Zobrazeno 1 - 7
of 7
pro vyhledávání: '"Gary Javadi"'
Publikováno v:
Synthesis. 2008:891-896
Herein is described the development and use of a novel bis(dialkylamino)sulfur difluoride reagent to effect the stereoselective conversion of a benzylic alcohol into a benzylic fluoride. A new method for the synthesis of 1 H-pyrazolo[3,4- D]pyrimidin
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::671ca93449c6ec54e4bf2df2bceef576
https://doi.org/10.1055/s-2008-1032181
https://doi.org/10.1055/s-2008-1032181
Autor:
Wenjie Li, Gary Javadi, Dongwei Cai, Robert D. Larsen, Mark S. Jensen, R. Scott Hoerrner, Dorian P. Nelson, Peter G. Dormer
Publikováno v:
The Journal of Organic Chemistry. 70:6034-6039
A practical synthesis of 2-[3-(4-fluoro-3-pyridin-3-yl-phenyl)-imidazo[1,2-a]pyrimidin-7-yl]-propan-2-ol (1), an oral GABA(A) alpha(2/3)-selective agonist, is described. The five-step process, which afforded 1 in 40% overall yield, included imidazopy
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::056f9e9e8fb3f7c76d5d32884da2085a
https://doi.org/10.1021/jo050741o
https://doi.org/10.1021/jo050741o
Publikováno v:
ChemInform. 36
An improved synthesis of N-isocyanoiminotriphenylphosphorane is reported. This reagent is a safe, stable, solid alternative to diazomethane and TMS-diazomethane in the Arndt-Eistert synthesis of diazoketones.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::491acf129b4a40c6b67172ad30af585d
https://doi.org/10.1002/chin.200521181
https://doi.org/10.1002/chin.200521181
Autor:
Mark S. Jensen, Wenjie Li, Robert D. Larsen, Gary Javadi, Dongwei Cai, Dorian P. Nelson, R. Scott Hoerrner
Publikováno v:
ChemInform. 35
Imidazo[1,2-a]pyrimidine can be arylated at the 3-position with aryl bromides in the presence of base and a catalytic amount of palladium. This provides an efficient one-step synthesis of 3-arylimidazo[1,2-a]pyrimidines from the unsubstituted heteroc
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fce8acdf97d89a92b309cec174151f5d
https://doi.org/10.1002/chin.200416140
https://doi.org/10.1002/chin.200416140
Autor:
Jennifer R. Chilenski, Daniel Zewge, Johnnie L. Leazer, Marjorie S. Waters, Robert A. Reamer, Fengrui Lang, Gary Javadi, Richard D. Tillyer, Matthew M. Bio, Amude M. Kassim, Ralph P. Volante, Anthony O. King, Zhiguo J. Song, Thorsten Rosner, David J. Mathre, David M. Tschaen
An efficient asymmetric synthesis of a selective estrogen receptor modulator (SERM) that has a dihydrobenzoxathiin core structure bearing two stereogenic centers is reported. The stereogenic centers were established by an unprecedented chiral sulfoxi
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bc80db2c69738e6ee5dafd2c3226a6f0
https://europepmc.org/articles/PMC395984/
https://europepmc.org/articles/PMC395984/
Publikováno v:
ChemInform. 32
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::a17fdcdca90d447dc7bcc5536fa0b752
https://doi.org/10.1002/chin.200109085
https://doi.org/10.1002/chin.200109085
Publikováno v:
Synthesis; 2005, Vol. 2005 Issue 1, p19-21, 3p