Zobrazeno 1 - 8
of 8
pro vyhledávání: '"Gábor Varró"'
Publikováno v:
Periodica Polytechnica Chemical Engineering. 67:31-40
An efficient stereoselective synthesis of a pivotal intermediate, a cyclic allyl alcohol derivative containing two methoxy groups [(±)-22], using for the preparation of (±)-trans-dihydronarciclasine analogues was elaborated starting from easily ava
Autor:
György Szabó, Olivér Éliás, Péter Erdélyi, Attila Potor, György I. Túrós, Benedek I. Károlyi, Gábor Varró, Ágnes Gy. Vaskó, Imre Bata, Gábor L. Kapus, Zoltán Dohányos, Amrita Á. Bobok, László Fodor, Márta Thán, Mónika Vastag, Zsolt Komlódi, Rita É. Soukupné Kedves, Éva Makó, Brigitta Süveges, István Greiner
Publikováno v:
Journal of Medicinal Chemistry. 65:7876-7895
Autor:
György, Szabó, Olivér, Éliás, Péter, Erdélyi, Attila, Potor, György I, Túrós, Benedek I, Károlyi, Gábor, Varró, Ágnes Gy, Vaskó, Imre, Bata, Gábor L, Kapus, Zoltán, Dohányos, Amrita Á, Bobok, László, Fodor, Márta, Thán, Mónika, Vastag, Zsolt, Komlódi, Rita É, Soukupné Kedves, Éva, Makó, Brigitta, Süveges, István, Greiner
Publikováno v:
Journal of medicinal chemistry. 65(11)
The discovery and characterization of novel naphthyridine derivatives with selective α5-GABA
Publikováno v:
Synthesis. 50:625-643
Several new trans-dihydronarciclasine analogues were stereoselectively synthesised by applying our feasible and efficient process developed recently. These new phenanthridone alkaloid derivatives were obtained in both racemic and optically active f
Publikováno v:
European journal of medicinal chemistry. 173
A series of (±)-trans-dihydronarciclasine and (±)-trans-dihydrolycoricidine derivatives with variously substituted ring A was synthesised and evaluated for their antiproliferative activity against 60 human tumour cell lines (NCI60), representing le
Publikováno v:
Monatshefte Fur Chemie
Some new trans-dihydronarciclasine derivatives containing a 1,4-benzodioxane moiety were stereoselectively synthesised using our feasible and efficient method developed recently. These new phenanthridone alkaloid analogues were obtained in both racem
Publikováno v:
Tetrahedron Letters. 57:1544-1546
A short and efficient stereoselective total synthesis of (±)-trans-dihydronarciclasine (1), a highly potent naturally occurring antineoplastic agent, was developed from readily available vanillin (7). The key intermediate of this new synthesis was a
Autor:
Alajos Grün, László Hegedűs, András Simon, István Kádas, Ibolya Leveles, Beáta G. Vértessy, Attila Balogh, Gábor Varró
Publikováno v:
Journal of natural products. 80(6)
A feasible and enantioselective total synthesis of (−)-trans-dihydronarciclasine [(−)-1], a highly biologically active alkaloid, was devised starting from vanillin (8). The key step of this new synthesis was an asymmetric, organocatalytic Michael