Zobrazeno 1 - 10 of 117 pro vyhledávání: '"García-Cárceles J"'
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Akademický článek
A Strategy for the Formal C-N Cross-Coupling of Tertiary Amines.
Autor: Ledwith PR; Department of Chemistry, University of Liverpool, Crown Street, Liverpool, United Kingdom, L69 7ZD., Cooney ML; Department of Chemistry, University of Liverpool, Crown Street, Liverpool, United Kingdom, L69 7ZD.; School of Chemistry, University of Bristol, Cantock's Close, Bristol, United Kingdom, BS8 1TS., Bahou KA; Department of Chemistry, University of Liverpool, Crown Street, Liverpool, United Kingdom, L69 7ZD., García-Cárceles J; School of Chemistry, University of Bristol, Cantock's Close, Bristol, United Kingdom, BS8 1TS., Thomson J; School of Chemistry, University of Bristol, Cantock's Close, Bristol, United Kingdom, BS8 1TS., Bower JF; Department of Chemistry, University of Liverpool, Crown Street, Liverpool, United Kingdom, L69 7ZD.
Publikováno v: Angewandte Chemie (International ed. in English) [Angew Chem Int Ed Engl] 2024 Dec 09; Vol. 63 (50), pp. e202411555. Date of Electronic Publication: 2024 Oct 22.
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2
Akademický článek
2-(Fluoromethoxy)-4'-( S -methanesulfonimidoyl)-1,1'-biphenyl (UCM-1306), an Orally Bioavailable Positive Allosteric Modulator of the Human Dopamine D 1 Receptor for Parkinson's Disease.
Autor: García-Cárceles J; Departamento de Química Orgánica, Universidad Complutense de Madrid, E-28040 Madrid, Spain., Vázquez-Villa H; Departamento de Química Orgánica, Universidad Complutense de Madrid, E-28040 Madrid, Spain., Brea J; Biofarma Research Group, USEF Screening Platform, CIMUS, USC, E-15782 Santiago de Compostela, Spain., Ladron de Guevara-Miranda D; Instituto de Investigación Biomédica de Málaga (IBIMA), E-29010 Málaga, Spain., Cincilla G; Molomics S.L., Parc Científic de Barcelona, Baldiri Reixac 4-8, E-08028 Barcelona, Spain., Sánchez-Martínez M; Molomics S.L., Parc Científic de Barcelona, Baldiri Reixac 4-8, E-08028 Barcelona, Spain., Sánchez-Merino A; Departamento de Química Orgánica, Universidad Complutense de Madrid, E-28040 Madrid, Spain., Algar S; Departamento de Química Orgánica, Universidad Complutense de Madrid, E-28040 Madrid, Spain., Teresa de Los Frailes M; Fundación Kærtor, Edificio EMPRENDIA, Planta 2, Oficina 4. Campus Vida, E-15706 Santiago de Compostela, Spain., Roberts RS; Fundación Kærtor, Edificio EMPRENDIA, Planta 2, Oficina 4. Campus Vida, E-15706 Santiago de Compostela, Spain., Ballesteros JA; Vivia Biotech S.L., Parque Científico de Madrid, E-28760 Madrid, Spain., Rodríguez de Fonseca F; Instituto de Investigación Biomédica de Málaga (IBIMA), E-29010 Málaga, Spain., Benhamú B; Departamento de Química Orgánica, Universidad Complutense de Madrid, E-28040 Madrid, Spain., Loza MI; Biofarma Research Group, USEF Screening Platform, CIMUS, USC, E-15782 Santiago de Compostela, Spain.; Fundación Kærtor, Edificio EMPRENDIA, Planta 2, Oficina 4. Campus Vida, E-15706 Santiago de Compostela, Spain., López-Rodríguez ML; Departamento de Química Orgánica, Universidad Complutense de Madrid, E-28040 Madrid, Spain.
Publikováno v: Journal of medicinal chemistry [J Med Chem] 2022 Sep 22; Vol. 65 (18), pp. 12256-12272. Date of Electronic Publication: 2022 Aug 31.
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3
Akademický článek
Discovery of V-0219: A Small-Molecule Positive Allosteric Modulator of the Glucagon-Like Peptide-1 Receptor toward Oral Treatment for "Diabesity".
Autor: Decara JM; Unidad de Gestión Clínica de Salud Mental, Instituto IBIMA, Hospital Regional Universitario, Málaga E-29010, Spain., Vázquez-Villa H; Departamento de Química Orgánica, Universidad Complutense de Madrid, Madrid E-28040, Spain., Brea J; Biofarma Research group, USEF Screening Platform, CIMUS, USC, Santiago de Compostela E-15782, Spain., Alonso M; Unidad de Gestión Clínica de Salud Mental, Instituto IBIMA, Hospital Regional Universitario, Málaga E-29010, Spain., Srivastava RK; Institute of Physiological Chemistry, University Medical Center of the Johannes Gutenberg, University of Mainz, Mainz 55128, Germany., Orio L; Departamento de Psicobiología, Facultad de Psicología, Universidad Complutense de Madrid, Madrid E-28040, Spain., Alén F; Departamento de Psicobiología, Facultad de Psicología, Universidad Complutense de Madrid, Madrid E-28040, Spain., Suárez J; Unidad de Gestión Clínica de Salud Mental, Instituto IBIMA, Hospital Regional Universitario, Málaga E-29010, Spain., Baixeras E; Unidad de Gestión Clínica de Salud Mental, Instituto IBIMA, Hospital Regional Universitario, Málaga E-29010, Spain., García-Cárceles J; Departamento de Química Orgánica, Universidad Complutense de Madrid, Madrid E-28040, Spain., Escobar-Peña A; Departamento de Química Orgánica, Universidad Complutense de Madrid, Madrid E-28040, Spain., Lutz B; Institute of Physiological Chemistry, University Medical Center of the Johannes Gutenberg, University of Mainz, Mainz 55128, Germany., Rodríguez R; Galchimia, O Pino, A Coruña E-15823, Spain., Codesido E; Galchimia, O Pino, A Coruña E-15823, Spain., Garcia-Ladona FJ; ABAXYS Therapeutics, Rue du Berceau, 91, Villers-la-Ville 1495, Belgium., Bennett TA; ViviaBiotech S.L., Parque Científico de Madrid, Madrid E-28760, Spain., Ballesteros JA; ViviaBiotech S.L., Parque Científico de Madrid, Madrid E-28760, Spain., Cruces J; Galchimia, O Pino, A Coruña E-15823, Spain., Loza MI; Biofarma Research group, USEF Screening Platform, CIMUS, USC, Santiago de Compostela E-15782, Spain., Benhamú B; Departamento de Química Orgánica, Universidad Complutense de Madrid, Madrid E-28040, Spain., Rodríguez de Fonseca F; Unidad de Gestión Clínica de Salud Mental, Instituto IBIMA, Hospital Regional Universitario, Málaga E-29010, Spain.; Departamento de Psicobiología, Facultad de Psicología, Universidad Complutense de Madrid, Madrid E-28040, Spain., López-Rodríguez ML; Departamento de Química Orgánica, Universidad Complutense de Madrid, Madrid E-28040, Spain.
Publikováno v: Journal of medicinal chemistry [J Med Chem] 2022 Apr 14; Vol. 65 (7), pp. 5449-5461. Date of Electronic Publication: 2022 Mar 29.
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4
Akademický článek
Kinase Inhibitors as Underexplored Antiviral Agents.
Autor: García-Cárceles J; Centro de Investigaciones Biológicas Margarita Salas (CSIC), Ramiro de Maeztu 9, 28040 Madrid, Spain., Caballero E; Centro de Investigaciones Biológicas Margarita Salas (CSIC), Ramiro de Maeztu 9, 28040 Madrid, Spain., Gil C; Centro de Investigaciones Biológicas Margarita Salas (CSIC), Ramiro de Maeztu 9, 28040 Madrid, Spain., Martínez A; Centro de Investigaciones Biológicas Margarita Salas (CSIC), Ramiro de Maeztu 9, 28040 Madrid, Spain.
Publikováno v: Journal of medicinal chemistry [J Med Chem] 2022 Jan 27; Vol. 65 (2), pp. 935-954. Date of Electronic Publication: 2021 May 10.
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5
Akademický článek
Complex Polyheterocycles and the Stereochemical Reassignment of Pileamartine A via Aza-Heck Triggered Aryl C-H Functionalization Cascades.
Autor: Jones BT; School of Chemistry, University of Bristol, Bristol, BS8 1TS, United Kingdom., García-Cárceles J; School of Chemistry, University of Bristol, Bristol, BS8 1TS, United Kingdom., Caiger L; School of Chemistry, University of Bristol, Bristol, BS8 1TS, United Kingdom., Hazelden IR; School of Chemistry, University of Bristol, Bristol, BS8 1TS, United Kingdom., Lewis RJ; Department of Medicinal Chemistry, Research and Early Development, Respiratory and Immunology, BioPharmaceuticals R&D, AstraZeneca, SE 43183 Mölndal, Sweden., Langer T; Chemical Development, Pharmaceutical Technology & Development, Operations, Astra Zeneca, Charter Way, Macclesfield, SK10 2NA, United Kingdom., Bower JF; Department of Chemistry, University of Liverpool, Crown Street, Liverpool, L69 7ZD, United Kingdom.
Publikováno v: Journal of the American Chemical Society [J Am Chem Soc] 2021 Sep 29; Vol. 143 (38), pp. 15593-15598. Date of Electronic Publication: 2021 Sep 21.
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6
Akademický článek
Host-Directed FDA-Approved Drugs with Antiviral Activity against SARS-CoV-2 Identified by Hierarchical In Silico/In Vitro Screening Methods.
Autor: Ginex T; Centro de Investigaciones Biológicas Margarita Salas-CSIC, Ramiro de Maeztu 9, 28040 Madrid, Spain., Garaigorta U; Centro Nacional de Biotecnología-CSIC, Calle Darwin 3, 28049 Madrid, Spain., Ramírez D; Instituto de Ciencias Biomédicas, Universidad Autónoma de Chile, Llano Subercaseaux 2801-piso 6, Santiago 7500912, Chile., Castro V; Centro Nacional de Biotecnología-CSIC, Calle Darwin 3, 28049 Madrid, Spain., Nozal V; Centro de Investigaciones Biológicas Margarita Salas-CSIC, Ramiro de Maeztu 9, 28040 Madrid, Spain., Maestro I; Centro de Investigaciones Biológicas Margarita Salas-CSIC, Ramiro de Maeztu 9, 28040 Madrid, Spain., García-Cárceles J; Centro de Investigaciones Biológicas Margarita Salas-CSIC, Ramiro de Maeztu 9, 28040 Madrid, Spain., Campillo NE; Centro de Investigaciones Biológicas Margarita Salas-CSIC, Ramiro de Maeztu 9, 28040 Madrid, Spain., Martinez A; Centro de Investigaciones Biológicas Margarita Salas-CSIC, Ramiro de Maeztu 9, 28040 Madrid, Spain., Gastaminza P; Centro Nacional de Biotecnología-CSIC, Calle Darwin 3, 28049 Madrid, Spain., Gil C; Centro de Investigaciones Biológicas Margarita Salas-CSIC, Ramiro de Maeztu 9, 28040 Madrid, Spain.
Publikováno v: Pharmaceuticals (Basel, Switzerland) [Pharmaceuticals (Basel)] 2021 Apr 06; Vol. 14 (4). Date of Electronic Publication: 2021 Apr 06.
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7
Akademický článek
Exploring 4,7-Disubstituted Pyrimido[4,5- d ]pyrimidines as Antiviral and Anticancer Agents.
Autor: Georgiou, Eleftheria A.1 (AUTHOR) elgeorgiou@pharm.uoa.gr, Paraskevas, Konstantinos1 (AUTHOR) kon.paraskevas@outlook.com, Koutra, Christina2 (AUTHOR) ckoutral@pharm.uoa.gr, Persoons, Leentje3 (AUTHOR) leentje.persoons@kuleuven.be, Schols, Dominique4 (AUTHOR) dominique.schols@kuleuven.be, De Jonghe, Steven4 (AUTHOR) steven.dejonghe@kuleuven.be, Kostakis, Ioannis K.1 (AUTHOR) ikkostakis@pharm.uoa.gr
Publikováno v: Molecules. Dec2024, Vol. 29 Issue 23, p5549. 14p.
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8
Akademický článek
Inhibition of Cancer Stem-like Cells by Curcumin and Other Polyphenol Derivatives in MDA-MB-231 TNBC Cells.
Autor: Ros, Maria1 (AUTHOR), Riesco-Llach, Gerard2 (AUTHOR) marta.planas@udg.edu, Polonio-Alcalá, Emma1 (AUTHOR), Morla-Barcelo, Pere Miquel3 (AUTHOR), Ruiz-Martínez, Santiago4 (AUTHOR), Feliu, Lidia2 (AUTHOR) lidia.feliu@udg.edu, Planas, Marta2 (AUTHOR), Puig, Teresa1 (AUTHOR) lidia.feliu@udg.edu
Publikováno v: International Journal of Molecular Sciences. Jul2024, Vol. 25 Issue 13, p7446. 21p.
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9
Akademický článek
Morpholine, Piperazine, and Piperidine Derivatives as Antidiabetic Agents.
Autor: Zolotareva, Darya1 (AUTHOR) zolotareva.2909@mail.ru, Zazybin, Alexey1 (AUTHOR) azazybin@yahoo.com, Dauletbakov, Anuar1 (AUTHOR) dayletbakovanuar@gmail.com, Belyankova, Yelizaveta1 (AUTHOR) belyankovae@gmail.com, Parache, Beatriz Giner2 (AUTHOR) bginer@usj.es, Tursynbek, Saniya1 (AUTHOR) erzhanovnasss@gmail.com, Seilkhanov, Tulegen3 (AUTHOR) tseilkhanov@mail.ru, Kairullinova, Anel1 (AUTHOR) anelkin.ka@gmail.com
Publikováno v: Molecules. Jul2024, Vol. 29 Issue 13, p1-18. 18p. 31 Diagrams, 1 Graph.
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10
Akademický článek
Drug Development for Alzheimer's and Parkinson's Disease: Where Do We Go Now?
Autor: Sequeira, Lisa1 (AUTHOR), Benfeito, Sofia1 (AUTHOR), Fernandes, Carlos1 (AUTHOR), Lima, Inês1 (AUTHOR), Peixoto, Joana1 (AUTHOR), Alves, Catarina1 (AUTHOR), Machado, Cláudia Sofia1 (AUTHOR), Gaspar, Alexandra1 (AUTHOR), Borges, Fernanda1 (AUTHOR) fborges@fc.up.pt, Chavarria, Daniel1 (AUTHOR) fborges@fc.up.pt
Publikováno v: Pharmaceutics. Jun2024, Vol. 16 Issue 6, p708. 30p.
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