Zobrazeno 1 - 10
of 174
pro vyhledávání: '"Giuseppe Caliendo"'
Autor:
José Britto-Júnior, Rafael Furlaneto, Antonio Tiago Lima, Mariana Gonçalves de Oliveira, Beatrice Severino, Francesco Frecentese, Ferdinando Fiorino, Giuseppe Caliendo, Marcelo Nicolás Muscará, Gilberto De Nucci
Publikováno v:
Frontiers in Pharmacology, Vol 15 (2024)
Introduction: The human umbilical artery (HUA), rat-isolated right atrium, and rat-isolated vas deferens present a basal release of 6-nitrodopamine (6-ND). The basal release of 6-ND from these tissues was significantly decreased (but not abolished) w
Externí odkaz:
https://doaj.org/article/2f38f458f02f4026a5a5f710af3f2c29
Autor:
Angela Corvino, Giuseppe Caliendo
Publikováno v:
International Journal of Molecular Sciences, Vol 25, Iss 14, p 7932 (2024)
This Special Issue aims to gather new research on hydrogen sulfide (H2S)-releasing compounds (Figure 1) as cutting-edge pharmacological tools and to advance the understanding of the critical role that H2S plays in physiological and pathological proce
Externí odkaz:
https://doaj.org/article/019e04016e894d0fafc9100587bcbb11
Autor:
Angela Corvino, Antonia Scognamiglio, Ferdinando Fiorino, Elisa Perissutti, Vincenzo Santagada, Giuseppe Caliendo, Beatrice Severino
Publikováno v:
International Journal of Molecular Sciences, Vol 25, Iss 13, p 7014 (2024)
Among the various drug discovery methods, a very promising modern approach consists in designing multi-target-directed ligands (MTDLs) able to modulate multiple targets of interest, including the pathways where hydrogen sulfide (H2S) is involved. By
Externí odkaz:
https://doaj.org/article/e3a803e5b57f4e9ba5776d43a99045b6
Autor:
Carmine Secondulfo, Valeria Visco, Nicola Virtuoso, Martino Fortunato, Serena Migliarino, Antonella Rispoli, Lucia La Mura, Adolfo Stellato, Giuseppe Caliendo, Emanuela Settembre, Fabiana Galluccio, Sarah Hamzeh, Giancarlo Bilancio
Publikováno v:
Life, Vol 14, Iss 5, p 617 (2024)
Chronic kidney disease (CKD) and cardiovascular disease (CVD) are highly prevalent conditions, each significantly contributing to the global burden of morbidity and mortality. CVD and CKD share a great number of common risk factors, such as hypertens
Externí odkaz:
https://doaj.org/article/82a77d76efc345648c789d6a9872c6e3
Autor:
Rosa Sparaco, Pierfrancesco Cinque, Antonia Scognamiglio, Angela Corvino, Giuseppe Caliendo, Ferdinando Fiorino, Elisa Magli, Elisa Perissutti, Vincenzo Santagada, Beatrice Severino, Paolo Luciano, Marcello Casertano, Anna Aiello, Gustavo Yuri Martins Viegas, Gilberto De Nucci, Francesco Frecentese
Publikováno v:
Molecules, Vol 29, Iss 7, p 1598 (2024)
4-Nitro and 7-nitro propranolol have been recently synthesized and characterized by us. (±)-4-NO2-propranolol has been shown to act as a selective antagonist of 6-nitrodopamine (6-ND) receptors in the right atrium of rats. As part of our follow-up t
Externí odkaz:
https://doaj.org/article/1faca57576ae452e9550a466612b7446
Autor:
Ida Cerqua, Elisabetta Granato, Angela Corvino, Beatrice Severino, Danilo D’Avino, Martina Simonelli, Elisa Perissutti, Antonia Scognamiglio, Davida Mirra, Bruno D’Agostino, Giuseppe Caliendo, Antonietta Rossi, Giuseppe Cirino, Chiara Maria Motta, Fiorentina Roviezzo
Publikováno v:
Frontiers in Pharmacology, Vol 14 (2023)
Introduction: Hydrogen sulfide (H2S) is emerging as an important potential therapeutic option for respiratory inflammatory diseases. In this study, we investigated the effectiveness of a novel corticosteroid derivative, that is chemically linked to a
Externí odkaz:
https://doaj.org/article/ebceb878295743ad82f57f721e77b614
Autor:
Giorgia Andreozzi, Maria Rosaria Ambrosio, Elisa Magli, Giovanni Maneli, Beatrice Severino, Angela Corvino, Rosa Sparaco, Elisa Perissutti, Francesco Frecentese, Vincenzo Santagada, Anna Leśniak, Magdalena Bujalska-Zadrożny, Giuseppe Caliendo, Pietro Formisano, Ferdinando Fiorino
Publikováno v:
Pharmaceuticals, Vol 16, Iss 10, p 1483 (2023)
Arylpiperazines represent one of the most important classes of 5-HT1AR ligands and have attracted considerable interests for their versatile properties in chemistry and pharmacology, leading to the research of new derivatives that has been focused on
Externí odkaz:
https://doaj.org/article/f809eadae0904facb28d7ccc4163c291
Autor:
Maria Rosaria Ambrosio, Elisa Magli, Giuseppe Caliendo, Rosa Sparaco, Paola Massarelli, Vittoria D’Esposito, Teresa Migliaccio, Giusy Mosca, Ferdinando Fiorino, Pietro Formisano
Publikováno v:
BMC Cancer, Vol 22, Iss 1, Pp 1-14 (2022)
Abstract Background Serotonin (or 5-Hydroxytryptamine, 5-HT) signals in mammary gland becomes dysregulated in cancer, also contributing to proliferation, metastasis, and angiogenesis. Thus, the discovery of novel compounds targeting serotonin signali
Externí odkaz:
https://doaj.org/article/1ff550da64d74d238fdea77957c3ed5d
Autor:
Angela Corvino, Valentina Citi, Ferdinando Fiorino, Francesco Frecentese, Elisa Magli, Elisa Perissutti, Vincenzo Santagada, Vincenzo Calderone, Alma Martelli, Era Gorica, Simone Brogi, Flavia Faganello Colombo, Caroline Nunes Capello, Heloisa Helena Araujo Ferreira, Maria Grazia Rimoli, Federica Sodano, Barbara Rolando, Francesca Pavese, Antonio Petti, Marcelo Nicolás Muscará, Giuseppe Caliendo, Beatrice Severino
Publikováno v:
Journal of Advanced Research, Vol 35, Iss , Pp 267-277 (2022)
Introduction: Hydrogen sulfide (H2S) is a fundamental biological endogenous gas-mediator in the respiratory system. It regulates pivotal patho-physiological processes such as oxidative stress, pulmonary circulation, airway tone and inflammation. Obje
Externí odkaz:
https://doaj.org/article/610e9a0c8bd745389a68efd1fc4472d6
Autor:
Valeria Visco, Carmine Izzo, Davide Bonadies, Federica Di Feo, Giuseppe Caliendo, Francesco Loria, Costantino Mancusi, Pierpaolo Chivasso, Paola Di Pietro, Nicola Virtuoso, Albino Carrizzo, Carmine Vecchione, Michele Ciccarelli
Publikováno v:
Journal of Cardiovascular Development and Disease, Vol 10, Iss 8, p 327 (2023)
Obesity is a growing public health epidemic worldwide and is implicated in slowing improved life expectancy and increasing cardiovascular (CV) risk; indeed, several obesity-related mechanisms drive structural, functional, humoral, and hemodynamic hea
Externí odkaz:
https://doaj.org/article/278cca19ee824e4b905769b4e4a3bbd3