Zobrazeno 1 - 7
of 7
pro vyhledávání: '"Gilles Piquet"'
Autor:
Marie L. Ancelin, Henri J. Vial, Michele Calas, Louis Giral, Gilles Piquet, Eric Rubi, Alan Thomas, Wallace Peters, Christian Slomianny, Socrates Herrera, F. Louis, Vincent Mouanda
Publikováno v:
Memorias do Instituto Oswaldo Cruz, Vol 89, Pp 85-90 (1994)
The systematic screening of more than 250 molecules against Plasmodium falciparum in vitro has previously shown that interfering with phospholipid metabolism is lethal to the malaria parasite. These compounds act by impairing choline transport in inf
Externí odkaz:
https://doaj.org/article/50ae495610d14d3c87ccba3f4d99658e
Autor:
Silvio Aime, Davide Corpillo, Chiara Bracco, Luca Barbero, Silvio Traversa, Giuseppe Digilio, Gilles Piquet, Esposito P
Publikováno v:
Journal of the American Chemical Society. 125:3458-3470
Two novel mono-PEGylated derivatives of hGRF(1-29)-NH(2) [human growth hormone-releasing factor, fragment 1-29] have been synthesized by regio-specific conjugation of Lys(12) or Lys(21) to a monomethoxy-PEG(5000) chain (compounds Lys(12)PEG-GRF and L
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f2d3262ee4ca58690a17a163f51250eb
https://doi.org/10.1021/ja021264j
https://doi.org/10.1021/ja021264j
Autor:
Gérard Cordina, Jean-Louis Aubagnac, Philippe Portefaix, Isabelle Gilles, Michèle Calas, Louis Giral, Gilles Piquet
Publikováno v:
Journal of Mass Spectrometry. 30:985-992
The fast atom bombardment (FAB), frit-FAB and electrospray ionization mass spectra of bis-ammonium salts, C2+ 2X−, were compared. The most informative spectra were the FAB mass spectra with m-nitrobenzyl alcohol as matrix and the Frit-FAB mass spec
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::59830beb70be43c849c7896ebf52cd79
https://doi.org/10.1002/jms.1190300708
https://doi.org/10.1002/jms.1190300708
Autor:
Gilles Piquet, Michèle Calas, Marie-Laure Ancelin, Yann Bordat, Mahama Ouattara, Zyta M. Ziora, Roger Escale, Henri Vial
Publikováno v:
Journal of Medicinal Chemistry
Journal of Medicinal Chemistry, American Chemical Society, 2007, 50 (25), pp.6307-6315. ⟨10.1021/jm0704752⟩
Journal of Medicinal Chemistry, American Chemical Society, 2007, 50 (25), pp.6307-6315. ⟨10.1021/jm0704752⟩
We describe the design, synthesis, and antimalarial activity of 60 bis-tertiary amine, bis-2(1 H)-imino-heterocycle, bis-amidine, and bis-guanidine series. Bis-tertiary amines with a linker from 12 to 16 methylene groups were active against the in vi
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::432965e910a2636db239fa82936e7dfa
https://hal.archives-ouvertes.fr/hal-00275406
https://hal.archives-ouvertes.fr/hal-00275406
Autor:
Valérie Vidal-Sailhan, Marie L. Ancelin, Henri Vial, Gilles Piquet, Philippe Portefaix, Michèle Calas, Gérard Cordina
Publikováno v:
Journal of medicinal chemistry. 43(3)
On the basis of a previous structure-activity relationship study, we identified some essential parameters, e.g. electronegativity and lipophilicity, required for polar head analogues to inhibit Plasmodium falciparum phospholipid metabolism, leading t
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d6f49fec4489d21e59458c93413ec82f
https://pubmed.ncbi.nlm.nih.gov/10669577
https://pubmed.ncbi.nlm.nih.gov/10669577
Autor:
Gilles Piquet, Michèle Calas, Marie L. Ancelin, Eric Rubi, Henri Vial, Vincent Mouanda, Alan W. Thomas, Christian Slomianny, F. Louis, Louis Giral, Wallace Peters, Sócrates Herrera
Publikováno v:
Memórias do Instituto Oswaldo Cruz, Volume: 89 Supplement 2, Pages: 85-90, Published: 1994
Memórias do Instituto Oswaldo Cruz., Vol 89, Pp 85-90 (1994)
Memórias do Instituto Oswaldo Cruz., Vol 89, Pp 85-90 (1994)
The systematic screening of more than 250 molecules against Plasmodium falciparum in vitro has previously shown that interfering with phospholipid metabolism is lethal to the malaria parasite. These compounds act by impairing choline transport in inf
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ca226948c5efa87135a3d5ebf1e57c29
http://www.scielo.br/scielo.php?script=sci_arttext&pid=S0074-02761994000600020&lng=en&tlng=en
http://www.scielo.br/scielo.php?script=sci_arttext&pid=S0074-02761994000600020&lng=en&tlng=en
Autor:
Michèle Calas, Henri Vial, Mahama Ouattara, Gilles Piquet, Zyta Ziora, Y. Bordat, Marie L. Ancelin, Roger Escale
Publikováno v:
Journal of Medicinal Chemistry; Nov2007, Vol. 50 Issue 25, p6307-6315, 9p