Zobrazeno 1 - 7
of 7
pro vyhledávání: '"Gabrielle, Brossard"'
Autor:
Rebecca M. Pruss, Claude Barberis, Jacques Simiand, Colette Lacour, D. Nisato, Gabrielle Brossard, Philippe Soubrie, Jean Wagnon, Guy Griebel, Claudine Serradeil-Le Gal, Gérard Le Fur, J P Maffrand, Marc Pascal, Bernard Scatton, Gilles Guillon
Publikováno v:
Journal of Pharmacology and Experimental Therapeutics. 300:1122-1130
(2S,4R)-1-[5-Chloro-1-[(2,4-dimethoxyphenyl)sulfonyl]-3-(2-methoxy-phenyl)-2-oxo-2,3-dihydro-1H-indol-3-yl]-4-hydroxy-N,N-dimethyl-2-pyrrolidine carboxamide (SSR149415), the first selective, nonpeptide vasopressin V1b receptor antagonist yet describe
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::58f67d43bd81433e1f53f82c12eebbf4
https://doi.org/10.1124/jpet.300.3.1122
https://doi.org/10.1124/jpet.300.3.1122
Autor:
G. Bertrand, Miguel Trueba, Ling Ling Cheng, Stoytcho Stoev, Claudine Serradeil-Le Gal, Nga Ching Wo, Gabrielle Brossard, Gilles Guillon, Maria A. Ventura, Brigitte Murat, Hazel H. Szeto, Ana Pena, Maurice Manning
Publikováno v:
Endocrinology. 148(9)
Recently, we synthesized and characterized the first selective V(1b) vasopressin (VP)/oxytocin receptor agonist, d[Cha(4)]arginine vasopressin. However, this agonist was only selective for the human receptors. We thus decided to design a selective V(
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e2e0c83be6fd4262ff0fec5867558924
https://pubmed.ncbi.nlm.nih.gov/17495006
https://pubmed.ncbi.nlm.nih.gov/17495006
Autor:
Rolf C. Gaillard, Gilles Guillon, Guy Griebel, Maurice Manning, Jacques Simiand, Sylvain Derick, Gabrielle Brossard, Claudine Serradeil-Le Gal
Publikováno v:
Stress (Amsterdam, Netherlands). 6(3)
By activating three distinct vasopressin receptor isoforms called V1a-R, V1b-R (V3-R) and V2-R, vasopressin (VP) mediates a wide number of biological effects in mammals and may be involved in several pathological states. Up to now only specific V1a a
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ac8400bbc4781876fe91cd25e363166d
https://pubmed.ncbi.nlm.nih.gov/13129813
https://pubmed.ncbi.nlm.nih.gov/13129813
Autor:
Claudine, Serradeil-Le Gal, Jean, Wagnon, Jacques, Simiand, Guy, Griebel, Colette, Lacour, Gilles, Guillon, Claude, Barberis, Gabrielle, Brossard, Philippe, Soubrié, Dino, Nisato, Marc, Pascal, Rebecca, Pruss, Bernard, Scatton, Jean-Pierre, Maffrand, Gérard, Le Fur
Publikováno v:
The Journal of pharmacology and experimental therapeutics. 300(3)
(2S,4R)-1-[5-Chloro-1-[(2,4-dimethoxyphenyl)sulfonyl]-3-(2-methoxy-phenyl)-2-oxo-2,3-dihydro-1H-indol-3-yl]-4-hydroxy-N,N-dimethyl-2-pyrrolidine carboxamide (SSR149415), the first selective, nonpeptide vasopressin V1b receptor antagonist yet describe
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::706a3b4df8cf7ddd6066ca67287cbf0e
https://pubmed.ncbi.nlm.nih.gov/11861823
https://pubmed.ncbi.nlm.nih.gov/11861823
Autor:
G. Le Fur, Danielle Raufaste, C Serradeil-Le Gal, Corinne Garcia, Claude Barberis, Lise Bankir, D Chicot, Gerard Valette, Colette Lacour, Gilles Guillon, G Galindo, Brigitte Pouzet, J P Maffrand, E. Marty, G Garcia, S Jard, Gabrielle Brossard, Loic Foulon, D. Nisato, P. Vilain
SR 121463A, a potent and selective, orally active, nonpeptide vasopressin V2 receptor antagonist, has been characterized in several in vitro and in vivo models. This compound displayed highly competitive and selective affinity for V2 receptors in rat
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fcafd48a6910b749c76f59700b5677f9
https://europepmc.org/articles/PMC507737/
https://europepmc.org/articles/PMC507737/
Autor:
Gal Claudine, Serradeil-Le, Sylvain, Derick, Gabrielle, Brossard, Maurice, Manning, Jacques, Simiand, Rolf, Gaillard, Guy, Griebel, Gilles, Guillon
Publikováno v:
Stress: The International Journal on the Biology of Stress; Sep2003, Vol. 6 Issue 3, p199-206, 8p, 1 Diagram, 1 Chart, 4 Graphs
Autor:
Brigitte Pouzet, Gérard Le Fur, Claudine Serradeil-Le Gal, Danièle Raufaste, E. Marty, Jean-Pierre Maffrand, Gabrielle Brossard
Publikováno v:
FEBS Letters. (2-3):185-191
Characterization and localization of leptin binding sites were investigated in rat kidneys using [125I]leptin as a ligand. [125I]Leptin specific binding was found in high amounts in rat renomedullary membranes. This binding was specific, saturable, t
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7884e91ada1286094f5e6bb77f6837a4