Zobrazeno 1 - 10
of 20
pro vyhledávání: '"Gildas Prie"'
Autor:
Abderrahman El Bouakher, Mohamed Akssira, Marie-Claude Viaud-Massuard, Mina Aadil, Gildas Prie
Publikováno v:
Tetrahedron. 69:5086-5091
An efficient synthesis leading to novel 2,4-disubstituted 3H-pyrido[3,2-e][1,4]diazepin-5-ones and 2,4-disubstituted 3H-pyrido[2,3-e][1,4]diazepin-5-ones derivatives is presented, using the condensation of ethyl 2-(benzylamino)acetate or ethyl 2-(4-m
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::2273e765bda4e36dde4bd1faf2a73531
https://doi.org/10.1016/j.tet.2013.04.089
https://doi.org/10.1016/j.tet.2013.04.089
Autor:
Mina Aadil, Ahmed El Hakmaoui, Said Lazar, Marie-Claude Viaud-Massuard, Mohamed Akssira, Abderrahman El Bouakher, Gildas Prie
Publikováno v:
Tetrahedron Letters. 53:6401-6405
An efficient method for synthesizing new pyrido[2,3-e]pyrrolo[1,2-a][1,4]diazepine-5,10-dione derivatives starting from l -proline methyl ester and 2-aminonicotinic acid is presented. This method employs Pd-catalyzed cross-coupling reaction on the co
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::f85e78594c2db57d786a695aaca86e00
https://doi.org/10.1016/j.tetlet.2012.09.041
https://doi.org/10.1016/j.tetlet.2012.09.041
Autor:
Mina Aadil, Said Lazar, Abderrahman El Bouakher, Mohamed Akssira, Marie-Claude Viaud-Massuard, Gildas Prie
Publikováno v:
Tetrahedron. 68:9572-9577
A novel methodology has been developed for the efficient synthesis of 1,4-pyridopyrrolodiazepine derivatives. The key reaction is the bromination under mild conditions by NBS of compounds resulting via peptide coupling of l -proline methyl ester with
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::8a677cd3514c0d2ed3186f115374d4f0
https://doi.org/10.1016/j.tet.2012.09.079
https://doi.org/10.1016/j.tet.2012.09.079
Publikováno v:
ChemInform. 46
7-Azaindoles are versatile building blocks, especially in medicinal chemistry, where they serve as bioisosteres of indoles or purines. Herein, we present a novel rhodium-catalyzed asymmetric 1,4-addition of arylboronic acids to 3-benzylidene-1H-pyrro
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::d6af9a70ecca109cfc114c8e868b5840
https://doi.org/10.1002/chin.201531208
https://doi.org/10.1002/chin.201531208
Publikováno v:
Journal of Organic Chemistry
Journal of Organic Chemistry, American Chemical Society, 2015, 80 (6), pp.3264-3269. ⟨10.1021/jo502784h⟩
Journal of Organic Chemistry, American Chemical Society, 2015, 80 (6), pp.3264-3269. ⟨10.1021/jo502784h⟩
International audience; 7-Azaindoles are versatile building blocks, especially in medicinal chemistry, where they serve as bioisosteres of indoles or purines. Herein, we present a novel rhodium-catalyzed asymmetric 1,4-addition of arylboronic acids t
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::debd3fa59e330667278eaf2ee9abf061
https://hal.archives-ouvertes.fr/hal-02903786
https://hal.archives-ouvertes.fr/hal-02903786
Autor:
Jerome F. Hayes, Michael Shipman, Sabitur Rahman, Gildas Prie, Natacha Prevost, Cyril Montagne, Jason J. Shiers
Publikováno v:
Tetrahedron. 62:8447-8457
2-Methyleneaziridinyl anions can be produced by selective deprotonation of the parent aziridine at C-3 using sec-BuLi/TMEDA. Subsequent reaction with a wide variety of electrophiles including MeI, ICH2CH2CH2CH2Cl, PhCH2Br, allyl bromide, Me3SiCl, Bu3
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::69b220ebdbf739630293126f3e2f5edc
https://doi.org/10.1016/j.tet.2006.06.083
https://doi.org/10.1016/j.tet.2006.06.083
Autor:
Pascal, Didier, Éric, Peyrin, Nicolas, Willand, Serge, Battu, Gaëlle, Bégaud, Aurélie, Bourderioux, Éric, Cavalli, Christian, Cavé, Igor, Clarot, Dominique, Clédat, Raphaël, Delépée, Anne, Denuziere, Fatima, El Garah, Marion, Flipo, Catherine, Foulon, Béatrice, Gargadennec, Karen, Gaudin, Jean-François, Goossens, Christine, Herrenknecht, Nicolas, Huang, Petter, Jordheim Lars, Julie, Karpenko, François-Xavier, Legrand, Christelle, Machon, Pascal, Marchand, Alain, Nicolay, Isabelle, Ourliac-Garnier, Catherine, Perrin, Marine, Peuchmaur, Laurence, Poirier, Gildas, Prié, Christophe, Rochais, Marc, Since, Martin, Soucé, Yen, Vo Hoang, Christelle, Wisniewski
Publikováno v:
In Chimie Analytique – Chimie Organique – Biophysique 2023:vi-vi
Publikováno v:
New Journal of Chemistry. 27:432-441
Stereoselective construction of 3-trifluoromethyl conjugated dienoates, trienoates or dienynoates was achieved from ethyl (Z)-4,4,4-trifluoro-3-iodobutenoate and alkenyltin or alkynyltin reagents through the Stille reaction or under Heck–Sonogashir
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3b3f169a22f0bd19ff4619a6ec9dee91
https://doi.org/10.1039/b207648a
https://doi.org/10.1039/b207648a
Publikováno v:
Journal of Fluorine Chemistry. 117:35-41
(E)- or (Z)-perfluorinated β-enaminoesters were prepared by direct addition of primary or secondary amines to ethyl perfluoroalkynoates without any catalyst.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::d5894e0067475927448f37af5a3b4e99
https://doi.org/10.1016/s0022-1139(02)00162-8
https://doi.org/10.1016/s0022-1139(02)00162-8
Autor:
Erika J, Obando Montoya, Céline, Mélin, Nathalie, Blanc, Arnaud, Lanoue, Emilien, Foureau, Leslie, Boudesocque, Gildas, Prie, Andrew J, Simkin, Joël, Crèche, Lucia, Atehortùa, Nathalie, Giglioli-Guivarc'h, Marc, Clastre, Vincent, Courdavault, Nicolas, Papon
Publikováno v:
Yeast (Chichester, England). 31(7)
Candida guilliermondii (teleomorph Meyerozyma guilliermondii) is an ascomycetous species belonging to the fungal CTG clade. This yeast remains actively studied as a result of its moderate clinical importance and most of all for its potential uses in
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::a0bf130f45c4c47cdc7a63e6c73e0c44
https://pubmed.ncbi.nlm.nih.gov/24700391
https://pubmed.ncbi.nlm.nih.gov/24700391