Zobrazeno 1 - 10
of 371
pro vyhledávání: '"Garbarg M"'
Publikováno v:
Proceedings of the National Academy of Sciences of the United States of America, 1988 Apr . 85(8), 2743-2747.
Externí odkaz:
https://www.jstor.org/stable/31512
Autor:
Garbarg M, W. Tertiuk, Charon Robin Ganellin, Athmani S, A. Fkyerat, Benny Bang-Andersen, Schwartz Jc, X Ligneau
Publikováno v:
ChemInform. 28
[[(4-Nitrophenyl)X]alkyl]imidazole isosteres (where X = NH, S, CH2S, O) of previously described [[(5-nitropyrid-2-yl)X]ethyl]imidazoles (where X = NH, S) have been synthesized and evaluated for H3-receptor histamine antagonism in vitro (Ki for [3H]hi
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::72ce2b5c61420cfa411b847f19bed17f
https://doi.org/10.1002/chin.199703168
https://doi.org/10.1002/chin.199703168
Autor:
Schwartz Jc, Garbarg M, Jean-Michel Batiment Arrang, Fabien Leurquin, Antonia Piripitsi, C. Robin Ganellin, W Schunack, X Ligneau
Publikováno v:
ChemInform. 30
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::dbe83441c6a5b33d517017434f0fbc34
https://doi.org/10.1002/chin.199913111
https://doi.org/10.1002/chin.199913111
Autor:
Schwartz, J.C., author, Giros, B., author, Gros, C., author, Llorens-Cortes, C., author, Arrang, J.M., author, Garbarg, M., author, Pollard, H., author
Publikováno v:
Migraine: A Spectrum of Ideas, 1990.
Externí odkaz:
https://doi.org/10.1093/acprof:oso/9780192618108.003.0018
Publikováno v:
PLoS ONE
PLoS ONE, Vol 8, Iss 9, p e73328 (2013)
PLoS ONE, Vol 8, Iss 9, p e73328 (2013)
Small conductance calcium-activated potassium channels (KCa2.1,2.2,2.3) are blocked with high affinity by both peptide toxins (e.g. apamin) and small molecule blockers (e.g. UCL 1848). In electrophysiological experiments, apamin shows subtype selecti
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9efdc09da8903aca99c1c21b43e1cfab
https://doi.org/10.1371/journal.pone.0073328
https://doi.org/10.1371/journal.pone.0073328
Autor:
W. Tertiuk, A. Fkyerat, Benny Bang-Andersen, X Ligneau, Athmani S, Schwartz Jc, Garbarg M, Charon Robin Ganellin
Publikováno v:
Journal of medicinal chemistry. 39(19)
[[(4-Nitrophenyl)X]alkyl]imidazole isosteres (where X = NH, S, CH2S, O) of previously described [[(5-nitropyrid-2-yl)X]ethyl]imidazoles (where X = NH, S) have been synthesized and evaluated for H3-receptor histamine antagonism in vitro (Ki for [3H]hi
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a8a95cd8ae6a4fb6cff5d0ff21b5d8d8
https://pubmed.ncbi.nlm.nih.gov/8809168
https://pubmed.ncbi.nlm.nih.gov/8809168
Publikováno v:
Europe PubMed Central
The histamine H3 receptor has been shown to inhibit pentagastrin-induced gastric acid secretion in dogs. Since pentagastrin releases histamine in dogs, we have now assessed whether the effects of H3-receptor ligands may be indirectly mediated by chan
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8783f3f3f49624c591b31d8074d6de55
http://hdl.handle.net/11568/51214
http://hdl.handle.net/11568/51214
Autor:
Ganellin, C. R., Fkyerat, A., Hosseini, S. K., Khalaf, Y. S., Piripitsi, A., Tertiuk, W., Arrang, J. M., Garbarg, M., Ligneau, X., Schwartz, J. C.
Se han sintetizado análogos de tioperamida. Los compuestos han sido ensayados in vitro para explorar los factores que permitan diseñar compuestos derivados de la tioperamida sin grupo tiourea que mejoren la penetración cerebral. Los compuestos má
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=od______1648::872bfcd6c6139271ad5e1874c26f0e2c
https://hdl.handle.net/10481/83675
https://hdl.handle.net/10481/83675
Publikováno v:
New Perspectives in Histamine Research ISBN: 9783034873116
Several alkyl-substituted histamine derivatives have been synthesized and investigated for their agonistic potency on three classes of histamine receptors. While all investigated compounds are full agonists at H3-receptors their relative potency vs.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::9fb11b040f1dd663d9ede64a9e2dd763
https://doi.org/10.1007/978-3-0348-7309-3_18
https://doi.org/10.1007/978-3-0348-7309-3_18