SR147778 [5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-ethyl-N-(1-piperidinyl)-1H-pyrazole-3-carboxamide], a new potent and selective antagonist of the CB1 cannabinoid receptor: biochemical and pharmacological characterization.

Autor: Murielle, Rinaldi-Carmona, Francis, Barth, Christian, Congy, Serge, Martinez, Didier, Oustric, Alain, Prio, Martine, Poncelet, Jeanne, Maruani, Michle, Arnone, Olivier, Finance, Philippe, Soubri, Grard, Le Fur

Publikováno v: The Journal of Pharmacology and Experimental Therapeutics; September 2004, Vol. 310 Issue: 3 p905-14, 10p

SSR126768A (4-chloro-3-[(3R)-(+)-5-chloro-1-(2,4-dimethoxybenzyl)-3-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl]-N-ethyl-N-(3-pyridylmethyl)-benzamide, hydrochloride): a new selective and orally active oxytocin receptor antagonist for the prevention of preterm labor.

Autor: Claudine, Serradeil-Le Gal, Grard, Valette, Loc, Foulon, Guy, Germain, Charles, Advenier, Emmanuel, Naline, Marc, Bardou, Jean-Pierre, Martinolle, Brigitte, Pouzet, Danielle, Raufaste, Corinne, Garcia, Elonore, Double-Cazanave, Maxime, Pauly, Marc, Pascal, Alain, Barbier, Bernard, Scatton, Jean-Pierre, Maffrand, Grard, Le Fur

Publikováno v: The Journal of Pharmacology and Experimental Therapeutics; April 2004, Vol. 309 Issue: 1 p414-24, 11p

SSR240600 [(R)-2-(1-[2-[4-[2-[3,5-bis(trifluoromethyl)phenyl]acetyl]-2-(3,4-dichlorophenyl)-2-morpholinyl]ethyl]- 4-piperidinyl)-2-methylpropanamide], a centrally active nonpeptide antagonist of the tachykinin neurokinin-1 receptor: I. biochemical and pharmacological characterization.

Autor: Xavier, Emonds-Alt, Vincenzo, Proietto, Rgis, Steinberg, Florence, Oury-Donat, Xavier, Vig, Pol, Vilain, Emmanuel, Naline, Samira, Daoui, Charles, Advenier, Grard, Le Fur, Jean-Pierre, Maffrand, Philippe, Soubri, Marc, Pascal

Publikováno v: The Journal of Pharmacology and Experimental Therapeutics; December 2002, Vol. 303 Issue: 3 p1171-9, 9p

Characterization of (2S,4R)-1-[5-chloro-1-[(2,4-dimethoxyphenyl)sulfonyl]-3-(2-methoxy-phenyl)-2-oxo-2,3-dihydro-1H-indol-3-yl]-4-hydroxy-N,N-dimethyl-2-pyrrolidine carboxamide (SSR149415), a selective and orally active vasopressin V1b receptor antagonist.

Autor: Claudine, Serradeil-Le Gal, Jean, Wagnon, Jacques, Simiand, Guy, Griebel, Colette, Lacour, Gilles, Guillon, Claude, Barberis, Gabrielle, Brossard, Philippe, Soubri, Dino, Nisato, Marc, Pascal, Rebecca, Pruss, Bernard, Scatton, Jean-Pierre, Maffrand, Grard, Le Fur

Publikováno v: The Journal of Pharmacology and Experimental Therapeutics; March 2002, Vol. 300 Issue: 3 p1122-30, 9p