Zobrazeno 1 - 9
of 9
pro vyhledávání: '"Ganesh S, Jedhe"'
Autor:
Douglas N. Brawley, David B. Sauer, Jianping Li, Xuhui Zheng, Akiko Koide, Ganesh S. Jedhe, Tiffany Suwatthee, Jinmei Song, Zheng Liu, Paramjit S. Arora, Shohei Koide, Victor J. Torres, Da-Neng Wang, Nathaniel J. Traaseth
Publikováno v:
Nature Chemical Biology. 18:706-712
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::1db806ee90dc70d50dd3d48cdf5c98e2
https://doi.org/10.1038/s41589-022-00994-9
https://doi.org/10.1038/s41589-022-00994-9
Autor:
Ganesh S, Jedhe, Paramjit S, Arora
Publikováno v:
Methods in enzymology. 656
Examination of complexes of proteins with biomolecular ligands reveals that proteins tend to interact with partners via folded sub-domains, in which the backbone possesses secondary structure. α-Helices comprising the largest class of protein second
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::edaec107a1a485a28d882d403619fb4e
https://pubmed.ncbi.nlm.nih.gov/34325784
https://pubmed.ncbi.nlm.nih.gov/34325784
Autor:
Douglas N, Brawley, David B, Sauer, Jianping, Li, Xuhui, Zheng, Akiko, Koide, Ganesh S, Jedhe, Tiffany, Suwatthee, Jinmei, Song, Zheng, Liu, Paramjit S, Arora, Shohei, Koide, Victor J, Torres, Da-Neng, Wang, Nathaniel J, Traaseth
Publikováno v:
Nature chemical biology. 18(7)
Membrane protein efflux pumps confer antibiotic resistance by extruding structurally distinct compounds and lowering their intracellular concentration. Yet, there are no clinically approved drugs to inhibit efflux pumps, which would potentiate the ef
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::c7105139bc843c447e1d6358cde618a1
https://pubmed.ncbi.nlm.nih.gov/35361991
https://pubmed.ncbi.nlm.nih.gov/35361991
Autor:
Ganesh S. Jedhe, Paramjit S. Arora
Publikováno v:
Synthetic and Enzymatic Modifications of the Peptide Backbone ISBN: 9780128212530
Examination of complexes of proteins with biomolecular ligands reveals that proteins tend to interact with partners via folded sub-domains, in which the backbone possesses secondary structure. α-Helices comprising the largest class of protein second
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::35ad59321e65935f2068181f2dbc1860
https://doi.org/10.1016/bs.mie.2021.04.007
https://doi.org/10.1016/bs.mie.2021.04.007
Autor:
Dhiman Sarkar, Rachna Borkute, Ganesh S. Jedhe, Mahendra A. Wagh, Sachin B. Baravkar, Amit S. Choudhari, Gangadhar J. Sanjayan
Publikováno v:
ChemistrySelect. 3:3122-3126
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::1e5bc2b56334011be136ac2bd5d2abbc
https://doi.org/10.1002/slct.201800027
https://doi.org/10.1002/slct.201800027
Autor:
Kuruppanthara N. Vijayadas, Gangadhar J. Sanjayan, Rajesh G. Gonnade, Dinesh R. Shinde, Pattuparambil R. Rajamohanan, Ekta Sangtani, Amol S. Kotmale, Ganesh S. Jedhe
Publikováno v:
RSC Advances. 6:35328-35331
This communication describes the competition between native β-turn (C10) and 2-aminobenzenesulfonic acid (SAnt)(orthanilic acid)-based pseudo β-turn (C11) in their hybrid peptides. Solid-state crystal structure and solution-state NMR studies reveal
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::a989b096dfadce06ec81879a51e3454c
https://doi.org/10.1039/c6ra05684a
https://doi.org/10.1039/c6ra05684a
Autor:
Ernest Hamel, Sangram S. Kale, Gangadhar J. Sanjayan, Ganesh S. Jedhe, Manas Kumar Santra, Sachin N. Meshram
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 25:1982-1985
We describe the design, synthesis and SAR profiling of a series of novel combretastatin–nocodazole conjugates as potential anticancer agents. The thiophene ring in the nocodazole moiety was replaced by a substituted phenyl ring from the combretasta
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6ded0e454f758b1c07a185808c0c9725
https://doi.org/10.1016/j.bmcl.2015.03.019
https://doi.org/10.1016/j.bmcl.2015.03.019
Autor:
Ganesh S. Jedhe, Santosh Pasha, Gangadhar J. Sanjayan, Amol S. Kotmale, Pattuparambil R. Rajamohanan
Publikováno v:
Chemical communications (Cambridge, England). 52(8)
We describe herein the design, synthesis and conformational investigation of Pro-Amb (proline-3-amino-2-methoxybenzoic acid) incorporated Angiotensin II and its truncated analogues. Solution-state NMR and CD studies suggest γ-turn-like conformation
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6fe975dd7b3a1f8cc6c2cf6b97d02951
https://pubmed.ncbi.nlm.nih.gov/26660361
https://pubmed.ncbi.nlm.nih.gov/26660361
Autor:
Rajesh G. Gonnade, Debasish Paul, Ganesh S. Jedhe, Gangadhar J. Sanjayan, Ernest Hamel, Manas Kumar Santra, Tam Luong Nguyen
Publikováno v:
Bioorganicmedicinal chemistry letters. 23(16)
A series of 1,5-disubstituted tetrazole-tethered combretastatin analogues with extended hydrogen-bond donors at the ortho-positions of the aryl A and B rings were developed and evaluated for their antitubulin and antiproliferative activity. We wanted
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bdd94281c3b791edcc014905b3aaed5d
https://pubmed.ncbi.nlm.nih.gov/23809851
https://pubmed.ncbi.nlm.nih.gov/23809851