Zobrazeno 1 - 10
of 43
pro vyhledávání: '"Gangloff, Anthony R."'
Autor:
Elaine Y.-L Kuo, Daun Putnam, Kenneth D. Rice, Gangloff Anthony R, Martin Wong, Dener Jeffrey M, William S Newcomb, Vivian R. Wang
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 11:2325-2330
Truncation of potent and selective dibasic inhibitors afforded monocharged inhibitors of human mast-cell tryptase. Using two classes of analogues as lead structures, several monocharged derivatives were identified with K(i) values ranging from 0.084
Autor:
Gangloff, Anthony R., Brown, Jason, de Jong, Ron, Dougan, Douglas R., Grimshaw, Charles E., Hixon, Mark, Jennings, Andy, Kamran, Ruhi, Kiryanov, Andre, O’Connell, Shawn, Taylor, Ewan, Vu, Phong
Publikováno v:
In Bioorganic & Medicinal Chemistry Letters 15 August 2013 23(16):4501-4505
Autor:
Nina Kann, Y. Wu, Muriel Cottard, Timothy L. Friebe, Tobias Rein, Javed Iqbal, Marc Demillequand, Björn Åkermark, Mikael Bergdahl, Gangloff Anthony R, M. M. Mader, Paul Helquist, Robert Hett
Publikováno v:
Pure and Applied Chemistry. 66:2063-2066
A number of new synthetic methods have been developed that are applicable to several types of antibiotics possessing macrocyclic lactone or lactam structures. These methods have permitted the synthe- sis of several key subunits of these compounds, an
Autor:
Javed Iqbal, Mikael Bergdahl, Gangloff Anthony R, Robert Hett, Timothy L. Friebe, Yinghui Wu, Paul Helquist
Publikováno v:
Tetrahedron Letters. 34:7371-7374
The right-hand portion (3) of the type A streptogramin antibiotics was synthesized in non-racemic form through use of a Horner-Wadsworth-Emmons reaction for diene construction, an asymmetric aldol condensation, and a zinc-promoted oxazole addition re
Publikováno v:
Tetrahedron. 49:5445-5459
Rhodium(II) acetate serves as a catalyst for the heterocycloaddition reaction of diazodicarbonyl compounds with nitriles to give functionalized 1,3-oxazole derivatives in a simple one-step procedure. In particular, dimethyl diazomalonate undergoes th
Autor:
Emma J. Shelton, Vivian R. Wang, David Sperandio, Gangloff Anthony R, Rice Kenneth D, Joane Litvak
Publikováno v:
Tetrahedron Letters. 42:1441-1443
Tetrabutylammonium fluoride (TBAF) was found to be a mild and efficient catalyst for the synthesis of 3,5-disubstituted-1,2,4-oxadiazoles. Using 0.1–1.0 equivalents of TBAF in THF for 1–24 h at room temperature, alkanoyl- and aroyloxyamidines wer
Publikováno v:
ChemInform. 24
Publikováno v:
ChemInform. 24
Rhodium(II) acetate serves as a catalyst for the heterocycloaddition reaction of diazodicarbonyl compounds with nitriles to give functionalized 1,3-oxazole derivatives in a simple one-step procedure. In particular, dimethyl diazomalonate undergoes th
Autor:
Yinghui Wu, Javed Iqbal, Mikael Bergdahl, Robert Hett, Gangloff Anthony R, Timothy L. Friebe, Paul Helquist
Publikováno v:
ChemInform. 25
The right-hand portion (3) of the type A streptogramin antibiotics was synthesized in non-racemic form through use of a Horner-Wadsworth-Emmons reaction for diene construction, an asymmetric aldol condensation, and a zinc-promoted oxazole addition re
Autor:
Emma J. Shelton, Gangloff Anthony R, David Sperandio, Rice Kenneth D, Vivian R. Wang, Joane Litvak
Publikováno v:
ChemInform. 32
Tetrabutylammonium fluoride (TBAF) was found to be a mild and efficient catalyst for the synthesis of 3,5-disubstituted-1,2,4-oxadiazoles. Using 0.1–1.0 equivalents of TBAF in THF for 1–24 h at room temperature, alkanoyl- and aroyloxyamidines wer