Zobrazeno 1 - 10
of 44
pro vyhledávání: '"Gaifa Lai"'
Autor:
Jay S. Fine, James Fossetta, Minglang Wu, Waldemar Gonsiorek, Carol Terminelli, Richard W. Bond, Daniel Lundell, J. Robert Merritt, Aki Cynthia J, Jianhua Chao, Zhenmin He, R. William Hipkin, James Jakway, Younong Yu, Taveras Arthur G, Diane Rindgen, Gaifa Lai, Rosemary Mayer-Ezel, Xuedong Fan, Michael P. Dwyer, Chao Jianping, Hongchen Qiu, Biju J. Purakkattle, Hong Bian
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 18:1318-1322
Comprehensive SAR studies were undertaken in the 3,4-diaminocyclobut-3-ene-1,2-dione class of CXCR2/CXCR1 receptor antagonists to explore the role of the heterocycle on chemokine receptor binding affinities, functional activity, as well as oral expos
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6b68dac44b7899c04fed455963d2ae1a
https://doi.org/10.1016/j.bmcl.2008.01.024
https://doi.org/10.1016/j.bmcl.2008.01.024
Publikováno v:
Synthetic Communications. 38:72-76
A convenient, five‐step preparation of 2‐acetyl‐4,5‐difluorothiophene from 2,3‐dibromothiophene is described.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::63a8d814cbbe6af3b3aeae5ecd31ce86
https://doi.org/10.1080/00397910701649064
https://doi.org/10.1080/00397910701649064
Autor:
Gaifa Lai
Publikováno v:
Synthetic Communications. 31:565-568
An efficient, two-step synthesis of N-benzylazetidine, starting from benzaldehyde and 3-bromopropylamine hydrobromide, is described. *Dedicated to Professor Huicai Wang on the occasion of his 70th birthday.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::293e54e5b43c55a9c3cf228af2c27019
https://doi.org/10.1081/scc-100000583
https://doi.org/10.1081/scc-100000583
Autor:
Cesar Colon, Gaifa Lai
Publikováno v:
Synthetic Communications. 29:3011-3016
A one-pot, four-step procedure was developed for the efficient preparation of (S)-benzyl 4-hydroxy-2-pentynoate (1) from (S)-3-butyn-2-ol (2), which involved as a key step the unusual lithiation of the silyl ether 5 with n-BuLi in the presence of a c
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::b4e3f7bb912d7ba0b7667eb9c21233f4
https://doi.org/10.1080/00397919908086476
https://doi.org/10.1080/00397919908086476
Autor:
Gaifa Lai, Mcallister Timothy L
Publikováno v:
Synthetic Communications. 29:409-413
A convenient, three-step preparation of (E)-3-(l-cyclohexenyl)-2-propenoic acid (1) from cyciohexanone was developed, which exploited the palladium(II) complex-catalyzed olefrnation of the triflate 3 as a key step.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::93c8907818fcb794c34b4c1c3c0d9325
https://doi.org/10.1080/00397919908085782
https://doi.org/10.1080/00397919908085782
Autor:
Gaifa Lai, Wayne K. Anderson
Publikováno v:
Synthetic Communications. 25:4087-4091
Five substituted allenic esters were prepared in good yields through the ortho ester Claisen rearrangement of primary and secondary propargyl alcohols.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::d206b3e7887aeea4f675ed3bc1c55038
https://doi.org/10.1080/00397919508011486
https://doi.org/10.1080/00397919508011486
Autor:
Gaifa Lai, Wayne K. Anderson
Publikováno v:
Synthesis. 1995:1287-1290
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::49b7344d65249754dc1b87bb77cc5f8a
https://doi.org/10.1055/s-1995-4434
https://doi.org/10.1055/s-1995-4434
Autor:
Gaifa Lai, Wayne K. Anderson
Publikováno v:
Tetrahedron Letters. 34:6849-6852
A nine-step synthesis of the benzimidazole analogue, 2 , of mycophenolic acid is reported involving both the BF 3 -Et 2 O catalysed aromatic amino- and the ortho ester Claisen rearrangements as key steps.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::d48531725abaa5d096b921cdb1669d00
https://doi.org/10.1016/s0040-4039(00)91811-2
https://doi.org/10.1016/s0040-4039(00)91811-2
Autor:
Gaifa Lai, Wayne K. Anderson
Publikováno v:
ChemInform. 25
A nine-step synthesis of the benzimidazole analogue, 2 , of mycophenolic acid is reported involving both the BF 3 -Et 2 O catalysed aromatic amino- and the ortho ester Claisen rearrangements as key steps.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::ec35e9048aa05c93fef9e58fb71f8beb
https://doi.org/10.1002/chin.199418134
https://doi.org/10.1002/chin.199418134
Autor:
Wayne K. Anderson, Gaifa Lai
Publikováno v:
ChemInform. 27
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::ec96165c2e47eb8593ad299dee23c9db
https://doi.org/10.1002/chin.199613072
https://doi.org/10.1002/chin.199613072