Zobrazeno 1 - 6
of 6
pro vyhledávání: '"Gary Bammert"'
Autor:
Daryl R. Sauer, Jonathan Greer, Charles J. Nichols, Craig D. Wegner, Jason A. Segreti, Kurt M. Mohning, Fortuna Haviv, John T. Randolph, E N Bush, Philip L. Waid, Gilbert Diaz, Leslie M. Besecke, Gary Bammert
Publikováno v:
Journal of Medicinal Chemistry. 47:1085-1097
The design and synthesis of a series of 11,12-cyclic carbamate derivatives of 6-O-methylerythromycin A that are novel, nonpeptide LHRH antagonists, is described. The macrolide antagonist 1, discovered during a screen of our chemical repository, was c
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3fabef2f09ac213c5e8373f774e466e4
https://doi.org/10.1021/jm030418i
https://doi.org/10.1021/jm030418i
Autor:
Crawford Bradley W, Craig D. Wegner, Wesley J. Dwight, Frey Lisa Marie, Fortuna Haviv, Eugene N. Bush, Rolf E. Swenson, Kurt M. Mohning, Gary Bammert, Yoshihiro Sugiura, Kaminski Michele A, Milan Bruncko, Jonathan Greer, Kaneyoshi Kato, Leslie M. Besecke, Mary Spangler, Gilbert Diaz, Jason A. Segreti
Publikováno v:
Peptides for the New Millennium ISBN: 0792364457
Fortuna Haviv, Wesley Dwight, Bradley Crawford, Rolf Swenson, Milan Bruncko, Michele Kaminski, Kaneyoshi Kato, Yoshihiro Sugiura, Lisa Frey, Gilbert Diaz, Gary Bammert, Eugene N. Bush, Leslie Besecke, Kurt Mohning, Jason Segreti, Mary Spangler, Craig
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::fbf25eab17aec1d40066ea8038c0376c
https://doi.org/10.1007/0-306-46881-6_97
https://doi.org/10.1007/0-306-46881-6_97
In vitro and in vivo activities of reduced-size antagonists of luteinizing hormone-releasing hormone
Autor:
Gilbert Diaz, Gary Bammert, Judith Knittle, Jonathan Greer, Charles J. Nichols, Edwin S. Johnson, Eugene N. Bush, Fortuna Haviv, Timothy D. Fitzpatrick, A. T. Nguyen
Publikováno v:
Journal of medicinal chemistry. 37(5)
A novel series of octapeptide LHRH antagonists was designed on the basis of the structure of the (2-9) fragment of a LHRH agonist. By adopting a systematic SAR study, we were able to improve first the in vitro activity and then the in vivo LH suppres
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8c162d80694001661dca74664a3820a3
https://pubmed.ncbi.nlm.nih.gov/7510341
https://pubmed.ncbi.nlm.nih.gov/7510341
Autor:
Timothy D. Fitzpatrick, Charles J. Nichols, J. Knittle, E. N. Bush, E. S. Johnson, J. Greer, Fortuna Haviv, A. T. Nguyen, N. S. Rhutasel, George A. Diaz, Gary Bammert
Publikováno v:
Peptides ISBN: 9789401042956
Peptides
Peptides
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::4873882e14c1c6259e5ea2a2451d4dcc
https://doi.org/10.1007/978-94-011-0683-2_130
https://doi.org/10.1007/978-94-011-0683-2_130
Autor:
N. S. Rhutasel, J. Greer, V. Cybulski, Fortuna Haviv, Gary Bammert, J. Leal, E. N. Bush, Mort Nicholas A, A. T. Nguyen, J. Knittle, George A. Diaz, Rolf E. Swenson
Publikováno v:
Peptides ISBN: 9789401042956
Peptides
Peptides
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::cf5d5a09d45cac6e5f7b3af2509fcae8
https://doi.org/10.1007/978-94-011-0683-2_150
https://doi.org/10.1007/978-94-011-0683-2_150
Autor:
Rolf E. Swenson, A. T. Nguyen, George A. Diaz, Charles J. Nichols, Timothy D. Fitzpatrick, Fortuna Haviv, E N Bush, Mort Nicholas A, Gary Bammert, N. S. Rhutasel
Publikováno v:
Journal of medicinal chemistry. 36(3)
Each peptide bond in leuprolide (1), deslorelin (13), and nafarelin (24) was separately substituted with N-methyl. The synthesized compounds were tested for in vitro receptor binding, LH release, and stability against chymotrypsin and intestinal degr
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2ea76c5aa0f04c3993bf67eb9877f6ff
https://pubmed.ncbi.nlm.nih.gov/8381183
https://pubmed.ncbi.nlm.nih.gov/8381183