1-yl)ethyl]piperazine (S15931) competitively

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::cc71d3ec2eee71f4f1d45e90f9d2051b
https://pubmed.ncbi.nlm.nih.gov/8301575

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S 14671: a naphtylpiperazine 5-hydroxytryptamine1A agonist of exceptional potency and high efficacy possessing antagonist activity at 5-hydroxytryptamine1C/2 receptors

Autor: M J, Millan, J M, Rivet, H, Canton, F, Lejeune, K, Bervoets, M, Brocco, A, Gobert, B, Lefebvre de Ladonchamps, S, Le Marouille-Girardon, L, Verriele

Publikováno v: The Journal of pharmacology and experimental therapeutics. 262(2)

The interaction at 5-hydroxytryptamine (5-HT) receptors of the novel naphtylpiperazine, S 14671 (1-[2-(2-thenoylamino)ethyl]-4[1-(7- methoxynaphtyl)]piperazine), was compared to that of the 5-HT1A ligands, 8-hydroxy-2-(di-n-propylamino)tetralin hydro

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::819996eda810ee1a949cef6f921c98f7
https://pubmed.ncbi.nlm.nih.gov/1323650

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Histopathological effects in Poecilia reticulata (guppy) exposed to methyl mercury chloride

Autor: Piet Wester, Hans H. Canton

Publikováno v: Toxicologic pathology. 20(1)

To evaluate the usefulness of histopathology in aquatic toxicity testing, studies were carried out on the small freshwater fish Poecilia reticulata (guppy) following aqueous methyl mercury chloride exposure. Fish were exposed to concentrations of 0,

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7b535940dcfcd49fb6a124cc9950905e
https://pubmed.ncbi.nlm.nih.gov/1411135

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