Zobrazeno 1 - 10
of 17
pro vyhledávání: '"Gerald S. Jones"'
7,10-Bis(2-mercapto-2-methyl)propyl-7,10-diazapalmitic acid: a novel, N2S2 ligand for technetium-99m
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 6:2399-2404
7,10-Bis(2-mercapto-2-methyl)propyl-7,10-diazapalmitic acid (7) was synthesized and evaluated as a new ligand for technetium-99m (99mTc). The title fatty acid analog, an achiral, bis(aminoethanethiol) derivative in which the amines are tertiary, gave
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::79a7bc62975fa2c3dce3efe2f99c196b
https://doi.org/10.1016/0960-894x(96)00440-4
https://doi.org/10.1016/0960-894x(96)00440-4
Publikováno v:
Nuclear Medicine and Biology. 21:117-123
The synthesis and biodistribution is described for a new 99mTc-labeled fatty acid. The requisite diaminodithiol (N2S2) ligand, 9,10-bis[N-(2'-methyl-2'-mercapto)propyl] aminooctadecanoic acid, was prepared in nine steps from ethyl oleate and characte
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::883511bd3fe93076166b1c57d893310a
https://doi.org/10.1016/0969-8051(94)90138-4
https://doi.org/10.1016/0969-8051(94)90138-4
Publikováno v:
Molecular Brain Research. 15:113-120
The agonist binding site of nicotinic acetylcholine receptors (AChRs) includes a disulfide bond that is easily reduced with dithiothreitol to a pair of thiols, and can be then either reoxidized with dithiobis(nitrobenzoic acid) (DTNB) or irreversibly
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0059a03c40108c8e8032ffdf2cb32cf9
https://doi.org/10.1016/0169-328x(92)90158-8
https://doi.org/10.1016/0169-328x(92)90158-8
Publikováno v:
The Journal of Infectious Diseases. 162:700-704
To determine the role of oxygen radicals in the killing of Mycobacterium tuberculosis by neutrophils, the effects of free-radical inhibitors and enzymes, catalase, superoxide dismutase, taurine, deferoxamine, and histidine were evaluated. Changes in
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2a0b214087b6e6b79e3d13076e451676
https://doi.org/10.1093/infdis/162.3.700
https://doi.org/10.1093/infdis/162.3.700
Autor:
Jennifer S. Daly, Gerald S. Jones
Publikováno v:
Journal of Pharmaceutical Sciences. 82:755-757
A series of phosphoranilidohydrazones of 5-nitro-2-furaldehyde was synthesized and evaluated for antibacterial activity. The series was prepared to examine the applicability of phosphoramidic hydrazones as carriers for the antibacterial nitrofuran mo
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::42b1887788b1ce9b686356cac5b53f3d
https://doi.org/10.1002/jps.2600820716
https://doi.org/10.1002/jps.2600820716
Publikováno v:
Bioconjugate chemistry. 10(4)
We synthesized three novel organoarsenicals as prototype bifunctional reagents for spatially close thiols, N-(4-arsenosophenyl) hexahydro-2-oxo-(3aS,4S,6aR)-1H-thieno[3, 4-d]imidazole-4-pentamide (1), 2-[4-[(4-arsenosophenyl)amino]-1, 4-dioxobutyl] h
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ebd77e4659434329e418d84f4171563a
https://pubmed.ncbi.nlm.nih.gov/10411461
https://pubmed.ncbi.nlm.nih.gov/10411461
Autor:
David R. Elmaleh, Gerald S. Jones, Robert N. Hanson, Lee W. Herman, H. Kizuka, H. William Strauss
Publikováno v:
Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine. 44(5)
A series of phentermine analogs, including the unsubstituted, the para-F, -Cl, -Br and -I, and the meta-CF3 derivatives, were labeled by [11C]methylation and evaluated in rats to determine the structure-localization relationships for this class of re
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::185137148600adf6170f84267e03f81c
https://pubmed.ncbi.nlm.nih.gov/8485509
https://pubmed.ncbi.nlm.nih.gov/8485509
Publikováno v:
Journal of pharmaceutical sciences. 81(4)
The p ‐aminobenzyl analogues ( 8a and 8b , respectively) of the cardioselective β ‐adrenergic receptor antagonists practolol and atenolol were prepared from the corresponding phenoxymethyloxiranes in 30 and 13% yields, respectively. The dissocia
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::236831f82ce8503ba01320933d3ed2db
https://pubmed.ncbi.nlm.nih.gov/1354250
https://pubmed.ncbi.nlm.nih.gov/1354250
Autor:
Gerald S. Jones
Publikováno v:
Performance & Instruction. 21:44-44
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::5f93661dab46e38a49ff895eb55c4743
https://doi.org/10.1002/pfi.4170210828
https://doi.org/10.1002/pfi.4170210828
Autor:
Gerald S. Jones, David R. Elmaleh
Publikováno v:
Organic Preparations and Procedures International. 22:112-113
(1990). A CONVENIENT ONE-POT SYNTHESIS OF 2-METHYL-2-BENZYLTHIOPROPANAL. Organic Preparations and Procedures International: Vol. 22, No. 1, pp. 112-113.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::b10a67d5fb997cd02f30cd097276a7c0
https://doi.org/10.1080/00304949009356679
https://doi.org/10.1080/00304949009356679